5D3X
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![BU of 5d3x by Molmil](/molmil-images/mine/5d3x) | Crystal Structure of the P-Rex1 PH domain with Inositol-(1,3,4,5)-Tetrakisphosphate Bound | 分子名称: | INOSITOL-(1,3,4,5)-TETRAKISPHOSPHATE, Phosphatidylinositol 3,4,5-trisphosphate-dependent Rac exchanger 1 protein | 著者 | Cash, J.N, Tesmer, J.J.G. | 登録日 | 2015-08-06 | 公開日 | 2016-04-20 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Structural and Biochemical Characterization of the Catalytic Core of the Metastatic Factor P-Rex1 and Its Regulation by PtdIns(3,4,5)P3. Structure, 24, 2016
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5D3Y
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![BU of 5d3y by Molmil](/molmil-images/mine/5d3y) | Crystal Structure of the P-Rex1 PH domain with Inositol-(1,3,4,5)-Tetrakisphosphate Bound | 分子名称: | INOSITOL-(1,3,4,5)-TETRAKISPHOSPHATE, Phosphatidylinositol 3,4,5-trisphosphate-dependent Rac exchanger 1 protein | 著者 | Cash, J.N, Tesmer, J.J.G. | 登録日 | 2015-08-06 | 公開日 | 2016-04-20 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structural and Biochemical Characterization of the Catalytic Core of the Metastatic Factor P-Rex1 and Its Regulation by PtdIns(3,4,5)P3. Structure, 24, 2016
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3ULP
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1I3E
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![BU of 1i3e by Molmil](/molmil-images/mine/1i3e) | HUMAN AZIDO-MET HEMOGLOBIN BART'S (GAMMA4) | 分子名称: | AZIDE ION, HEMOGLOBIN GAMMA CHAINS, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Kidd, R.D, Baker, H.M, Mathews, A.J, Brittain, T, Baker, E.N. | 登録日 | 2001-02-15 | 公開日 | 2001-09-12 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Oligomerization and ligand binding in a homotetrameric hemoglobin: two high-resolution crystal structures of hemoglobin Bart's (gamma(4)), a marker for alpha-thalassemia. Protein Sci., 10, 2001
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4UWG
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![BU of 4uwg by Molmil](/molmil-images/mine/4uwg) | Discovery of (2S)-8-((3R)-3-Methylmorpholin-4-yl)-1-(3-methyl-2-oxo- butyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido(1,2-a)pyrimidin-6- one: a Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors | 分子名称: | (8S)-2-(morpholin-4-yl)-9-[2-(propan-2-yloxy)ethyl]-8-(trifluoromethyl)-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one, PHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT TYPE 3, SULFATE ION | 著者 | Pasquier, B, El-Ahmad, Y, Filoche-Romme, B, Dureuil, C, Fassy, F, Abecassis, P.Y, Mathieu, M, Bertrand, T, Benard, T, Barriere, C, ElBatti, S, Letallec, J.P, Sonnefraud, V, Brollo, M, Delbarre, L, Loyau, V, Pilorge, F, Bertin, L, Richepin, P, Arigon, J, Labrosse, J.R, Clement, J, Durand, F, Combet, R, Perraut, P, Leroy, V, Gay, F, Lefrancois, D, Bretin, F, Marquette, J.P, Michot, N, Caron, A, Castell, C, Schio, L, McCort, G, Goulaouic, H, Garcia-Echeverria, C, Ronan, B. | 登録日 | 2014-08-12 | 公開日 | 2014-11-26 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Discovery of (2S)-8-[(3R)-3-Methylmorpholin-4-Yl]-1-(3-Methyl-2-Oxobutyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido[1,2-A]Pyrimidin-6-One: A Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors. J.Med.Chem., 58, 2015
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2XYU
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![BU of 2xyu by Molmil](/molmil-images/mine/2xyu) | Crystal structure of EphA4 kinase domain in complex with VUF 12058 | 分子名称: | 5-(5-FLUORO-2-METHYLPHENYL)-6,7,8,9-TETRAHYDRO-3H-PYRAZOLO[3,4-C]ISOQUINOLIN-1-AMINE, EPHRIN TYPE-A RECEPTOR 4,, GLYCEROL | 著者 | Farenc, C.J.A, Celie, P.H.N, vanLinden, O.P.J, Siegal, G. | 登録日 | 2010-11-19 | 公開日 | 2011-11-30 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.117 Å) | 主引用文献 | Fragment Based Lead Discovery of Small Molecule Inhibitors for the Epha4 Receptor Tyrosine Kinase. Eur.J.Med.Chem., 47, 2012
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2FVF
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![BU of 2fvf by Molmil](/molmil-images/mine/2fvf) | |
6WIG
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![BU of 6wig by Molmil](/molmil-images/mine/6wig) | Structure of STENOFOLIA Protein HD domain bound with DNA | 分子名称: | DNA (5'-D(P*CP*TP*TP*GP*AP*AP*TP*AP*AP*AP*TP*CP*AP*TP*TP*AP*AP*TP*TP*TP*GP*C)-3'), DNA (5'-D(P*GP*CP*AP*AP*AP*TP*TP*AP*AP*TP*GP*AP*TP*TP*TP*AP*TP*TP*CP*AP*AP*G)-3'), STENOFOLIA | 著者 | Deng, J, Peng, S, Pathak, P. | 登録日 | 2020-04-09 | 公開日 | 2021-08-11 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure of the unique tetrameric STENOFOLIA homeodomain bound with target promoter DNA. Acta Crystallogr D Struct Biol, 77, 2021
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7YGH
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![BU of 7ygh by Molmil](/molmil-images/mine/7ygh) | |
6XWB
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![BU of 6xwb by Molmil](/molmil-images/mine/6xwb) | |
7RDB
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![BU of 7rdb by Molmil](/molmil-images/mine/7rdb) | Crystal structure of Tspan15 large extracellular loop (Tspan15 LEL) | 分子名称: | Tetraspanin-15 | 著者 | Lipper, C.H, Gabriel, K.H, Seegar, T.C.M, Durr, K.L, Tomlinson, M.G, Blacklow, S.C. | 登録日 | 2021-07-09 | 公開日 | 2021-11-03 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | Crystal structure of the Tspan15 LEL domain reveals a conserved ADAM10 binding site. Structure, 30, 2022
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7PAY
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![BU of 7pay by Molmil](/molmil-images/mine/7pay) | Structure of the human heterotetrameric cis-prenyltransferase complex in complex with magnesium and GGsPP | 分子名称: | Dehydrodolichyl diphosphate synthase complex subunit DHDDS, Dehydrodolichyl diphosphate synthase complex subunit NUS1, MAGNESIUM ION, ... | 著者 | Giladi, M, Lisnyansky Bar-El, M, Haitin, Y. | 登録日 | 2021-07-30 | 公開日 | 2022-06-01 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis for long-chain isoprenoid synthesis by cis -prenyltransferases. Sci Adv, 8, 2022
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2G70
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![BU of 2g70 by Molmil](/molmil-images/mine/2g70) | Structure of human PNMT in complex with inhibitor 3-hydroxymethyl-7-nitro-THIQ and AdoMet (SAM) | 分子名称: | PHOSPHATE ION, Phenylethanolamine N-methyltransferase, S-ADENOSYLMETHIONINE, ... | 著者 | Tyndall, J.D.A, Gee, C.L, Martin, J.L. | 登録日 | 2006-02-27 | 公開日 | 2007-02-13 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Enzyme Adaptation to Inhibitor Binding: A Cryptic Binding Site in Phenylethanolamine N-Methyltransferase J.Med.Chem., 50, 2007
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7PB0
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![BU of 7pb0 by Molmil](/molmil-images/mine/7pb0) | Structure of the human heterotetrameric cis-prenyltransferase complex in complex with magnesium, GGsPP and IsPP | 分子名称: | 3-methylbut-3-enylsulfanyl(phosphonooxy)phosphinic acid, Dehydrodolichyl diphosphate synthase complex subunit DHDDS, Dehydrodolichyl diphosphate synthase complex subunit NUS1, ... | 著者 | Giladi, M, Lisnyansky Bar-El, M, Haitin, Y. | 登録日 | 2021-07-30 | 公開日 | 2022-06-01 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.301 Å) | 主引用文献 | Structural basis for long-chain isoprenoid synthesis by cis -prenyltransferases. Sci Adv, 8, 2022
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8DSK
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![BU of 8dsk by Molmil](/molmil-images/mine/8dsk) | Structure of the N358Y variant of serine hydroxymethyltransferase 8 in complex with PLP, glycine, and formyl tetrahydrofolate | 分子名称: | 1,2-ETHANEDIOL, N-GLYCINE-[3-HYDROXY-2-METHYL-5-PHOSPHONOOXYMETHYL-PYRIDIN-4-YL-METHANE], N-[4-({[(6S)-2-amino-5-formyl-4-oxo-3,4,5,6,7,8-hexahydropteridin-6-yl]methyl}amino)benzoyl]-L-glutamic acid, ... | 著者 | Korasick, D.A, Beamer, L.J. | 登録日 | 2022-07-22 | 公開日 | 2023-10-18 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Structural and functional analysis of two SHMT8 variants associated with soybean cyst nematode resistance. Febs J., 291, 2024
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5C2I
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![BU of 5c2i by Molmil](/molmil-images/mine/5c2i) | Crystal structure of Anabaena sp. DyP-type peroxidese (AnaPX) | 分子名称: | 1,2-ETHANEDIOL, ACETIC ACID, Alr1585 protein, ... | 著者 | Yoshida, T, Amano, Y, Tsuge, H, Sugano, Y. | 登録日 | 2015-06-16 | 公開日 | 2015-12-16 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Anabaena sp. DyP-type peroxidase is a tetramer consisting of two asymmetric dimers. Proteins, 84, 2016
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4R53
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3ZZH
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![BU of 3zzh by Molmil](/molmil-images/mine/3zzh) | Crystal structure of the amino acid kinase domain from Saccharomyces cerevisiae acetylglutamate kinase in complex with its feed- back inhibitor L-arginine | 分子名称: | 1,2-ETHANEDIOL, ACETYLGLUTAMATE KINASE, ARGININE, ... | 著者 | de Cima, S, Gil-Ortiz, F, Crabeel, M, Fita, I, Rubio, V. | 登録日 | 2011-09-01 | 公開日 | 2012-05-02 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Insight on an Arginine Synthesis Metabolon from the Tetrameric Structure of Yeast Acetylglutamate Kinase Plos One, 7, 2012
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6FKU
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![BU of 6fku by Molmil](/molmil-images/mine/6fku) | Structure and function of aldehyde dehydrogenase from Thermus thermophilus: An enzyme with an evolutionarily-distinct C-terminal arm (Recombinant protein with shortened C-terminal, in complex with NADP) | 分子名称: | Aldehyde dehydrogenase, DI(HYDROXYETHYL)ETHER, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Hayes, K.A, Noor, M.R, Djeghader, A, Soulimane, T. | 登録日 | 2018-01-24 | 公開日 | 2018-09-26 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The quaternary structure of Thermus thermophilus aldehyde dehydrogenase is stabilized by an evolutionary distinct C-terminal arm extension. Sci Rep, 8, 2018
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3ZZG
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![BU of 3zzg by Molmil](/molmil-images/mine/3zzg) | Crystal structure of the amino acid kinase domain from Saccharomyces cerevisiae acetylglutamate kinase without ligands | 分子名称: | ACETYLGLUTAMATE KINASE | 著者 | de Cima, S, Gil-Ortiz, F, Crabeel, M, Fita, I, Rubio, V. | 登録日 | 2011-09-01 | 公開日 | 2012-05-02 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Insight on an Arginine Synthesis Metabolon from the Tetrameric Structure of Yeast Acetylglutamate Kinase Plos One, 7, 2012
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6VO6
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![BU of 6vo6 by Molmil](/molmil-images/mine/6vo6) | Crystal Structure of Cj1427, an Essential NAD-dependent Dehydrogenase from Campylobacter jejuni, in the Presence of NADH and GDP | 分子名称: | 1,2-ETHANEDIOL, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, CHLORIDE ION, ... | 著者 | Anderson, T.K, Spencer, K.D, Thoden, J.B, Huddleston, J.P, Raushel, F.M, Holden, H.M. | 登録日 | 2020-01-30 | 公開日 | 2020-04-01 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural Analysis of Cj1427, an Essential NAD-Dependent Dehydrogenase for the Biosynthesis of the Heptose Residues in the Capsular Polysaccharides ofCampylobacter jejuni. Biochemistry, 59, 2020
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8WBB
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![BU of 8wbb by Molmil](/molmil-images/mine/8wbb) | |
8WBE
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![BU of 8wbe by Molmil](/molmil-images/mine/8wbe) | |
8WBD
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![BU of 8wbd by Molmil](/molmil-images/mine/8wbd) | |
1I3D
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![BU of 1i3d by Molmil](/molmil-images/mine/1i3d) | HUMAN CARBONMONOXY HEMOGLOBIN BART'S (GAMMA4) | 分子名称: | CARBON MONOXIDE, HEMOGLOBIN GAMMA CHAINS, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Kidd, R.D, Baker, H.M, Mathews, A.J, Brittain, T, Baker, E.N. | 登録日 | 2001-02-15 | 公開日 | 2001-09-12 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Oligomerization and ligand binding in a homotetrameric hemoglobin: two high-resolution crystal structures of hemoglobin Bart's (gamma(4)), a marker for alpha-thalassemia. Protein Sci., 10, 2001
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