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PDB: 8 件

3GP2
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BU of 3gp2 by Molmil
Calmodulin bound to peptide from calmodulin kinase II (CaMKII)
分子名称: CALCIUM ION, Calcium/calmodulin-dependent protein kinase type II delta chain, Calmodulin
著者Ng, H.L, Alber, T.A, Wand, A.J.
登録日2009-03-20
公開日2010-04-07
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.46 Å)
主引用文献Calmodulin bound to peptide from calmodulin kinase II (CaMKII)
To be Published
7ZRQ
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BU of 7zrq by Molmil
1.68 Angstrom crystal structure of Ca/CaM-E140G:CaMKIIdelta peptide complex
分子名称: CALCIUM ION, Calcium/calmodulin-dependent protein kinase type II subunit delta, Calmodulin-1, ...
著者Helassa, N, Antonyuk, S.
登録日2022-05-04
公開日2022-12-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Calmodulin variant E140G associated with long QT syndrome impairs CaMKII delta autophosphorylation and L-type calcium channel inactivation.
J.Biol.Chem., 299, 2022
2WEL
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BU of 2wel by Molmil
Crystal structure of SU6656-bound calcium/calmodulin-dependent protein kinase II delta in complex with calmodulin
分子名称: (3Z)-N,N-DIMETHYL-2-OXO-3-(4,5,6,7-TETRAHYDRO-1H-INDOL-2-YLMETHYLIDENE)-2,3-DIHYDRO-1H-INDOLE-5-SULFONAMIDE, 1,2-ETHANEDIOL, CALCIUM ION, ...
著者Pike, A.C.W, Rellos, P, Salah, E, Burgess-Brown, N, Keates, T, Muniz, J, Sethi, R, Roos, A, Filippakopoulos, P, von Delft, F, Edwards, A, Weigelt, J, Arrowsmith, C.H, Bountra, C, Knapp, S.
登録日2009-03-31
公開日2009-04-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of the Camkiidelta/Calmodulin Complex Reveals the Molecular Mechanism of Camkii Kinase Activation.
Plos Biol., 8, 2010
5VLO
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BU of 5vlo by Molmil
The structure of human CamKII with bound inhibitor
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, Calcium/calmodulin-dependent protein kinase type II subunit delta, N-[(2S)-2-(diethylamino)propyl]-2-[(2S)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide
著者Somoza, J.R, Villasenor, A.G.
登録日2017-04-25
公開日2017-08-23
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Inhibitors of CamKII
To Be Published
6AYW
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The structure of human CamKII with bound inhibitor
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, Calcium/calmodulin-dependent protein kinase type II subunit delta, N-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide
著者Somoza, J.R, Villasenor, A.G.
登録日2017-09-08
公開日2017-11-15
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献The structure of human CamKII with bound inhibitor
To Be Published
2VN9
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BU of 2vn9 by Molmil
Crystal Structure of Human Calcium Calmodulin dependent Protein Kinase II delta isoform 1, CAMKD
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II DELTA CHAIN, CHLORIDE ION, ...
著者Roos, A.K, Rellos, P, Salah, E, Pike, A.C.W, Fedorov, O, Pilka, E.S, von Delft, F, Arrowsmith, C.H, Weigelt, J, Edwards, A, Bountra, C, Knapp, S.
登録日2008-01-31
公開日2008-02-26
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of the Camkiidelta/Calmodulin Complex Reveals the Molecular Mechanism of Camkii Kinase Activation.
Plos Biol., 8, 2010
7ZRP
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BU of 7zrp by Molmil
2.65 Angstrom crystal structure of Ca/CaM:CaMKIIdelta peptide complex
分子名称: CALCIUM ION, Calcium/calmodulin-dependent protein kinase type II subunit delta, Calmodulin-1, ...
著者Helassa, N, Antonyuk, S.
登録日2022-05-04
公開日2022-12-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Calmodulin variant E140G associated with long QT syndrome impairs CaMKII delta autophosphorylation and L-type calcium channel inactivation.
J.Biol.Chem., 299, 2022
2W2C
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BU of 2w2c by Molmil
STRUCTURE OF THE TETRADECAMERIC OLIGOMERISATION DOMAIN OF CALCIUM- CALMODULIN DEPENDENT PROTEIN KINASE II DELTA
分子名称: ACETATE ION, CADMIUM ION, CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II DELTA CHAIN
著者Pike, A.C.W, Rellos, P, Sethi, R, Salah, E, Burgess-Brown, N, Shrestha, L, Roos, A, Murray, J.W, von Delft, F, Edwards, A, Arrowsmith, C.H, Weigelt, J, Bountra, C, Knapp, S.
登録日2008-10-28
公開日2008-12-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the Camkiidelta/Calmodulin Complex Reveals the Molecular Mechanism of Camkii Kinase Activation.
Plos Biol., 8, 2010

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件を2024-08-07に公開中

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