Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 63 件

4O33
DownloadVisualize
BU of 4o33 by Molmil
Crystal Structure of human PGK1 3PG and terazosin(TZN) ternary complex
分子名称: 3-PHOSPHOGLYCERIC ACID, Phosphoglycerate kinase 1, [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl][(2R)-tetrahydrofuran-2-yl]methanone
著者Li, X.L, Finci, L.I, Wang, J.H.
登録日2013-12-18
公開日2014-10-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Terazosin activates Pgk1 and Hsp90 to promote stress resistance.
Nat.Chem.Biol., 11, 2015
6Y3A
DownloadVisualize
BU of 6y3a by Molmil
Structure of Plasmodium vivax phosphoglycerate kinase
分子名称: BROMIDE ION, POTASSIUM ION, Phosphoglycerate kinase
著者Blaszczyk, B.K, Hyvonen, M.
登録日2020-02-17
公開日2020-02-26
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Phosphoglycerate Kinase as a potential target for antimalarial therapy
to be published
6YJE
DownloadVisualize
BU of 6yje by Molmil
Plasmoodium vivax phosphoglycerate kinase bound to nitrofuran inhibitor from PEG3350 and ammonium acetate at pH 5.5
分子名称: (2~{S})-2-(5-nitrofuran-2-yl)-2,3,5,6,7,8-hexahydro-1~{H}-[1]benzothiolo[2,3-d]pyrimidin-4-one, Phosphoglycerate kinase
著者Blaszczyk, B.K, Hyvonen, M.
登録日2020-04-03
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献Phosphoglycerate Kinase as a potential target for antimalarial therapy
to be published
6YJF
DownloadVisualize
BU of 6yjf by Molmil
Plasmoodium vivax phosphoglycerate kinase bound to nitrofuran inhibitor from PEGSmear at pH 6.5
分子名称: (2~{S})-2-(5-nitrofuran-2-yl)-2,3,5,6,7,8-hexahydro-1~{H}-[1]benzothiolo[2,3-d]pyrimidin-4-one, GLYCEROL, Phosphoglycerate kinase
著者Hyvonen, M, Brear, P, Blaszczyk, B.K.
登録日2020-04-03
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Phosphoglycerate Kinase as a potential target for antimalarial therapy
to be published
4DG5
DownloadVisualize
BU of 4dg5 by Molmil
Crystal structure of staphylococcal Phosphoglycerate kinase
分子名称: Phosphoglycerate kinase
著者Roychowdhury, A, Mukherjee, S, Dutta, D, Das, A.K.
登録日2012-01-25
公開日2013-01-30
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure based functional analysis of Staphylococcal Phosphoglycerate kinase
To be Published
3ZLB
DownloadVisualize
BU of 3zlb by Molmil
Crystal structure of phosphoglycerate kinase from Streptococcus pneumoniae
分子名称: GLYCEROL, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
著者Bernardo-Garcia, N, Hermoso, J.A.
登録日2013-01-30
公開日2014-02-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献Pneumococcal phosphoglycerate kinase interacts with plasminogen and its tissue activator.
Thromb. Haemost., 111, 2014
4O3F
DownloadVisualize
BU of 4o3f by Molmil
Crystal Structure of mouse PGK1 3PG and terazosin(TZN) ternary complex
分子名称: 3-PHOSPHOGLYCERIC ACID, Phosphoglycerate kinase 1, [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl][(2R)-tetrahydrofuran-2-yl]methanone
著者Li, X.L, Finci, I.L, Wang, J.H.
登録日2013-12-18
公開日2014-10-29
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.106 Å)
主引用文献Terazosin activates Pgk1 and Hsp90 to promote stress resistance.
Nat.Chem.Biol., 11, 2015
3ZOZ
DownloadVisualize
BU of 3zoz by Molmil
The structure of human phosphoglycerate kinase with bound bromide, a stimulating anion.
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, BROMIDE ION, ...
著者Bowler, M.W.
登録日2013-02-26
公開日2014-03-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Identification of the Activating Anion Binding Site in Human Phosphoglycerate Kinase
To be Published
3UWD
DownloadVisualize
BU of 3uwd by Molmil
Crystal Structure of Phosphoglycerate Kinase from Bacillus Anthracis
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, MAGNESIUM ION, ...
著者Zheng, H, Chruszcz, M, Porebski, P, Kudritska, M, Grimshaw, S, Savchenko, A, Anderson, W.F, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2011-12-01
公開日2012-01-11
最終更新日2022-04-13
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Crystal structures of putative phosphoglycerate kinases from B. anthracis and C. jejuni.
J.Struct.Funct.Genom., 13, 2012
2P9T
DownloadVisualize
BU of 2p9t by Molmil
Crystal Structure of Phosphoglycerate Kinase-2 bound to 3-phosphoglycerate
分子名称: 3-PHOSPHOGLYCERIC ACID, Phosphoglycerate kinase, testis specific
著者Sawyer, G.M, Monzingo, A.F, Poteet, E.C, Robertus, J.D.
登録日2007-03-26
公開日2007-11-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-ray analysis of phosphoglycerate kinase 2, a sperm-specific isoform from Mus musculus.
Proteins, 71, 2007
4AXX
DownloadVisualize
BU of 4axx by Molmil
The catalytically active fully closed conformation of human phosphoglycerate kinase in complex with ADP 3-phosphoglycerate and beryllium trifluoride
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, BERYLLIUM TRIFLUORIDE ION, ...
著者Bowler, M.W.
登録日2012-06-15
公開日2013-06-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Catalytic Activity in the Transitions State Analogue Stabilised Conformation of a Phosphoryl Transfer Enzyme
To be Published
4EHJ
DownloadVisualize
BU of 4ehj by Molmil
An X-ray Structure of a Putative Phosphogylcerate Kinase from Francisella tularensis subsp. tularensis SCHU S4
分子名称: Phosphoglycerate kinase, SULFATE ION
著者Brunzelle, J.S, Wawrzak, Z, Skarina, T, Gordon, E, Anderson, W.F, Savchenko, A, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2012-04-02
公開日2012-05-09
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献An X-ray Structure of a Putative Phosphogylcerate Kinase from Francisella tularensis subsp. tularensis SCHU S4
To be Published
1VJD
DownloadVisualize
BU of 1vjd by Molmil
Structure of pig muscle PGK complexed with ATP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, PHOSPHATE ION, phosphoglycerate kinase
著者Flachner, B, Kovari, Z, Varga, A, Gugolya, Z, Vonderviszt, F, Naray-Szabo, G, Vas, M.
登録日2004-02-03
公開日2004-03-30
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Role of phosphate chain mobility of MgATP in completing the 3-phosphoglycerate kinase catalytic site: binding, kinetic, and crystallographic studies with ATP and MgATP.
Biochemistry, 43, 2004
4NG4
DownloadVisualize
BU of 4ng4 by Molmil
Structure of phosphoglycerate kinase (CBU_1782) from Coxiella burnetii
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Phosphoglycerate kinase
著者Franklin, M.C, Cheung, J, Rudolph, M, Cassidy, M, Gary, E, Burshteyn, F, Love, J.
登録日2013-11-01
公開日2015-06-24
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.78 Å)
主引用文献Structural genomics for drug design against the pathogen Coxiella burnetii.
Proteins, 83, 2015
1V6S
DownloadVisualize
BU of 1v6s by Molmil
Crystal Structure of Phosphoglycerate Kinase from Thermus thermophilus HB8
分子名称: GLYCEROL, Phosphoglycerate kinase, SODIUM ION
著者Mizutani, H, Kunishima, N, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2003-12-04
公開日2003-12-23
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal Structure of Phosphoglycerate Kinase from Thermus thermophilus HB8
To be Published
2P9Q
DownloadVisualize
BU of 2p9q by Molmil
Crystal Structure of Phosphoglycerate Kinase-2
分子名称: Phosphoglycerate kinase, testis specific
著者Sawyer, G.M, Monzingo, A.F, Poteet, E.C, Robertus, J.D.
登録日2007-03-26
公開日2007-11-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献X-ray analysis of phosphoglycerate kinase 2, a sperm-specific isoform from Mus musculus.
Proteins, 71, 2007
2PAA
DownloadVisualize
BU of 2paa by Molmil
Crystal structure of phosphoglycerate kinase-2 bound to atp and 3pg
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-TRIPHOSPHATE, Phosphoglycerate kinase, ...
著者Sawyer, G.M, Monzingo, A.F, Poteet, E.C, Robertus, J.D.
登録日2007-03-27
公開日2007-11-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献X-ray analysis of phosphoglycerate kinase 2, a sperm-specific isoform from Mus musculus.
Proteins, 71, 2007
1VJC
DownloadVisualize
BU of 1vjc by Molmil
Structure of pig muscle PGK complexed with MgATP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, phosphoglycerate kinase
著者Flachner, B, Kovari, Z, Varga, A, Gugolya, Z, Vonderviszt, F, Naray-Szabo, G, Vas, M.
登録日2004-02-03
公開日2004-03-30
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Role of phosphate chain mobility of MgATP in completing the 3-phosphoglycerate kinase catalytic site: binding, kinetic, and crystallographic studies with ATP and MgATP.
Biochemistry, 43, 2004
5MXM
DownloadVisualize
BU of 5mxm by Molmil
The X-ray structure of human M190I phosphoglycerate kinase 1 mutant
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, ...
著者Ilari, A, Fiorillo, A, Cipollone, A, Petrosino, M.
登録日2017-01-23
公開日2018-02-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献The phosphoglycerate kinase 1 variants found in carcinoma cells display different catalytic activity and conformational stability compared to the native enzyme.
PLoS ONE, 13, 2018
5NP8
DownloadVisualize
BU of 5np8 by Molmil
PGK1 in complex with CRT0063465 (3-[2-(4-bromophenyl)-5,7-dimethyl-pyrazolo[1,5-a]pyrimidin-6-yl]propanoic acid)
分子名称: 1,2-ETHANEDIOL, 3-PHOSPHOGLYCERIC ACID, 3-[2-(4-bromophenyl)-5,7-dimethyl-pyrazolo[1,5-a]pyrimidin-6-yl]propanoic acid, ...
著者Turnbull, A.P, Bilsland, A.E, Liu, Y, Sumpton, D, Stevenson, K, Cairney, C.J, Roffey, J, Jenkinson, D, Keith, W.N.
登録日2017-04-13
公開日2018-05-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A Novel Pyrazolopyrimidine Ligand of Human PGK1 and Stress Sensor DJ1 Modulates the Shelterin Complex and Telomere Length Regulation.
Neoplasia, 21, 2019
5M1R
DownloadVisualize
BU of 5m1r by Molmil
X-ray structure of human G166D PGK-1 mutant
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Phosphoglycerate kinase 1
著者Ilari, A, Cipollone, A, Fiorillo, A, Petrosino, M.
登録日2016-10-10
公開日2017-12-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献The phosphoglycerate kinase 1 variants found in carcinoma cells display different catalytic activity and conformational stability compared to the native enzyme.
PLoS ONE, 13, 2018
5O7D
DownloadVisualize
BU of 5o7d by Molmil
The X-ray structure of human R38M phosphoglycerate kinase 1 mutant
分子名称: ADENOSINE-5'-DIPHOSPHATE, Phosphoglycerate kinase 1
著者Ilari, A, Fiorillo, A, Cipollone, A, Petrosino, M.
登録日2017-06-08
公開日2018-06-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献The phosphoglycerate kinase 1 variants found in carcinoma cells display different catalytic activity and conformational stability compared to the native enzyme.
PLoS ONE, 13, 2018
5M6Z
DownloadVisualize
BU of 5m6z by Molmil
The X-ray structure of human M189I PGK-1 mutant in partially closed conformation
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Ilari, A, Fiorillo, A, Petrosino, M, Cipollone, A.
登録日2016-10-26
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献The phosphoglycerate kinase 1 variants found in carcinoma cells display different catalytic activity and conformational stability compared to the native enzyme.
PLoS ONE, 13, 2018
2WZB
DownloadVisualize
BU of 2wzb by Molmil
The catalytically active fully closed conformation of human phosphoglycerate kinase in complex with ADP, 3PG and magnesium trifluoride
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, ...
著者Bowler, M.W, Cliff, M.J, Marston, J.P.M, Baxter, N.J, Hownslow, A.M.H, Varga, A.V, Szabo, J, Vas, M, Blackburn, G.M, Waltho, J.P.
登録日2009-11-27
公開日2010-04-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.47 Å)
主引用文献Transition State Analogue Structures of Human Phosphoglycerate Kinase Establish the Importance of Charge Balance in Catalysis.
J.Am.Chem.Soc., 132, 2010
2WZD
DownloadVisualize
BU of 2wzd by Molmil
The catalytically active fully closed conformation of human phosphoglycerate kinase K219A mutant in complex with ADP, 3PG and aluminium trifluoride
分子名称: 3-PHOSPHOGLYCERIC ACID, ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, ...
著者Bowler, M.W, Cliff, M.J, Marston, J.P.M, Baxter, N.J, Hownslow, A.M.H, Varga, A.V, Szabo, J, Vas, M, Blackburn, G.M, Waltho, J.P.
登録日2009-11-27
公開日2010-04-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Transition State Analogue Structures of Human Phosphoglycerate Kinase Establish the Importance of Charge Balance in Catalysis.
J.Am.Chem.Soc., 132, 2010

221051

件を2024-06-12に公開中

PDB statisticsPDBj update infoContact PDBjnumon