5OWI
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![BU of 5owi by Molmil](/molmil-images/mine/5owi) | The dynamic dimer structure of the chaperone Trigger Factor (conformer 1) | 分子名称: | Trigger factor | 著者 | Morgado, L, Burmann, B.M, Sharpe, T, Mazur, A, Hiller, S. | 登録日 | 2017-09-01 | 公開日 | 2017-11-29 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | The dynamic dimer structure of the chaperone Trigger Factor. Nat Commun, 8, 2017
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6U9O
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![BU of 6u9o by Molmil](/molmil-images/mine/6u9o) | Human IMPDH2 treated with ATP, IMP, NAD+, and 2 mM GTP. Fully compressed filament segment reconstruction. | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ... | 著者 | Johnson, M.C, Kollman, J.M. | 登録日 | 2019-09-09 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.36 Å) | 主引用文献 | Cryo-EM structures demonstrate human IMPDH2 filament assembly tunes allosteric regulation. Elife, 9, 2020
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6UA5
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![BU of 6ua5 by Molmil](/molmil-images/mine/6ua5) | Human IMPDH2 treated with ATP, IMP, NAD+, and 2 mM GTP. Free interfacial octamer reconstruction. | 分子名称: | INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase 2, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Johnson, M.C, Kollman, J.M. | 登録日 | 2019-09-10 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.79 Å) | 主引用文献 | Cryo-EM structures demonstrate human IMPDH2 filament assembly tunes allosteric regulation. Elife, 9, 2020
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6UEL
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![BU of 6uel by Molmil](/molmil-images/mine/6uel) | CPS1 bound to allosteric inhibitor H3B-193 | 分子名称: | Carbamoyl-phosphate synthase [ammonia], mitochondrial, N~1~-[(4-fluorophenyl)methyl]-N~1~-methyl-N~4~-(4-methyl-1,3-thiazol-2-yl)piperidine-1,4-dicarboxamide, ... | 著者 | Larsen, N.A, Nguyen, T.V. | 登録日 | 2019-09-21 | 公開日 | 2020-03-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Small Molecule Inhibition of CPS1 Activity through an Allosteric Pocket. Cell Chem Biol, 27, 2020
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4O7V
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![BU of 4o7v by Molmil](/molmil-images/mine/4o7v) | |
6U8S
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![BU of 6u8s by Molmil](/molmil-images/mine/6u8s) | Human IMPDH2 treated with ATP, IMP, NAD+, and 2 mM GTP. Filament assembly interface reconstruction. | 分子名称: | INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase 2, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Johnson, M.C, Kollman, J.M. | 登録日 | 2019-09-05 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | Cryo-EM structures demonstrate human IMPDH2 filament assembly tunes allosteric regulation. Elife, 9, 2020
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4O7L
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![BU of 4o7l by Molmil](/molmil-images/mine/4o7l) | |
6UA2
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![BU of 6ua2 by Molmil](/molmil-images/mine/6ua2) | Human IMPDH2 treated with ATP, IMP, NAD+, and 2 mM GTP. Bent (2/4 compressed, 2/4 extended) segment reconstruction. | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ... | 著者 | Johnson, M.C, Kollman, J.M. | 登録日 | 2019-09-10 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (4.2 Å) | 主引用文献 | Cryo-EM structures demonstrate human IMPDH2 filament assembly tunes allosteric regulation. Elife, 9, 2020
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6UAJ
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![BU of 6uaj by Molmil](/molmil-images/mine/6uaj) | Human IMPDH2 treated with ATP, IMP, NAD+, and 2 mM GTP. Free canonical octamer reconstruction. | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ... | 著者 | Johnson, M.C, Kollman, J.M. | 登録日 | 2019-09-10 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.84 Å) | 主引用文献 | Cryo-EM structures demonstrate human IMPDH2 filament assembly tunes allosteric regulation. Elife, 9, 2020
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6UC2
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4O83
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![BU of 4o83 by Molmil](/molmil-images/mine/4o83) | |
5VK4
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![BU of 5vk4 by Molmil](/molmil-images/mine/5vk4) | |
4ORM
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![BU of 4orm by Molmil](/molmil-images/mine/4orm) | Crystal structure of Plasmodium falciparum dihydroorotate dehydrogenase bound with Inhibitor DSM338 (N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-5-methyl-2-(trifluoromethyl)[1,2,4]triazolo[1,5-a]pyrimidin-7-amine) | 分子名称: | Dihydroorotate dehydrogenase (quinone), mitochondrial, FLAVIN MONONUCLEOTIDE, ... | 著者 | Deng, X, Phillips, M.A. | 登録日 | 2014-02-11 | 公開日 | 2014-06-04 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.07 Å) | 主引用文献 | Fluorine Modulates Species Selectivity in the Triazolopyrimidine Class of Plasmodium falciparum Dihydroorotate Dehydrogenase Inhibitors. J.Med.Chem., 57, 2014
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4O7Z
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![BU of 4o7z by Molmil](/molmil-images/mine/4o7z) | |
4O7N
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![BU of 4o7n by Molmil](/molmil-images/mine/4o7n) | |
4O7Y
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![BU of 4o7y by Molmil](/molmil-images/mine/4o7y) | |
4OC9
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![BU of 4oc9 by Molmil](/molmil-images/mine/4oc9) | 2.35 Angstrom resolution crystal structure of putative O-acetylhomoserine (thiol)-lyase (metY) from Campylobacter jejuni subsp. jejuni NCTC 11168 with N'-Pyridoxyl-Lysine-5'-Monophosphate at position 205 | 分子名称: | GLYCEROL, IMIDAZOLE, PHOSPHATE ION, ... | 著者 | Halavaty, A.S, Brunzelle, J.S, Wawrzak, Z, Onopriyenko, O, Savchenko, A, Anderson, W.F, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2014-01-08 | 公開日 | 2014-03-12 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | 2.35 Angstrom resolution crystal structure of putative O-acetylhomoserine (thiol)-lyase (metY) from Campylobacter jejuni subsp. jejuni NCTC 11168 with N'-Pyridoxyl-Lysine-5'-Monophosphate at position 205 To be Published
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4O7T
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![BU of 4o7t by Molmil](/molmil-images/mine/4o7t) | SAICAR synthetase (Type-2) in complex with ADP, ASP and TMP | 分子名称: | ACETATE ION, ADENOSINE-5'-DIPHOSPHATE, ASPARTIC ACID, ... | 著者 | Manjunath, K, Jeyakanthan, J, Sekar, K. | 登録日 | 2013-12-26 | 公開日 | 2014-12-31 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | SAICAR synthetase (Type-2) in complex with ADP, ASP and TMP To be Published
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4O7R
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4O84
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![BU of 4o84 by Molmil](/molmil-images/mine/4o84) | |
4PAW
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![BU of 4paw by Molmil](/molmil-images/mine/4paw) | Structure of hypothetical protein HP1257. | 分子名称: | Orotate phosphoribosyltransferase, PHOSPHATE ION, THIOCYANATE ION, ... | 著者 | Battaile, K.P, Lam, R, Lam, K, Romanov, V, Jones, K, Soloveychik, M, Pai, E.F, Chirgadze, N.Y. | 登録日 | 2014-04-10 | 公開日 | 2015-05-06 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Structure of hypothetical protein HP1257. To Be Published
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4MAM
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![BU of 4mam by Molmil](/molmil-images/mine/4mam) | The crystal structure of phosphoribosylaminoimidazole carboxylase ATPase subunit of Francisella tularensis subsp. tularensis SCHU S4 in complex with an ADP analog, AMP-CP | 分子名称: | GLYCEROL, PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER, Phosphoribosylaminoimidazole carboxylase, ... | 著者 | Tan, K, Zhou, M, Kwon, K, Anderson, W.F, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2013-08-16 | 公開日 | 2013-08-28 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.474 Å) | 主引用文献 | The crystal structure of phosphoribosylaminoimidazole carboxylase ATPase subunit of Francisella tularensis subsp. tularensis SCHU S4 in complex with an ADP analog, AMP-CP To be Published
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6I1S
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![BU of 6i1s by Molmil](/molmil-images/mine/6i1s) | Crystal structure of the ACVR1 (ALK2) kinase in complex with FKBP12 and the inhibitor E6201 | 分子名称: | (4~{S},5~{R},6~{Z},9~{S},10~{S},12~{E})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione, 1,2-ETHANEDIOL, Activin receptor type-1, ... | 著者 | Williams, E.P, Pinkas, D.M, Fortin, J, Newman, J.A, Bradshaw, W.J, Mahajan, P, Kupinska, K, Burgess-Brown, N, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Bullock, A.N. | 登録日 | 2018-10-30 | 公開日 | 2019-09-11 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Mutant ACVR1 Arrests Glial Cell Differentiation to Drive Tumorigenesis in Pediatric Gliomas. Cancer Cell, 37, 2020
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5KXJ
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![BU of 5kxj by Molmil](/molmil-images/mine/5kxj) | Crystal Structure of L-Aspartate Oxidase from Salmonella typhimurium in the Complex with Substrate L-Aspartate | 分子名称: | 1,2-ETHANEDIOL, ASPARTIC ACID, GLYCEROL, ... | 著者 | Kim, Y, Osipiuk, J, Mulligan, R, Makowska-Grzyska, M, Maltseva, N, Shatsman, S, Gu, M, Anderson, W.F, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-07-20 | 公開日 | 2016-08-03 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Crystal Structure of L-Aspartate Oxidase from Salmonella typhimurium in the Complex with Substrate L-Aspartate To Be Published
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8I9O
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![BU of 8i9o by Molmil](/molmil-images/mine/8i9o) | |