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4QUB
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BU of 4qub by Molmil
Caspase-3 K137A
Descriptor: ACE-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE INHIBITOR, AZIDE ION, Caspase-3
Authors:Cade, C, Swartz, P.D, MacKenzie, S.H, Clark, A.C.
Deposit date:2014-07-10
Release date:2014-11-05
Last modified:2017-11-22
Method:X-RAY DIFFRACTION (1.689 Å)
Cite:Modifying caspase-3 activity by altering allosteric networks.
Biochemistry, 53, 2014
4IYR
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BU of 4iyr by Molmil
Crystal structure of full-length caspase-6 zymogen
Descriptor: Caspase-6
Authors:Cao, Q, Wang, X.-J, Li, L.-F, Su, X.-D.
Deposit date:2013-01-29
Release date:2014-01-15
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.697 Å)
Cite:The regulatory mechanism of the caspase 6 pro-domain revealed by crystal structure and biochemical assays.
Acta Crystallogr.,Sect.D, 70, 2014
4JQY
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BU of 4jqy by Molmil
Human procaspase-3, crystal form 1
Descriptor: Procaspase-3
Authors:Thomsen, N.D, Wells, J.A.
Deposit date:2013-03-20
Release date:2013-05-08
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.495 Å)
Cite:Structural snapshots reveal distinct mechanisms of procaspase-3 and -7 activation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4JQZ
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BU of 4jqz by Molmil
Human procaspase-3, crystal form 2
Descriptor: Procaspase-3
Authors:Thomsen, N.D, Wells, J.A.
Deposit date:2013-03-20
Release date:2013-05-08
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.889 Å)
Cite:Structural snapshots reveal distinct mechanisms of procaspase-3 and -7 activation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4JJ7
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BU of 4jj7 by Molmil
Caspase-3 specific unnatural amino acid-based peptides
Descriptor: Caspase inhibitor, Caspase-8, DITHIANE DIOL
Authors:Vickers, C.J, Gonzalez-Paez, G.E, Wolan, D.W.
Deposit date:2013-03-07
Release date:2013-06-12
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.178 Å)
Cite:Selective Detection of Caspase-3 versus Caspase-7 Using Activity-Based Probes with Key Unnatural Amino Acids.
Acs Chem.Biol., 8, 2013
4JR2
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BU of 4jr2 by Molmil
Human procaspase-7/caspase-7 heterodimer bound to Ac-DEVD-CMK
Descriptor: Ac-DEVD-CMK, CHLORIDE ION, Procaspase-7
Authors:Thomsen, N.D, Wells, J.A.
Deposit date:2013-03-20
Release date:2013-05-08
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Structural snapshots reveal distinct mechanisms of procaspase-3 and -7 activation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4JJE
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BU of 4jje by Molmil
Caspase-3 specific unnatural amino acid peptides
Descriptor: Caspase inhibitor, Caspase-3
Authors:Vickers, C.J, Gonzalez-Paez, G.E, Wolan, D.W.
Deposit date:2013-03-07
Release date:2013-06-12
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.481 Å)
Cite:Selective Detection of Caspase-3 versus Caspase-7 Using Activity-Based Probes with Key Unnatural Amino Acids.
Acs Chem.Biol., 8, 2013
4JR1
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BU of 4jr1 by Molmil
Human procaspase-7 bound to Ac-DEVD-CMK
Descriptor: Ac-DEVD-CMK, CHLORIDE ION, Procaspase-7
Authors:Thomsen, N.D, Wells, J.A.
Deposit date:2013-03-20
Release date:2013-05-08
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.149 Å)
Cite:Structural snapshots reveal distinct mechanisms of procaspase-3 and -7 activation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4JB8
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BU of 4jb8 by Molmil
Caspase-7 in Complex with DARPin C7_16
Descriptor: Caspase-7 subunit p11, Caspase-7 subunit p20, DARPin C7_16
Authors:Fluetsch, A, Seeger, M.A, Gruetter, M.G.
Deposit date:2013-02-19
Release date:2013-08-21
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Design, construction, and characterization of a second-generation DARPin library with reduced hydrophobicity.
Protein Sci., 22, 2013
4JR0
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BU of 4jr0 by Molmil
Human procaspase-3 bound to Ac-DEVD-CMK
Descriptor: Ac-DEVD-CMK, CHLORIDE ION, Procaspase-3
Authors:Thomsen, N.D, Wells, J.A.
Deposit date:2013-03-20
Release date:2013-05-08
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.796 Å)
Cite:Structural snapshots reveal distinct mechanisms of procaspase-3 and -7 activation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4JJ8
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BU of 4jj8 by Molmil
Caspase-3 specific unnatural amino acid peptides
Descriptor: Caspase Inhibitor, Caspase-7
Authors:Vickers, C.J, Gonzalez-Paez, G.E, Wolan, D.W.
Deposit date:2013-03-07
Release date:2013-06-12
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.937 Å)
Cite:Selective Detection of Caspase-3 versus Caspase-7 Using Activity-Based Probes with Key Unnatural Amino Acids.
Acs Chem.Biol., 8, 2013
4HQ0
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BU of 4hq0 by Molmil
Crystal Structure of mutant form of Caspase-7
Descriptor: Caspase-7
Authors:Lee, Y, Kang, H.J, Bae, K.-H, Kim, S.J, Chung, S.J.
Deposit date:2012-10-25
Release date:2013-09-11
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structural asymmetry of procaspase-7 bound to a specific inhibitor
Acta Crystallogr.,Sect.D, 69, 2013
4HVA
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BU of 4hva by Molmil
Mechanistic and Structural Understanding of Uncompetitive Inhibitors of Caspase-6
Descriptor: Caspase-6, N-[(2R)-1-(3-cyanophenyl)-3-hydroxypropan-2-yl]-5-(3,4-dimethoxyphenyl)furan-3-carboxamide, VEID Inhibitor
Authors:Murray, J.M, Steffek, M.
Deposit date:2012-11-05
Release date:2013-03-20
Method:X-RAY DIFFRACTION (2.074 Å)
Cite:Mechanistic and structural understanding of uncompetitive inhibitors of caspase-6.
Plos One, 7, 2012
6BFJ
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BU of 6bfj by Molmil
Caspase-3 Mutant - T245D,S249D
Descriptor: AZIDE ION, Ac-Asp-Glu-Val-Asp-CMK, Caspase-3
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-26
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.543 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
5IAB
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BU of 5iab by Molmil
Caspase 3 V266D
Descriptor: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ACE-ASP-GLU-VAL-ASK, Caspase-3
Authors:Maciag, J.J, Mackenzie, S.H, Tucker, M.B, Schipper, J.L, Swartz, P.D, Clark, A.C.
Deposit date:2016-02-21
Release date:2016-10-26
Method:X-RAY DIFFRACTION (1.79 Å)
Cite:Tunable allosteric library of caspase-3 identifies coupling between conserved water molecules and conformational selection.
Proc.Natl.Acad.Sci.USA, 113, 2016
5IC6
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BU of 5ic6 by Molmil
Crystal structure of caspase-7 DEVE peptide complex
Descriptor: Caspase-7 subunit p11, Caspase-7 subunit p20, DEVE peptide
Authors:Seaman, J.E, Julien, O, Lee, P.S, Rettenmaier, T.J, Thomsen, N.D, Wells, J.A.
Deposit date:2016-02-22
Release date:2016-07-20
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Cacidases: caspases can cleave after aspartate, glutamate and phosphoserine residues.
Cell Death Differ., 23, 2016
5IAR
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BU of 5iar by Molmil
Caspase 3 V266W
Descriptor: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ACE-ASP-GLU-VAL-ASK, Caspase-3, ...
Authors:Maciag, J.J, Mackenzie, S.H, Tucker, M.B, Schipper, J.L, Swartz, P.D, Clark, A.C.
Deposit date:2016-02-21
Release date:2016-10-26
Method:X-RAY DIFFRACTION (1.76 Å)
Cite:Tunable allosteric library of caspase-3 identifies coupling between conserved water molecules and conformational selection.
Proc.Natl.Acad.Sci.USA, 113, 2016
5I9T
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BU of 5i9t by Molmil
Caspase 3 V266C
Descriptor: ACE-ASP-GLU-VAL-ASK, ACETATE ION, Caspase-3
Authors:Maciag, J.J, Mackenzie, S.H, Tucker, M.B, Schipper, J.L, Swartz, P.D, Clark, A.C.
Deposit date:2016-02-20
Release date:2016-10-26
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Tunable allosteric library of caspase-3 identifies coupling between conserved water molecules and conformational selection.
Proc.Natl.Acad.Sci.USA, 113, 2016
6BG0
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BU of 6bg0 by Molmil
Caspase-3 Mutant - D9A,D28A,S150D
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3, ...
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-27
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (2.125 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BFL
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BU of 6bfl by Molmil
Caspase-3 Mutant- D9A,D28A,T245D
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-26
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.87 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BFO
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BU of 6bfo by Molmil
Caspase-3 Mutant- T245D
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, Caspase-3, ...
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-26
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.54 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BG4
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BU of 6bg4 by Molmil
Caspase-3 Mutant- T152D
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, AZIDE ION, CHLORIDE ION, ...
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-27
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.87 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BDV
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BU of 6bdv by Molmil
Crystal structure of Caspase 3 S150A
Descriptor: AZIDE ION, Acetyl-Asp-Glu-Val-Asp-CMK, CHLORIDE ION, ...
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-24
Release date:2018-02-14
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.938 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BG1
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BU of 6bg1 by Molmil
Caspase-3 Mutant - D9A,D28A,S150E
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, Caspase-3, SODIUM ION
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-27
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.88 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018
6BFK
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BU of 6bfk by Molmil
Caspase-3 Mutant- T245A
Descriptor: AC-ASP-GLU-VAL-ASP-CMK, Caspase-3, SODIUM ION
Authors:Thomas, M.E, Grinshpon, R, Swartz, P.D, Clark, A.C.
Deposit date:2017-10-26
Release date:2018-02-21
Last modified:2018-04-25
Method:X-RAY DIFFRACTION (1.753 Å)
Cite:Modifications to a common phosphorylation network provide individualized control in caspases.
J. Biol. Chem., 293, 2018

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