6U1Q
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![BU of 6u1q by Molmil](/molmil-images/mine/6u1q) | Crystal Structure of VpsO (VC0937) Kinase domain | Descriptor: | O-PHOSPHOTYROSINE, VpsO | Authors: | Tripathi, S.M, Schwechheimer, C, Herbert, K, Porcella, M.E, Brown, E.R, Yildiz, F.H, Rubin, S.M. | Deposit date: | 2019-08-16 | Release date: | 2020-08-19 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (2.87 Å) | Cite: | A tyrosine phosphoregulatory system controls exopolysaccharide biosynthesis and biofilm formation in Vibrio cholerae. Plos Pathog., 16, 2020
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6U1P
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![BU of 6u1p by Molmil](/molmil-images/mine/6u1p) | Crystal structure of VpsU (VC0916) from Vibrio cholerae | Descriptor: | GLYCEROL, Low molecular weight phosphotyrosine protein phosphatase | Authors: | Tripathi, S.M, Schwechheimer, C, Herbert, K, Osorio, J, Yildiz, F.H, Rubin, S.M. | Deposit date: | 2019-08-16 | Release date: | 2020-08-19 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (2.201 Å) | Cite: | A tyrosine phosphoregulatory system controls exopolysaccharide biosynthesis and biofilm formation in Vibrio cholerae. Plos Pathog., 16, 2020
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8CUR
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![BU of 8cur by Molmil](/molmil-images/mine/8cur) | Crystal structure of Cdk2 in complex with Cyclin A inhibitor 6-[(E)-2-(4-chlorophenyl)ethenyl]-2-{[(2R)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Descriptor: | 6-[(E)-2-(4-chlorophenyl)ethenyl]-2-{[(2R)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid, Cyclin-dependent kinase 2 | Authors: | Tripathi, S.M, Tambo, C.S, Kiss, G, Rubin, S.M. | Deposit date: | 2022-05-17 | Release date: | 2023-04-05 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Biolayer Interferometry Assay for Cyclin-Dependent Kinase-Cyclin Association Reveals Diverse Effects of Cdk2 Inhibitors on Cyclin Binding Kinetics. Acs Chem.Biol., 18, 2023
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2VOJ
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![BU of 2voj by Molmil](/molmil-images/mine/2voj) | Ternary complex of M. tuberculosis Rv2780 with NAD and pyruvate | Descriptor: | (2S)-2-HYDROXYPROPANOIC ACID, ALANINE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | Authors: | Tripathi, S.M, Ramachandran, R. | Deposit date: | 2008-02-18 | Release date: | 2008-03-04 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Crystal Structures of the Mycobacterium Tuberculosis Secretory Antigen Alanine Dehydrogenase (Rv2780) in Apo and Ternary Complex Forms Captures "Open" and "Closed" Enzyme Conformations. Proteins: Struct., Funct., Bioinf., 72, 2008
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2VOE
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![BU of 2voe by Molmil](/molmil-images/mine/2voe) | Crystal structure of Rv2780 from M. tuberculosis H37Rv | Descriptor: | ALANINE DEHYDROGENASE | Authors: | Tripathi, S.M, Ramachandran, R. | Deposit date: | 2008-02-17 | Release date: | 2008-03-04 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Crystal Structures of the Mycobacterium Tuberculosis Secretory Antigen Alanine Dehydrogenase (Rv2780) in Apo and Ternary Complex Forms Captures "Open" and "Closed" Enzyme Conformations. Proteins, 72, 2008
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2CJH
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![BU of 2cjh by Molmil](/molmil-images/mine/2cjh) | |
2CIN
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![BU of 2cin by Molmil](/molmil-images/mine/2cin) | |
2CJD
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![BU of 2cjd by Molmil](/molmil-images/mine/2cjd) | |
2CJG
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![BU of 2cjg by Molmil](/molmil-images/mine/2cjg) | Lysine aminotransferase from M. tuberculosis in bound PMP form | Descriptor: | 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, L-LYSINE-EPSILON AMINOTRANSFERASE | Authors: | Tripathi, S.M, Ramachandran, R. | Deposit date: | 2006-04-01 | Release date: | 2006-08-14 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Direct Evidence for a Glutamate Switch Necessary for Substrate Recognition: Crystal Structures of Lysine Epsilon-Aminotransferase (Rv3290C) from Mycobacterium Tuberculosis H37Rv. J.Mol.Biol., 362, 2006
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2JJH
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![BU of 2jjh by Molmil](/molmil-images/mine/2jjh) | E243 mutant of M. tuberculosis Rv3290C | Descriptor: | 2-OXOGLUTARIC ACID, L-LYSINE EPSILON AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE | Authors: | Tripathi, S.M, Ramachandran, R. | Deposit date: | 2008-04-04 | Release date: | 2009-06-30 | Last modified: | 2020-01-15 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Mutational Analysis of Mycobacterium Tuberculosis Lysine Epsilon-Aminotransferase and Inhibitor Co-Crystal Structures, Reveals Distinct Binding Modes. Biochem.Biophys.Res.Commun., 463, 2015
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2JJE
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2JJG
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2JJF
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![BU of 2jjf by Molmil](/molmil-images/mine/2jjf) | N328A mutant of M. tuberculosis Rv3290c | Descriptor: | L-LYSINE EPSILON AMINOTRANSFERASE | Authors: | tripathi, S.M, Ramachandran, R. | Deposit date: | 2008-04-04 | Release date: | 2009-06-30 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Mutational Analysis of Mycobacterium Tuberculosis Lysine Epsilon-Aminotransferase and Inhibitor Co-Crystal Structures, Reveals Distinct Binding Modes. Biochem.Biophys.Res.Commun., 463, 2015
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4JWU
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![BU of 4jwu by Molmil](/molmil-images/mine/4jwu) | Crystal structure of Cytochrome P450cam-putidaredoxin complex | Descriptor: | 1,1'-hexane-1,6-diyldipyrrolidine-2,5-dione, CALCIUM ION, Camphor 5-monooxygenase, ... | Authors: | Tripathi, S.M, Li, H, Poulos, T.L. | Deposit date: | 2013-03-27 | Release date: | 2013-06-19 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Structural basis for effector control and redox partner recognition in cytochrome P450. Science, 340, 2013
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4JX1
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![BU of 4jx1 by Molmil](/molmil-images/mine/4jx1) | Crystal structure of reduced Cytochrome P450cam-putidaredoxin complex bound to camphor and 5-exo-hydroxycamphor | Descriptor: | 1,1'-hexane-1,6-diyldipyrrolidine-2,5-dione, 5-EXO-HYDROXYCAMPHOR, CALCIUM ION, ... | Authors: | Tripathi, S.M, Li, H, Poulos, T.L. | Deposit date: | 2013-03-27 | Release date: | 2013-06-19 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.087 Å) | Cite: | Structural basis for effector control and redox partner recognition in cytochrome P450. Science, 340, 2013
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4JWS
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![BU of 4jws by Molmil](/molmil-images/mine/4jws) | Crystal structure of Cytochrome P450cam-putidaredoxin complex | Descriptor: | 1,1'-hexane-1,6-diyldipyrrolidine-2,5-dione, CALCIUM ION, Camphor 5-monooxygenase, ... | Authors: | Tripathi, S.M, Li, H, Poulos, T.L. | Deposit date: | 2013-03-27 | Release date: | 2013-06-19 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.15 Å) | Cite: | Structural basis for effector control and redox partner recognition in cytochrome P450. Science, 340, 2013
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4IMH
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![BU of 4imh by Molmil](/molmil-images/mine/4imh) | |
6CPB
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7N40
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![BU of 7n40 by Molmil](/molmil-images/mine/7n40) | Crystal structure of LIN9-RbAp48-LIN37, a MuvB subcomplex | Descriptor: | Histone-binding protein RBBP4, Isoform 2 of Protein lin-9 homolog, Protein lin-37 homolog | Authors: | Asthana, A, Ramanan, P, Tripathi, S.M, Rubin, S.M. | Deposit date: | 2021-06-02 | Release date: | 2022-02-09 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.55 Å) | Cite: | The MuvB complex binds and stabilizes nucleosomes downstream of the transcription start site of cell-cycle dependent genes. Nat Commun, 13, 2022
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6NBL
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![BU of 6nbl by Molmil](/molmil-images/mine/6nbl) | Cytochrome P450cam-putidaredoxin complex bound to camphor and cyanide | Descriptor: | 1,1'-hexane-1,6-diyldipyrrolidine-2,5-dione, CALCIUM ION, CAMPHOR, ... | Authors: | Follmer, A.H, Tripathi, S.M, Poulos, T.L. | Deposit date: | 2018-12-07 | Release date: | 2019-03-06 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (2.15 Å) | Cite: | Ligand and Redox Partner Binding Generates a New Conformational State in Cytochrome P450cam (CYP101A1). J. Am. Chem. Soc., 141, 2019
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6P8F
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![BU of 6p8f by Molmil](/molmil-images/mine/6p8f) | Crystal structure of CDK4 in complex with CyclinD1 and P27 | Descriptor: | Cyclin-dependent kinase 4, Cyclin-dependent kinase inhibitor 1B, G1/S-specific cyclin-D1 | Authors: | Guiley, K.Z, Stevenson, J.W, Lou, K, Barkovich, K.J, Bunch, K, Tripathi, S.M, Shokat, K.M, Rubin, S.M. | Deposit date: | 2019-06-07 | Release date: | 2019-12-25 | Method: | X-RAY DIFFRACTION (2.89 Å) | Cite: | p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition. Science, 366, 2019
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6P8H
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![BU of 6p8h by Molmil](/molmil-images/mine/6p8h) | Crystal structure of CDK4 in complex with CyclinD1 and P21 | Descriptor: | Cyclin-dependent kinase 4, Cyclin-dependent kinase inhibitor 1, G1/S-specific cyclin-D1 | Authors: | Guiley, K.Z, Stevenson, J.W, Lou, K, Barkovich, K.J, Bunch, K, Tripathi, S.M, Shokat, K.M, Rubin, S.M. | Deposit date: | 2019-06-07 | Release date: | 2019-12-25 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (3.19 Å) | Cite: | p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition. Science, 366, 2019
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6P8G
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![BU of 6p8g by Molmil](/molmil-images/mine/6p8g) | Crystal structure of CDK4 in complex with CyclinD1 and P27 | Descriptor: | Cyclin-dependent kinase 4, Cyclin-dependent kinase inhibitor 1B, G1/S-specific cyclin-D1 | Authors: | Guiley, K.Z, Stevenson, J.W, Lou, K, Barkovich, K.J, Bunch, K, Tripathi, S.M, Shokat, K.M, Rubin, S.M. | Deposit date: | 2019-06-07 | Release date: | 2019-12-25 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition. Science, 366, 2019
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6P8E
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![BU of 6p8e by Molmil](/molmil-images/mine/6p8e) | Crystal structure of CDK4 in complex with CyclinD1 and P27 | Descriptor: | Cyclin-dependent kinase 4, Cyclin-dependent kinase inhibitor 1B, G1/S-specific cyclin-D1, ... | Authors: | Guiley, K.Z, Stevenson, J.W, Lou, K, Barkovich, K.J, Bunch, K, Tripathi, S.M, Shokat, K.M, Rubin, S.M. | Deposit date: | 2019-06-07 | Release date: | 2019-12-25 | Last modified: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | p27 allosterically activates cyclin-dependent kinase 4 and antagonizes palbociclib inhibition. Science, 366, 2019
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7MJ9
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![BU of 7mj9 by Molmil](/molmil-images/mine/7mj9) | HLA-A*02:01 bound to Neuroblastoma Derived mutant IGFBPL1 peptide | Descriptor: | Beta-2-microglobulin, Insulin-like growth factor-binding protein-like 1 altered peptide, MHC class I antigen | Authors: | Toor, J.S, Tripathi, S.M, Truong, H.V, Yarmarkovich, M, Maris, J.M, Sgourakis, N.G. | Deposit date: | 2021-04-19 | Release date: | 2021-08-18 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | Cross-HLA targeting of intracellular oncoproteins with peptide-centric CARs. Nature, 599, 2021
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