6UZ8
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![BU of 6uz8 by Molmil](/molmil-images/mine/6uz8) | Cryo-EM structure of human TRPC6 in complex with agonist AM-0883 | 分子名称: | (5-chloro-1'H-spiro[indole-3,4'-piperidin]-1'-yl)[(2R)-2,3-dihydro-1,4-benzodioxin-2-yl]methanone, 2-[[(2~{S})-2-decanoyloxy-3-dodecanoyloxy-propoxy]-oxidanyl-phosphoryl]oxyethyl-trimethyl-azanium, CHOLESTEROL HEMISUCCINATE, ... | 著者 | Bai, Y, Yu, X, Huang, X, Chen, H. | 登録日 | 2019-11-14 | 公開日 | 2020-03-18 | 実験手法 | ELECTRON MICROSCOPY (2.84 Å) | 主引用文献 | Structural basis for pharmacological modulation of the TRPC6 channel. Elife, 9, 2020
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7DXF
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![BU of 7dxf by Molmil](/molmil-images/mine/7dxf) | |
7DXG
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![BU of 7dxg by Molmil](/molmil-images/mine/7dxg) | Structure of SAR7334-bound TRPC6 at 2.9 angstrom | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 4-[[(1R,2R)-2-[(3R)-3-azanylpiperidin-1-yl]-2,3-dihydro-1H-inden-1-yl]oxy]-3-chloranyl-benzenecarbonitrile, CALCIUM ION, ... | 著者 | Chen, L, Guo, W. | 登録日 | 2021-01-18 | 公開日 | 2022-02-02 | 最終更新日 | 2024-06-05 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structural mechanism of human TRPC3 and TRPC6 channel regulation by their intracellular calcium-binding sites. Neuron, 110, 2022
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6UZA
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![BU of 6uza by Molmil](/molmil-images/mine/6uza) | Cryo-EM structure of human TRPC6 in complex with antagonist AM-1473 | 分子名称: | 2-[[(2~{S})-2-decanoyloxypropoxy]-oxidanyl-phosphoryl]oxyethyl-trimethyl-azanium, 4-({(1R,2R)-2-[(3R)-3-aminopiperidin-1-yl]-2,3-dihydro-1H-inden-1-yl}oxy)benzonitrile, CHOLESTEROL HEMISUCCINATE, ... | 著者 | Bai, Y, Yu, X, Huang, X, Chen, H. | 登録日 | 2019-11-14 | 公開日 | 2020-03-18 | 実験手法 | ELECTRON MICROSCOPY (3.08 Å) | 主引用文献 | Structural basis for pharmacological modulation of the TRPC6 channel. Elife, 9, 2020
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7A6U
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![BU of 7a6u by Molmil](/molmil-images/mine/7a6u) | Cryo-EM structure of the cytoplasmic domain of human TRPC6 | 分子名称: | Short transient receptor potential channel 6, UNKNOWN ATOM OR ION | 著者 | Grieben, M, Pike, A.C.W, Wang, D, Mukhopadhyay, S.M.M, Chalk, R, Marsden, B.D, Burgess-Brown, N.A, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Carpenter, E.P, Structural Genomics Consortium (SGC) | 登録日 | 2020-08-26 | 公開日 | 2020-09-30 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.62 Å) | 主引用文献 | Cryo-EM structure of the cytoplasmic domain of human TRPC6 TO BE PUBLISHED
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5YX9
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![BU of 5yx9 by Molmil](/molmil-images/mine/5yx9) | |