2ETB
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2ETA
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8EKQ
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![BU of 8ekq by Molmil](/molmil-images/mine/8ekq) | Apo rat TRPV2 in nanodiscs, state 2 | 分子名称: | 1,2-DIDECANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, Transient receptor potential cation channel subfamily V member 2 | 著者 | Pumroy, R.A, Moiseenkova-Bell, V.Y. | 登録日 | 2022-09-21 | 公開日 | 2023-09-27 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.6 Å) | 主引用文献 | Functional and structural insights into activation of TRPV2 by weak acids. Embo J., 43, 2024
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8EKP
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![BU of 8ekp by Molmil](/molmil-images/mine/8ekp) | Apo rat TRPV2 in nanodiscs, state 1 | 分子名称: | 1,2-DIDECANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, Transient receptor potential cation channel subfamily V member 2 | 著者 | Pumroy, R.A, Moiseenkova-Bell, V.Y. | 登録日 | 2022-09-21 | 公開日 | 2023-09-27 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.75 Å) | 主引用文献 | Functional and structural insights into activation of TRPV2 by weak acids. Embo J., 43, 2024
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8FFM
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![BU of 8ffm by Molmil](/molmil-images/mine/8ffm) | Wildtype rat TRPV2 in nanodiscs bound to RR and 2-APB | 分子名称: | 1,2-DIDECANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, 2-aminoethyl diphenylborinate, Transient receptor potential cation channel subfamily V member 2, ... | 著者 | Pumroy, R.A, Protopopova, A.D, Rocereta, J.A, De Jesus-Perez, J.J, Fluck, E.C, Moiseenkova-Bell, V.Y. | 登録日 | 2022-12-09 | 公開日 | 2024-02-07 | 最終更新日 | 2024-02-21 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Molecular details of ruthenium red pore block in TRPV channels. Embo Rep., 25, 2024
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7ZJD
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8EKR
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![BU of 8ekr by Molmil](/molmil-images/mine/8ekr) | Apo rat TRPV2 in nanodiscs, state 3 | 分子名称: | 1,2-DIDECANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, Transient receptor potential cation channel subfamily V member 2 | 著者 | Pumroy, R.A, Moiseenkova-Bell, V.Y. | 登録日 | 2022-09-21 | 公開日 | 2023-09-27 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Functional and structural insights into activation of TRPV2 by weak acids. Embo J., 43, 2024
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7SX3
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![BU of 7sx3 by Molmil](/molmil-images/mine/7sx3) | Human NALCN-FAM155A-UNC79-UNC80 channelosome with CaM bound, conformation 1/2 | 分子名称: | (1R)-2-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL (11E)-OCTADEC-11-ENOATE, (1S)-2-{[(2-AMINOETHOXY)(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kschonsak, M, Chua, H.C, Weidling, C, Chakouri, N, Noland, C.L, Schott, K, Chang, T, Tam, C, Patel, N, Arthur, C.P, Leitner, A, Ben-Johny, M, Ciferri, C, Pless, S.A, Payandeh, J. | 登録日 | 2021-11-22 | 公開日 | 2021-12-29 | 最終更新日 | 2022-03-16 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural architecture of the human NALCN channelosome. Nature, 603, 2022
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8EKS
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2ETC
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7ZJE
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![BU of 7zje by Molmil](/molmil-images/mine/7zje) | C16-2 | 分子名称: | Transient receptor potential cation channel subfamily V member 2,Enhanced green fluorescent protein | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-10 | 公開日 | 2023-01-18 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (3.12 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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6U88
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8SLX
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8SLY
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![BU of 8sly by Molmil](/molmil-images/mine/8sly) | Rat TRPV2 bound with 2 CBD ligands in nanodiscs | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, SODIUM ION, Transient receptor potential cation channel subfamily V member 2, ... | 著者 | Tan, X, Swartz, K.J. | 登録日 | 2023-04-24 | 公開日 | 2023-05-31 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.32 Å) | 主引用文献 | Cannabidiol sensitizes TRPV2 channels to activation by 2-APB. Elife, 12, 2023
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7ZJH
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![BU of 7zjh by Molmil](/molmil-images/mine/7zjh) | TRPV2-C16+Pro-2 | 分子名称: | Transient receptor potential cation channel subfamily V member 2 | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-11 | 公開日 | 2023-01-18 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (3.39 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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6U8A
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7ZJI
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6WKN
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![BU of 6wkn by Molmil](/molmil-images/mine/6wkn) | PL-bound rat TRPV2 in nanodiscs | 分子名称: | Transient receptor potential cation channel subfamily V member 2, piperlongumine | 著者 | Pumroy, R.P, Moiseenkova-Bell, V.Y. | 登録日 | 2020-04-16 | 公開日 | 2021-04-21 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.46 Å) | 主引用文献 | Allosteric Antagonist Modulation of TRPV2 by Piperlongumine Impairs Glioblastoma Progression. Acs Cent.Sci., 7, 2021
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8FFL
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![BU of 8ffl by Molmil](/molmil-images/mine/8ffl) | Wildtype rat TRPV2 in nanodiscs bound to RR | 分子名称: | 1,2-DIDECANOYL-SN-GLYCERO-3-PHOSPHOETHANOLAMINE, Transient receptor potential cation channel subfamily V member 2 | 著者 | Pumroy, R.A, Protopopova, A.D, Rocereta, J.A, De Jesus-Perez, J.J, Fluck, E.C, Moiseenkova-Bell, V.Y. | 登録日 | 2022-12-09 | 公開日 | 2024-02-07 | 最終更新日 | 2024-02-21 | 実験手法 | ELECTRON MICROSCOPY (3.47 Å) | 主引用文献 | Molecular details of ruthenium red pore block in TRPV channels. Embo Rep., 25, 2024
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7ZJG
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![BU of 7zjg by Molmil](/molmil-images/mine/7zjg) | Probenecid | 分子名称: | Transient receptor potential cation channel subfamily V member 2 | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-11 | 公開日 | 2023-01-18 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (3.49 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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7N0M
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![BU of 7n0m by Molmil](/molmil-images/mine/7n0m) | Inactivated state of 2-APB-bound wildtype rat TRPV2 in nanodiscs | 分子名称: | 2-aminoethyl diphenylborinate, Transient receptor potential cation channel subfamily V member 2 | 著者 | Pumroy, R.A, Protopopova, A.D, Gallo, P.N, Moiseenkova-Bell, V.Y. | 登録日 | 2021-05-25 | 公開日 | 2022-05-04 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural insights into TRPV2 activation by small molecules. Nat Commun, 13, 2022
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7SX4
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![BU of 7sx4 by Molmil](/molmil-images/mine/7sx4) | Human NALCN-FAM155A-UNC79-UNC80 channelosome with CaM bound, conformation 2/2 | 分子名称: | (1R)-2-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL (11E)-OCTADEC-11-ENOATE, (1S)-2-{[(2-AMINOETHOXY)(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Kschonsak, M, Chua, H.C, Weidling, C, Chakouri, N, Noland, C.L, Schott, K, Chang, T, Tam, C, Patel, N, Arthur, C.P, Leitner, A, Ben-Johny, M, Ciferri, C, Pless, S.A, Payandeh, J. | 登録日 | 2021-11-22 | 公開日 | 2021-12-29 | 最終更新日 | 2022-03-16 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural architecture of the human NALCN channelosome. Nature, 603, 2022
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6BO5
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![BU of 6bo5 by Molmil](/molmil-images/mine/6bo5) | TRPV2 ion channel in partially closed state | 分子名称: | Transient receptor potential cation channel subfamily V member 2 | 著者 | Dosey, T.L, Wang, Z. | 登録日 | 2017-11-18 | 公開日 | 2018-12-05 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structures of TRPV2 in distinct conformations provide insight into role of the pore turret. Nat.Struct.Mol.Biol., 26, 2019
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6U84
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7T37
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![BU of 7t37 by Molmil](/molmil-images/mine/7t37) | Activated state of 2-APB and CBD-bound wildtype rat TRPV2 in nanodiscs | 分子名称: | 2-aminoethyl diphenylborinate, Transient receptor potential cation channel subfamily V member 2, cannabidiol | 著者 | Pumroy, R.A, Protopopova, A.D, Gallo, P.N, Moiseenkova-Bell, V.Y. | 登録日 | 2021-12-07 | 公開日 | 2022-05-04 | 最終更新日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structural insights into TRPV2 activation by small molecules. Nat Commun, 13, 2022
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