8Q1A
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![BU of 8q1a by Molmil](/molmil-images/mine/8q1a) | The Crystal Structure of Human Carbonic Anhydrase IX in Complex with inhibitor | Descriptor: | 1,1,3-tris(oxidanylidene)-2-pentyl-1,2-benzothiazole-6-sulfonamide, Carbonic anhydrase 9, GLYCEROL, ... | Authors: | Leitans, J, Tars, K. | Deposit date: | 2023-07-31 | Release date: | 2023-11-08 | Last modified: | 2023-12-06 | Method: | X-RAY DIFFRACTION (2.35 Å) | Cite: | Structural Basis of Saccharin Derivative Inhibition of Carbonic Anhydrase IX. Chemmedchem, 18, 2023
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6TL6
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![BU of 6tl6 by Molmil](/molmil-images/mine/6tl6) | |
6TL5
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![BU of 6tl5 by Molmil](/molmil-images/mine/6tl5) | |
7SQN
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![BU of 7sqn by Molmil](/molmil-images/mine/7sqn) | |
7MWT
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![BU of 7mwt by Molmil](/molmil-images/mine/7mwt) | |
7MWU
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![BU of 7mwu by Molmil](/molmil-images/mine/7mwu) | |
7MWV
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![BU of 7mwv by Molmil](/molmil-images/mine/7mwv) | |
6WPU
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![BU of 6wpu by Molmil](/molmil-images/mine/6wpu) | |
6X0H
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![BU of 6x0h by Molmil](/molmil-images/mine/6x0h) | |
6X0J
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![BU of 6x0j by Molmil](/molmil-images/mine/6x0j) | |
6X0I
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![BU of 6x0i by Molmil](/molmil-images/mine/6x0i) | |
5KOX
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![BU of 5kox by Molmil](/molmil-images/mine/5kox) | |
8TCV
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![BU of 8tcv by Molmil](/molmil-images/mine/8tcv) | Structure of PYCR1 complexed with 4-bromobenzene-1,3-dicarboxylic acid | Descriptor: | 4-bromobenzene-1,3-dicarboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | Authors: | Tanner, J.J, Meeks, K.R. | Deposit date: | 2023-07-02 | Release date: | 2024-03-06 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.74 Å) | Cite: | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCZ
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![BU of 8tcz by Molmil](/molmil-images/mine/8tcz) | |
8TCW
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![BU of 8tcw by Molmil](/molmil-images/mine/8tcw) | |
6XP1
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![BU of 6xp1 by Molmil](/molmil-images/mine/6xp1) | |
8TCX
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![BU of 8tcx by Molmil](/molmil-images/mine/8tcx) | Structure of PYCR1 complexed with 2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carboxylic acid | Descriptor: | 2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | Authors: | Tanner, J.J, Meeks, K.R. | Deposit date: | 2023-07-02 | Release date: | 2024-03-06 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.72 Å) | Cite: | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TD0
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![BU of 8td0 by Molmil](/molmil-images/mine/8td0) | Structure of PYCR1 complexed with 5-oxo-7a-phenyl-hexahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylic acid | Descriptor: | (3R,4S,7aR)-5-oxo-7a-phenylhexahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylic acid, Pyrroline-5-carboxylate reductase 1, mitochondrial, ... | Authors: | Tanner, J.J, Meeks, K.R. | Deposit date: | 2023-07-02 | Release date: | 2024-03-06 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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8TCU
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![BU of 8tcu by Molmil](/molmil-images/mine/8tcu) | |
8TD1
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![BU of 8td1 by Molmil](/molmil-images/mine/8td1) | |
8TCY
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![BU of 8tcy by Molmil](/molmil-images/mine/8tcy) | Structure of PYCR1 complexed with 7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid | Descriptor: | 7-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid, DI(HYDROXYETHYL)ETHER, Pyrroline-5-carboxylate reductase 1, ... | Authors: | Tanner, J.J, Meeks, K.R. | Deposit date: | 2023-07-02 | Release date: | 2024-03-06 | Last modified: | 2024-03-20 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography. J.Chem.Inf.Model., 64, 2024
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6X9D
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![BU of 6x9d by Molmil](/molmil-images/mine/6x9d) | |
7STE
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![BU of 7ste by Molmil](/molmil-images/mine/7ste) | Rad24-RFC ADP state | Descriptor: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Checkpoint protein RAD24, ... | Authors: | Castaneda, J.C, Schrecker, M, Remus, D, Hite, R.K. | Deposit date: | 2021-11-12 | Release date: | 2022-04-06 | Last modified: | 2024-06-05 | Method: | ELECTRON MICROSCOPY (2.73 Å) | Cite: | Mechanisms of loading and release of the 9-1-1 checkpoint clamp. Nat.Struct.Mol.Biol., 29, 2022
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6XP2
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![BU of 6xp2 by Molmil](/molmil-images/mine/6xp2) | |
6X9C
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![BU of 6x9c by Molmil](/molmil-images/mine/6x9c) | |