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PDB: 102 件

1SWV
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Crystal structure of the D12A mutant of phosphonoacetaldehyde hydrolase complexed with magnesium
分子名称: MAGNESIUM ION, phosphonoacetaldehyde hydrolase
著者Zhang, G, Morais, M.C, Dai, J, Zhang, W, Dunaway-Mariano, D, Allen, K.N.
登録日2004-03-30
公開日2004-10-05
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Investigation of metal ion binding in phosphonoacetaldehyde hydrolase identifies sequence markers for metal-activated enzymes of the HAD enzyme superfamily
Biochemistry, 43, 2004
1SWW
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Crystal structure of the phosphonoacetaldehyde hydrolase D12A mutant complexed with magnesium and substrate phosphonoacetaldehyde
分子名称: MAGNESIUM ION, PHOSPHONOACETALDEHYDE, phosphonoacetaldehyde hydrolase
著者Zhang, G, Morais, M.C, Dai, J, Zhang, W, Dunaway-Mariano, D, Allen, K.N.
登録日2004-03-30
公開日2004-10-05
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Investigation of metal ion binding in phosphonoacetaldehyde hydrolase identifies sequence markers for metal-activated enzymes of the HAD enzyme superfamily
Biochemistry, 43, 2004
1OQD
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Crystal structure of sTALL-1 and BCMA
分子名称: Tumor necrosis factor ligand superfamily member 13B, soluble form, Tumor necrosis factor receptor superfamily member 17
著者Zhang, G.
登録日2003-03-07
公開日2003-05-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Ligand-receptor binding revealed by the TNF family member TALL-1.
Nature, 423, 2003
1OQE
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Crystal structure of sTALL-1 with BAFF-R
分子名称: Tumor necrosis factor ligand superfamily member 13B, soluble form, Tumor necrosis factor receptor superfamily member 13C
著者Zhang, G.
登録日2003-03-07
公開日2003-05-13
最終更新日2018-01-31
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Ligand-receptor binding revealed by the TNF family member TALL-1.
Nature, 423, 2003
1HSJ
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SARR MBP FUSION STRUCTURE
分子名称: FUSION PROTEIN CONSISTING OF STAPHYLOCOCCUS ACCESSORY REGULATOR PROTEIN R AND MALTOSE BINDING PROTEIN, alpha-D-glucopyranose
著者Zhang, G.
登録日2000-12-26
公開日2001-06-06
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of the SarR protein from Staphylococcus aureus.
Proc.Natl.Acad.Sci.USA, 98, 2001
1PTQ
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PROTEIN KINASE C DELTA CYS2 DOMAIN
分子名称: PROTEIN KINASE C DELTA TYPE, ZINC ION
著者Zhang, G, Hurley, J.H.
登録日1995-05-11
公開日1995-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of the cys2 activator-binding domain of protein kinase C delta in complex with phorbol ester.
Cell(Cambridge,Mass.), 81, 1995
1PTR
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PROTEIN KINASE C DELTA CYS2 DOMAIN COMPLEXED WITH PHORBOL-13-ACETATE
分子名称: 13-ACETYLPHORBOL, PROTEIN KINASE C DELTA TYPE, ZINC ION
著者Zhang, G, Hurley, J.H.
登録日1995-05-11
公開日1995-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of the cys2 activator-binding domain of protein kinase C delta in complex with phorbol ester.
Cell(Cambridge,Mass.), 81, 1995
1ZOL
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native beta-PGM
分子名称: MAGNESIUM ION, beta-phosphoglucomutase
著者Zhang, G, Tremblay, L.W, Dai, J, Wang, L, Dunaway-Mariano, D, Allen, K.N.
登録日2005-05-13
公開日2005-08-30
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Catalytic cycling in beta-phosphoglucomutase: a kinetic and structural analysis
Biochemistry, 44, 2005
2LSP
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solution structures of BRD4 second bromodomain with NF-kB-K310ac peptide
分子名称: Bromodomain-containing protein 4, NF-kB-K310ac peptide
著者Zhang, G, Liu, R, Zhong, Y, Plotnikov, A.N, Zhang, W, Rusinova, E, Gerona-Nevarro, G, Moshkina, N, Joshua, J, Chuang, P.Y, Ohlmeyer, M, He, J, Zhou, M.-M.
登録日2012-05-03
公開日2012-07-18
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Down-regulation of NF-kappa B transcriptional activity in HIV-associated kidney disease by BRD4 inhibition.
J.Biol.Chem., 287, 2012
2P5B
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The complex structure of JMJD2A and trimethylated H3K36 peptide
分子名称: FE (II) ION, Histone H3, JmjC domain-containing histone demethylation protein 3A, ...
著者Zhang, G, Chen, Z, Zang, J, Hong, X, Shi, Y.
登録日2007-03-14
公開日2007-06-12
最終更新日2013-11-27
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Structural basis of the recognition of a methylated histone tail by JMJD2A.
Proc.Natl.Acad.Sci.USA, 104, 2007
1AB8
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RAT TYPE II ADENYLYL CYCLASE C2 DOMAIN/FORSKOLIN COMPLEX
分子名称: ADENYLYL CYCLASE, FORSKOLIN
著者Zhang, G, Hurley, J.H.
登録日1997-02-04
公開日1997-05-15
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of the adenylyl cyclase catalytic core.
Nature, 386, 1997
1BDF
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STRUCTURE OF ESCHERICHIA COLI RNA POLYMERASE ALPHA SUBUNIT N-TERMINAL DOMAIN
分子名称: RNA POLYMERASE ALPHA SUBUNIT
著者Zhang, G, Darst, S.A.
登録日1998-05-08
公開日1999-05-11
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure of the Escherichia coli RNA polymerase alpha subunit amino-terminal domain.
Science, 281, 1998
7F0X
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A SARS-CoV-2 neutralizing antibody
分子名称: Antibody, Spike protein S1
著者Zhang, G, Li, X, Guo, Y, Wang, Y, Yuan, S.
登録日2021-06-07
公開日2022-06-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A SARS-CoV-2 neutralizing antibody
To Be Published
7F12
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A SARS-CoV-2 neutralizing antibody
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody, Spike protein S1
著者Zhang, G, Li, X, Guo, Y, Wang, Y, Yuan, S.
登録日2021-06-07
公開日2022-06-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献A SARS-CoV-2 neutralizing antibody
To Be Published
7F15
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A SARS-CoV-2 neutralizing antibody
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Antibody, Spike protein S1
著者Zhang, G, Li, X, Guo, Y, Wang, Y, Yuan, S.
登録日2021-06-07
公開日2022-06-15
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献A SARS-CoV-2 neutralizing antibody
To Be Published
4KEG
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Crystal Structure of MBP Fused Human SPLUNC1
分子名称: MAGNESIUM ION, Maltose-binding periplasmic/Palate lung and nasal epithelium clone fusion protein, octyl beta-D-glucopyranoside
著者Ning, F, Wang, C, Niu, L, Chu, H.W, Zhang, G.
登録日2013-04-25
公開日2014-04-30
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Lipid Ligands of the SPLUNC1 Protein
To be Published
5HRJ
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Crystal structure of the scavenger receptor cysteine-rich domain 5 (SRCR5) from porcine CD163
分子名称: Scavenger receptor cysteine-rich type 1 protein M130
著者Ma, H, Jiang, L, Qiao, S, Zhang, G, Li, R.
登録日2016-01-23
公開日2017-07-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of the scavenger receptor cysteine-rich domain 5 (SRCR5) from porcine CD163
To Be Published
2YIQ
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Structural analysis of checkpoint kinase 2 in complex with inhibitor PV1322
分子名称: (E)-5-(1-(2-CARBAMIMIDOYLHYDRAZONO)ETHYL)-N-(1H-INDOL-6-YL)-1H-INDOLE-2-CARBOXAMIDE, NITRATE ION, SERINE/THREONINE-PROTEIN KINASE CHK2
著者Lountos, G.T, Jobson, A.G, Tropea, J.E, Self, C, Zhang, G, Pommier, Y, Shoemaker, R.H, Waugh, D.S.
登録日2011-05-16
公開日2011-09-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献X-Ray Structures of Checkpoint Kinase 2 in Complex with Inhibitors that Target its Gatekeeper-Dependent Hydrophobic Pocket.
FEBS Lett., 585, 2011
2W7X
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Cellular inhibition of checkpoint kinase 2 and potentiation of cytotoxic drugs by novel Chk2 inhibitor PV1019
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, N-[4-[(E)-N-carbamimidamido-C-methyl-carbonimidoyl]phenyl]-7-nitro-1H-indole-2-carboxamide, ...
著者Jobson, A.G, Lountos, G.T, Lorenzi, P.L, Llamas, J, Connelly, J, Tropea, J.E, Onda, A, Kondapaka, S, Zhang, G, Caplen, N.J, Caredellina, J.H, Monks, A, Self, C, Waugh, D.S, Shoemaker, R.H, Pommier, Y.
登録日2009-01-06
公開日2009-09-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Cellular Inhibition of Chk2 Kinase and Potentiation of Camptothecins and Radiation by the Novel Chk2 Inhibitor Pv1019.
J.Pharmacol.Exp.Ther., 331, 2009
6R8I
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PP4R3A EVH1 domain bound to FxxP motif
分子名称: SER-LEU-PRO-PHE-THR-PHE-LYS-VAL-PRO-ALA-PRO-PRO-PRO-SER-LEU-PRO-PRO-SER, Serine/threonine-protein phosphatase 4 regulatory subunit 3A
著者Ueki, Y, Kruse, T, Weisser, M.B, Sundell, G.N, Yoo Larsen, M.S, Lopez Mendez, B, Jenkins, N.P, Garvanska, D.H, Cressey, L, Zhang, G, Davey, N, Montoya, G, Ivarsson, Y, Kettenbach, A, Nilsson, J.
登録日2019-04-02
公開日2019-10-16
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.517 Å)
主引用文献A Consensus Binding Motif for the PP4 Protein Phosphatase.
Mol.Cell, 76, 2019
6K0L
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The crystal structure of simian CD163 SRCR5
分子名称: Scavenger receptor cysteine-rich type 1 protein M130
著者Ma, H, Li, R, Jiang, L, Qiao, S, Zhang, G.
登録日2019-05-07
公開日2020-05-13
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Structural comparison of CD163 SRCR5 from different species sheds some light on its involvement in porcine reproductive and respiratory syndrome virus-2 infection in vitro.
Vet Res, 52, 2021
1FEZ
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THE CRYSTAL STRUCTURE OF BACILLUS CEREUS PHOSPHONOACETALDEHYDE HYDROLASE COMPLEXED WITH TUNGSTATE, A PRODUCT ANALOG
分子名称: MAGNESIUM ION, PHOSPHONOACETALDEHYDE HYDROLASE, TUNGSTATE(VI)ION
著者Morais, M.C, Zhang, W, Baker, A.S, Zhang, G, Dunaway-Mariano, D, Allen, K.N.
登録日2000-07-24
公開日2000-10-04
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The crystal structure of bacillus cereus phosphonoacetaldehyde hydrolase: insight into catalysis of phosphorus bond cleavage and catalytic diversification within the HAD enzyme superfamily.
Biochemistry, 39, 2000
1RQL
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Crystal Structure of Phosponoacetaldehyde Hydrolase Complexed with Magnesium and the Inhibitor Vinyl Sulfonate
分子名称: MAGNESIUM ION, Phosphonoacetaldehyde Hydrolase, VINYLSULPHONIC ACID
著者Morais, M.C, Zhang, G, Zhang, W, Olsen, D.B, Dunaway-Mariano, D, Allen, K.N.
登録日2003-12-05
公開日2004-04-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献X-ray crystallographic and site-directed mutagenesis analysis of the mechanism of Schiff-base formation in phosphonoacetaldehyde hydrolase catalysis
J.Biol.Chem., 279, 2004
1RQN
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Phosphonoacetaldehyde hydrolase complexed with magnesium
分子名称: MAGNESIUM ION, Phosphonoacetaldehyde Hydrolase
著者Morais, M.C, Zhang, G, Zhang, W, Olsen, D.B, Dunaway-Mariano, D, Allen, K.N.
登録日2003-12-05
公開日2004-04-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献X-ray crystallographic and site-directed mutagenesis analysis of the mechanism of Schiff-base formation in phosphonoacetaldehyde hydrolase catalysis
J.Biol.Chem., 279, 2004
2YCR
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Crystal structure of checkpoint kinase 2 in complex with inhibitor PV976
分子名称: 1,3-BIS{4-[(1E)-N-(4,5-DIHYDRO-1H-IMIDAZOL-2-YL)ETHANEHYDRAZONOYL]PHENYL}UREA, NITRATE ION, SERINE/THREONINE-PROTEIN KINASE CHK2
著者Lountos, G.T, Jobson, A.G, Tropea, J.E, Self, C.R, Pommier, Y, Shoemaker, R.H, Zhang, G, Waugh, D.S.
登録日2011-03-16
公開日2011-11-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Characterization of Inhibitor Complexes with Checkpoint Kinase 2 (Chk2), a Drug Target for Cancer Therapy.
J.Struct.Biol., 176, 2011

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