6AK2
Crystal structure of the syntenin PDZ1 domain in complex with the peptide inhibitor KSL-128018
Summary for 6AK2
Entry DOI | 10.2210/pdb6ak2/pdb |
Descriptor | Syntenin-1, peptide inhibitor KSL-128018 (3 entities in total) |
Functional Keywords | signaling protein, signaling protein-inhibitor complex, signaling protein/inhibitor |
Biological source | Rattus norvegicus (Rat) More |
Total number of polymer chains | 4 |
Total formula weight | 19482.44 |
Authors | Jin, Z.Y.,Park, J.H.,Yun, J.H.,Haugaard-Kedstrom, L.M.,Lee, W.T. (deposition date: 2018-08-29, release date: 2019-09-04, Last modification date: 2023-11-22) |
Primary citation | Haugaard-Kedstrom, L.M.,Clemmensen, L.S.,Sereikaite, V.,Jin, Z.,Fernandes, E.F.A.,Wind, B.,Abalde-Gil, F.,Daberger, J.,Vistrup-Parry, M.,Aguilar-Morante, D.,Leblanc, R.,Egea-Jimenez, A.L.,Albrigtsen, M.,Jensen, K.E.,Jensen, T.M.T.,Ivarsson, Y.,Vincentelli, R.,Hamerlik, P.,Andersen, J.H.,Zimmermann, P.,Lee, W.,Stromgaard, K. A High-Affinity Peptide Ligand Targeting Syntenin Inhibits Glioblastoma. J.Med.Chem., 64:1423-1434, 2021 Cited by PubMed: 33502198DOI: 10.1021/acs.jmedchem.0c00382 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.868 Å) |
Structure validation
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