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7NFW
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Human 14-3-3 sigma in complex with human Estrogen Receptor alpha peptide
分子名称: 14-3-3 protein sigma, Estrogen receptor
著者Roversi, P, Falcicchio, M, Doveston, R.
登録日2021-02-08
公開日2021-02-17
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Cooperative stabilisation of 14-3-3 sigma protein-protein interactions via covalent protein modification.
Chem Sci, 12, 2021
7NIP
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BU of 7nip by Molmil
titin N2A unique sequence (UN2A) core
分子名称: Isoform 11 of Titin
著者Zhou, T, Kovermann, M, Fleming, J.R, Mayans, O.
登録日2021-02-13
公開日2021-03-03
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献Molecular Characterisation of Titin N2A and Its Binding of CARP Reveals a Titin/Actin Cross-linking Mechanism.
J.Mol.Biol., 433, 2021
7NQZ
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BU of 7nqz by Molmil
Plasmodium falciparum Hsp70-x chaperone nucleotide binding domain in complex with Z1827898537
分子名称: (3S)-N-benzylpyrrolidin-3-amine, AMP PHOSPHORAMIDATE, CHLORIDE ION, ...
著者Mohamad, N, O'Donoghue, A, Kantsadi, A.L, Vakonakis, I.
登録日2021-03-02
公開日2021-03-10
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.319 Å)
主引用文献Structures of P. falciparum Hsp70-x nucleotide binding domain with small molecule ligands
To Be Published
7NFY
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BU of 7nfy by Molmil
P1a-state of wild type human mitochondrial LONP1 protease with bound substrate protein and ATPgS
分子名称: ADENOSINE-5'-DIPHOSPHATE, Lon protease homolog, mitochondrial, ...
著者Mohammed, I, Schmitz, K.A, Schenck, N, Maier, T, Abrahams, J.P.
登録日2021-02-08
公開日2021-02-24
最終更新日2025-07-09
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Catalytic cycling of human mitochondrial Lon protease.
Structure, 30, 2022
7NG5
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P1c-state of wild type human mitochondrial LONP1 protease with bound substrate protein in presence of ATP/ADP mix
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Lon protease homolog, ...
著者Mohammed, I, Schmitz, K.A, Schenck, N, Maier, T, Abrahams, J.P.
登録日2021-02-08
公開日2021-02-24
最終更新日2025-07-09
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Catalytic cycling of human mitochondrial Lon protease.
Structure, 30, 2022
7NQR
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Plasmodium falciparum Hsp70-x chaperone nucleotide binding domain in complex with Z287256168
分子名称: (S)-N-(1-cyclopropylethyl)-6-methylpicolinamide, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, AMP PHOSPHORAMIDATE, ...
著者Mohamad, N, O'Donoghue, A, Kantsadi, A.L, Vakonakis, I.
登録日2021-03-02
公開日2021-03-10
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Structures of P. falciparum Hsp70-x nucleotide binding domain with small molecule ligands
To Be Published
7NMU
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BU of 7nmu by Molmil
Crystal structure of human platelet glycoprotein VI in complex with an inhibitory nanobody.
分子名称: CALCIUM ION, Nanobody 2, Platelet glycoprotein VI
著者Slater, A, Jonas, E, Watson, S.P.
登録日2021-02-23
公開日2021-03-10
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural characterization of a novel GPVI-nanobody complex reveals a biologically active domain-swapped GPVI dimer.
Blood, 137, 2021
7NQS
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BU of 7nqs by Molmil
Plasmodium falciparum Hsp70-x chaperone nucleotide binding domain in complex with Z1203107138
分子名称: 1-ethyl-N-[(4-fluorophenyl)methyl]-1H-pyrazole-4-carboxamide, AMP PHOSPHORAMIDATE, GLYCEROL, ...
著者Mohamad, N, O'Donoghue, A, Kantsadi, A.L, Vakonakis, I.
登録日2021-03-02
公開日2021-03-17
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Structures of P. falciparum Hsp70-x nucleotide binding domain with small molecule ligands
To Be Published
7NG4
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BU of 7ng4 by Molmil
P1b-state of wild type human mitochondrial LONP1 protease with bound endogenous substrate protein and in presence of ATP/ADP mix
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Lon protease homolog, ...
著者Mohammed, I, Schmitz, K.A, Schenck, N, Maier, T, Abrahams, J.P.
登録日2021-02-08
公開日2021-02-24
最終更新日2025-07-02
実験手法ELECTRON MICROSCOPY (4.4 Å)
主引用文献Catalytic cycling of human mitochondrial Lon protease.
Structure, 30, 2022
7NFV
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BU of 7nfv by Molmil
Structure of SARS-CoV-2 Papain-like protease PLpro
分子名称: CHLORIDE ION, GLYCEROL, PHOSPHATE ION, ...
著者Srinivasan, V, Gunther, S, Reinke, P, Werner, N, Falke, S, Brognaro, H, Ullah, N, Andaleeb, H, Perbandt, M, Alves Franca, B, Schwinzer, M, Wang, M, Sprenger, J, Lieske, J, Ginn, H, Lane, T.J, Yefanov, O, Gelisio, L, Koua, F, Saouane, S, Tolstikova, A, Groessler, M, Fleckenstein, H, Ewert, W, Trost, F, Lorenzen, K, Schubert, R, Han, H, Schmidt, C, Brings, L, Ehrt, C, Rarey, M, Galchenkova, M, Gevorkov, Y, Li, C, Perk, A, Awel, S, Hinrichs, W, Meents, A, Betzel, C.
登録日2021-02-07
公開日2021-02-24
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Antiviral activity of natural phenolic compounds in complex at an allosteric site of SARS-CoV-2 papain-like protease.
Commun Biol, 5, 2022
7NQU
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Plasmodium falciparum Hsp70-x chaperone nucleotide binding domain in complex with Z396380540
分子名称: AMP PHOSPHORAMIDATE, CHLORIDE ION, GLYCEROL, ...
著者Mohamad, N, O'Donoghue, A, Kantsadi, A.L, Vakonakis, I.
登録日2021-03-02
公開日2021-03-10
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Structures of P. falciparum Hsp70-x nucleotide binding domain with small molecule ligands
To Be Published
7NQ5
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BU of 7nq5 by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 3-(2-(benzyloxy)phenyl)-5-methyl-1H-1,2,4-triazole
分子名称: 1,2-ETHANEDIOL, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 3-methyl-5-(2-phenylmethoxyphenyl)-4~{H}-1,2,4-triazole, ...
著者Chung, C.
登録日2021-03-01
公開日2021-03-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors.
J.Med.Chem., 64, 2021
7NRS
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Conformation 1 of straight filament from primary age-related tauopathy brain
分子名称: Microtubule-associated protein tau
著者Shi, Y, Murzin, A.G, Falcon, B, Epstein, A, Machin, J, Tempest, P, Newell, K.L, Vidal, R, Garringer, H.J, Sahara, N, Higuchi, M, Ghetti, B, Jang, M, Scheres, S.H.W, Goedert, M.
登録日2021-03-04
公開日2021-03-24
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.68 Å)
主引用文献Cryo-EM structures of tau filaments from Alzheimer's disease with PET ligand APN-1607.
Acta Neuropathol, 141, 2021
7NPN
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BU of 7npn by Molmil
B-brick bare in 5 mM Mg2+
分子名称: SCAFFOLD STRAND, STAPLE STRAND
著者Bertosin, E, Stoemmer, P, Feigl, E, Wenig, M, Honemann, M, Dietz, H.
登録日2021-02-27
公開日2021-03-31
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (10.38 Å)
主引用文献Cryo-Electron Microscopy and Mass Analysis of Oligolysine-Coated DNA Nanostructures.
Acs Nano, 15, 2021
7NIO
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BU of 7nio by Molmil
Crystal structure of the SARS-CoV-2 helicase APO form
分子名称: SARS-CoV-2 helicase NSP13, ZINC ION
著者Newman, J.A, Yosaatmadja, Y, Douangamath, A, Bountra, C, Gileadi, O.
登録日2021-02-12
公開日2021-03-17
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure, mechanism and crystallographic fragment screening of the SARS-CoV-2 NSP13 helicase.
Nat Commun, 12, 2021
7NRV
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BU of 7nrv by Molmil
Paired helical filament from Alzheimer's disease with PET ligand APN-1607
分子名称: Microtubule-associated protein tau
著者Shi, Y, Murzin, A.G, Falcon, B, Epstein, A, Machin, J, Tempest, P, Newell, K.L, Vidal, R, Garringer, H.J, Sahara, N, Higuchi, M, Ghetti, B, Jang, M, Scheres, S.H.W, Goedert, M.
登録日2021-03-04
公開日2021-03-24
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Cryo-EM structures of tau filaments from Alzheimer's disease with PET ligand APN-1607.
Acta Neuropathol, 141, 2021
7NQ8
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BU of 7nq8 by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH N-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(pyridin-2-ylmethoxy)benzamide
分子名称: 1,2-ETHANEDIOL, Bromodomain-containing protein 2, N-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(pyridin-2-ylmethoxy)benzamide
著者Chung, C.W.
登録日2021-03-01
公開日2021-03-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.602 Å)
主引用文献Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors.
J.Med.Chem., 64, 2021
7NRQ
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Paired helical filament from primary age-related tauopathy brain
分子名称: Microtubule-associated protein tau
著者Shi, Y, Murzin, A.G, Falcon, B, Epstein, A, Machin, J, Tempest, P, Newell, K.L, Vidal, R, Garringer, H.J, Sahara, N, Higuchi, M, Ghetti, B, Jang, M, Scheres, S.H.W, Goedert, M.
登録日2021-03-04
公開日2021-03-24
最終更新日2025-07-09
実験手法ELECTRON MICROSCOPY (2.76 Å)
主引用文献Cryo-EM structures of tau filaments from Alzheimer's disease with PET ligand APN-1607.
Acta Neuropathol, 141, 2021
7NQI
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BU of 7nqi by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide
分子名称: 1,2-ETHANEDIOL, 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide, Bromodomain-containing protein 2
著者Chung, C.W.
登録日2021-03-01
公開日2021-03-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.603 Å)
主引用文献Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors.
J.Med.Chem., 64, 2021
7NQ9
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BU of 7nq9 by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 2-benzyl-N-cyclopropyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide
分子名称: 1,2-ETHANEDIOL, 6-benzyl-N4-((1r,3r)-3-hydroxycyclobutyl)-N2-methylpyridine-2,4-dicarboxamide, Bromodomain-containing protein 2
著者Chung, C.W.
登録日2021-03-01
公開日2021-03-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.602 Å)
主引用文献Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors.
J.Med.Chem., 64, 2021
7NQ7
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BU of 7nq7 by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH (S)-N-ethyl-3-(1-methyl-1H-1,2,3-triazol-4-yl)-4-(1-phenylethoxy)benzamide
分子名称: 1,2-ETHANEDIOL, Bromodomain-containing protein 2, ~{N}-ethyl-3-(1-methyl-1,2,3-triazol-4-yl)-4-[(1~{S})-1-phenylethoxy]benzamide
著者Chung, C.
登録日2021-03-01
公開日2021-03-24
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors.
J.Med.Chem., 64, 2021
7NRT
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Conformation 2 of straight filament from primary age-related tauopathy brain
分子名称: Microtubule-associated protein tau
著者Shi, Y, Murzin, A.G, Falcon, B, Epstein, A, Machin, J, Tempest, P, Newell, K.L, Vidal, R, Garringer, H.J, Sahara, N, Higuchi, M, Ghetti, B, Jang, M, Scheres, S.H.W, Goedert, M.
登録日2021-03-04
公開日2021-03-24
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (2.68 Å)
主引用文献Cryo-EM structures of tau filaments from Alzheimer's disease with PET ligand APN-1607.
Acta Neuropathol, 141, 2021
7NOW
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Complex of Nucleoporin-98 and nanobody MS98-27 solved at 1.85A resolution
分子名称: Anti-Nup98 nanobody MS98-27, Nuclear pore complex protein Nup98, SODIUM ION, ...
著者Sola-Colom, M, Trakhanov, S, Goerlich, D.
登録日2021-02-26
公開日2021-04-07
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A checkpoint function for Nup98 in nuclear pore formation suggested by novel inhibitory nanobodies.
Embo J., 2024
7NRX
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BU of 7nrx by Molmil
Straight filament from Alzheimer's disease with PET ligand APN-1607
分子名称: Microtubule-associated protein tau
著者Shi, Y, Murzin, A.G, Falcon, B, Epstein, A, Machin, J, Tempest, P, Newell, K.L, Vidal, R, Garringer, H.J, Sahara, N, Higuchi, M, Ghetti, B, Jang, M, Scheres, S.H.W, Goedert, M.
登録日2021-03-04
公開日2021-03-24
最終更新日2024-07-10
実験手法ELECTRON MICROSCOPY (3.55 Å)
主引用文献Cryo-EM structures of tau filaments from Alzheimer's disease with PET ligand APN-1607.
Acta Neuropathol, 141, 2021
7NN0
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Crystal structure of the SARS-CoV-2 helicase in complex with AMP-PNP
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, SARS-CoV-2 helicase NSP13, ...
著者Newman, J.A, Yosaatmadja, Y, Douangamath, A, Bountra, C, Gileadi, O.
登録日2021-02-23
公開日2021-03-24
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (3.04 Å)
主引用文献Structure, mechanism and crystallographic fragment screening of the SARS-CoV-2 NSP13 helicase.
Nat Commun, 12, 2021

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