7NTK
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7NTJ
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7X2E
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4XHV
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![BU of 4xhv by Molmil](/molmil-images/mine/4xhv) | Crystal structure of Drosophila Spinophilin-PDZ and a C-terminal peptide of Neurexin | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, LP20995p, ... | 著者 | Driller, J.H, Muhammad, K.G.H, Reddy, S, Rey, U, Boehme, M.A, Hollmann, C, Ramesh, N, Depner, H, Luetzkendorf, J, Matkovic, T, Bergeron, D, Quentin, C, Schmoranzer, J, Goettfert, F, Holt, M, Wahl, M.C, Hell, S.W, Walter, A, Sigrist, S.J, Loll, B. | 登録日 | 2015-01-06 | 公開日 | 2015-07-01 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.23 Å) | 主引用文献 | Presynaptic spinophilin tunes neurexin signalling to control active zone architecture and function. Nat Commun, 6, 2015
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6MS1
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![BU of 6ms1 by Molmil](/molmil-images/mine/6ms1) | Crystal structure of the human Scribble PDZ1 domain bound to the PDZ-binding motif of APC | 分子名称: | 1,2-ETHANEDIOL, APC C-terminus peptide, Protein scribble homolog | 著者 | How, J.Y, Kvansakul, M, Caria, S, Humbert, P.O. | 登録日 | 2018-10-16 | 公開日 | 2019-02-06 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Crystal structure of the human Scribble PDZ1 domain bound to the PDZ-binding motif of APC. FEBS Lett., 593, 2019
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6MYE
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![BU of 6mye by Molmil](/molmil-images/mine/6mye) | Crystal structure of human Scribble PDZ1 domain in complex with internal PDZ binding motif of Src homology 3 domain-containing guanine nucleotide exchange factor (SGEF) | 分子名称: | FORMIC ACID, Protein scribble homolog, Rho guanine nucleotide exchange factor 26, ... | 著者 | Sun, Y.J, Hou, T, Gakhar, L, Fuentes, E.J. | 登録日 | 2018-11-01 | 公開日 | 2019-04-10 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | SGEF forms a complex with Scribble and Dlg1 and regulates epithelial junctions and contractility. J.Cell Biol., 218, 2019
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6MYF
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6NH9
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5ZYS
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![BU of 5zys by Molmil](/molmil-images/mine/5zys) | Structure of Nephrin/MAGI1 complex | 分子名称: | Membrane-associated guanylate kinase, WW and PDZ domain-containing protein 1, Nephrin | 著者 | Weng, Z.F, Shng, Y, Zhu, J.W, Zhang, R.G. | 登録日 | 2018-05-28 | 公開日 | 2019-01-23 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Structural Basis of Highly Specific Interaction between Nephrin and MAGI1 in Slit Diaphragm Assembly and Signaling. J. Am. Soc. Nephrol., 29, 2018
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4AMH
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![BU of 4amh by Molmil](/molmil-images/mine/4amh) | Influence of circular permutation on the folding pathway of a PDZ domain | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DISKS LARGE HOMOLOG 1, GLYCEROL | 著者 | Hultqvist, G, Punekar, A.S, Chi, C.N, Selmer, M, Gianni, S, Jemth, P. | 登録日 | 2012-03-10 | 公開日 | 2012-12-05 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Tolerance of Protein Folding to a Circular Permutation in a Pdz Domain Plos One, 7, 2012
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6OV7
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6HKS
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6V84
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6AK2
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![BU of 6ak2 by Molmil](/molmil-images/mine/6ak2) | Crystal structure of the syntenin PDZ1 domain in complex with the peptide inhibitor KSL-128018 | 分子名称: | Syntenin-1, peptide inhibitor KSL-128018 | 著者 | Jin, Z.Y, Park, J.H, Yun, J.H, Haugaard-Kedstrom, L.M, Lee, W.T. | 登録日 | 2018-08-29 | 公開日 | 2019-09-04 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.868 Å) | 主引用文献 | A High-Affinity Peptide Ligand Targeting Syntenin Inhibits Glioblastoma. J.Med.Chem., 64, 2021
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6AR4
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6NID
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4YYX
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4Z33
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![BU of 4z33 by Molmil](/molmil-images/mine/4z33) | Crystal structure of the syntenin PDZ1 and PDZ2 tandem in complex with the Frizzled 7 C-terminal fragment and PIP2 | 分子名称: | ACETATE ION, D-MYO-INOSITOL-4,5-BISPHOSPHATE, GLYCEROL, ... | 著者 | Egea-Jimenez, A.L, Gallardo, R, Garcia-Pino, A, Ivarsson, Y, Wawrzyniak, A.M, Kashyap, R, Loris, R, Schymkowitz, J, Rousseau, F, Zimmermann, P. | 登録日 | 2015-03-30 | 公開日 | 2016-06-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of the syntenin PDZ1 and PDZ2 tandem in complex with the Frizzled 7 C-terminal fragment and PIP2 To Be Published
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4Z8J
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6UBH
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![BU of 6ubh by Molmil](/molmil-images/mine/6ubh) | Structure of the MM7 Erbin PDZ variant in complex with a high-affinity peptide | 分子名称: | Erbin, SODIUM ION, peptide | 著者 | Singer, A.U, Teyra, J, McLaughlin, M, Ernst, A, Sicheri, F, Sidhu, S.S. | 登録日 | 2019-09-11 | 公開日 | 2020-07-29 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Comprehensive Assessment of the Relationship Between Site -2 Specificity and Helix alpha 2 in the Erbin PDZ Domain. J.Mol.Biol., 433, 2021
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6GBD
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6GBE
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4YDP
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6BJO
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![BU of 6bjo by Molmil](/molmil-images/mine/6bjo) | PICK1 PDZ domain in complex with the small molecule inhibitor BIO124. | 分子名称: | (2S)-({4-(4-bromophenyl)-1-[1-(tert-butoxycarbonyl)-L-prolyl]piperidine-4-carbonyl}amino)(cyclopentyl)acetic acid, PRKCA-binding protein | 著者 | Marcotte, D.J. | 登録日 | 2017-11-06 | 公開日 | 2018-01-10 | 最終更新日 | 2018-02-28 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Lock and chop: A novel method for the generation of a PICK1 PDZ domain and piperidine-based inhibitor co-crystal structure. Protein Sci., 27, 2018
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6BJN
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