3UD1
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3UD2
| Crystal structure of Selenomethionine ZU5A-ZU5B protein domains of human erythrocyte ankyrin | 分子名称: | Ankyrin-1, CHLORIDE ION, ETHANOL, ... | 著者 | Yasunaga, M, Ipsaro, J.J, Mondragon, A. | 登録日 | 2011-10-27 | 公開日 | 2012-02-22 | 最終更新日 | 2019-12-25 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Structurally Similar but Functionally Diverse ZU5 Domains in Human Erythrocyte Ankyrin. J.Mol.Biol., 417, 2012
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7XRZ
| Crystal structure of BRIL and SRP2070_Fab complex | 分子名称: | IGG HEAVY CHAIN, IGG LIGHT CHAIN, Soluble cytochrome b562 | 著者 | Suzuki, M, Miyagi, H, Yasunaga, M, Asada, H, Iwata, S, Saito, J. | 登録日 | 2022-05-12 | 公開日 | 2023-05-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural insight into an anti-BRIL Fab as a G-protein-coupled receptor crystallization chaperone. Acta Crystallogr D Struct Biol, 79, 2023
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8GNG
| Crystal structure of human adenosine A2A receptor in complex with istradefylline. | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 8-[(~{E})-2-(3,4-dimethoxyphenyl)ethenyl]-1,3-diethyl-7-methyl-purine-2,6-dione, Adenosine receptor A2a, ... | 著者 | Suzuki, M, Saito, J, Miyagi, H, Yasunaga, M. | 登録日 | 2022-08-23 | 公開日 | 2023-03-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | In Vitro Pharmacological Profile of KW-6356, a Novel Adenosine A 2A Receptor Antagonist/Inverse Agonist. Mol.Pharmacol., 103, 2023
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8GNE
| Crystal structure of human adenosine A2A receptor in complex with an insurmountable inverse agonist, KW-6356. | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, Adenosine receptor A2a,Soluble cytochrome b562, ... | 著者 | Suzuki, M, Saito, J, Miyagi, H, Yasunaga, M. | 登録日 | 2022-08-23 | 公開日 | 2023-03-22 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | In Vitro Pharmacological Profile of KW-6356, a Novel Adenosine A 2A Receptor Antagonist/Inverse Agonist. Mol.Pharmacol., 103, 2023
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7C6A
| Crystal structure of AT2R-BRIL and SRP2070_Fab complex | 分子名称: | IgG Light Chain, IgG heavy chain, SAR1, ... | 著者 | Suzuki, M, Miyagi, H, Asada, H, Yasunaga, M, Suno, C, Takahashi, Y, Saito, J, Iwata, S. | 登録日 | 2020-05-21 | 公開日 | 2020-07-29 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | The discovery of a new antibody for BRIL-fused GPCR structure determination. Sci Rep, 10, 2020
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7CMM
| Crystal structure of TEAD1-YBD in complex with K-975 | 分子名称: | N-[3-(4-chloranylphenoxy)-4-methyl-phenyl]propanamide, Transcriptional enhancer factor TEF-1 | 著者 | Tsuji, Y, Suzuki, M, Yasunaga, M, Hamguchi, K, Saito, J. | 登録日 | 2020-07-28 | 公開日 | 2021-02-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesothelioma. Am J Cancer Res, 10, 2020
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7C61
| Crystal structure of 5-HT1B-BRIL and SRP2070_Fab complex | 分子名称: | 5-hydroxytryptamine receptor 1B,Soluble cytochrome b562,5-hydroxytryptamine receptor 1B, Ergotamine, IGG HEAVY CHAIN, ... | 著者 | Suzuki, M, Miyagi, H, Asada, H, Yasunaga, M, Suno, C, Takahashi, Y, Saito, J, Iwata, S. | 登録日 | 2020-05-21 | 公開日 | 2020-07-29 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The discovery of a new antibody for BRIL-fused GPCR structure determination. Sci Rep, 10, 2020
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