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PDB: 9 results

1C72
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BU of 1c72 by Molmil
TYR115, GLN165 AND TRP209 CONTRIBUTE TO THE 1,2-EPOXY-3-(P-NITROPHENOXY)PROPANE CONJUGATING ACTIVITIES OF GLUTATHIONE S-TRANSFERASE CGSTM1-1
Descriptor: 1-HYDROXY-2-S-GLUTATHIONYL-3-PARA-NITROPHENOXY-PROPANE, PROTEIN (GLUTATHIONE S-TRANSFERASE)
Authors:Chern, M.K, Wu, T.C, Hsieh, C.H, Chou, C.C, Liu, L.F, Kuan, I.C, Yeh, Y.H, Hsiao, C.D, Tam, M.F.
Deposit date:2000-02-02
Release date:2000-08-30
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Tyr115, gln165 and trp209 contribute to the 1, 2-epoxy-3-(p-nitrophenoxy)propane-conjugating activity of glutathione S-transferase cGSTM1-1.
J.Mol.Biol., 300, 2000
3BM9
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Discovery of Benzisoxazoles as Potent Inhibitors of Chaperone Hsp90
Descriptor: 4-bromo-6-(6-hydroxy-1,2-benzisoxazol-3-yl)benzene-1,3-diol, Heat shock protein HSP 90-alpha
Authors:Gopalsamy, A, Shi, M, Vogan, E.M, Golas, J, Jacob, J, Johnson, J, Lee, F, Nilakantan, R, Peterson, R, Svenson, K, Tam, M.S, Wen, Y, Chopra, R, Ellingboe, J, Arndt, K, Boschelli, F.
Deposit date:2007-12-12
Release date:2008-07-08
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Discovery of benzisoxazoles as potent inhibitors of chaperone heat shock protein 90.
J.Med.Chem., 51, 2008
3BMY
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Discovery of Benzisoxazoles as Potent Inhibitors of Chaperone Hsp90
Descriptor: 4-chloro-6-{5-[(2-morpholin-4-ylethyl)amino]-1,2-benzisoxazol-3-yl}benzene-1,3-diol, Heat shock protein HSP 90-alpha
Authors:Gopalsamy, A, Shi, M, Vogan, E.M, Golas, J, Jacob, J, Johnson, J, Lee, F, Nilakantan, R, Peterson, R, Svenson, K, Tam, M.S, Wen, Y, Chopra, R, Ellingboe, J, Arndt, K, Boschelli, F.
Deposit date:2007-12-13
Release date:2008-07-08
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Discovery of benzisoxazoles as potent inhibitors of chaperone heat shock protein 90.
J.Med.Chem., 51, 2008
1GSU
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BU of 1gsu by Molmil
AN AVIAN CLASS-MU GLUTATHIONE S-TRANSFERASE, CGSTM1-1 AT 1.94 ANGSTROM RESOLUTION
Descriptor: CLASS-MU GLUTATHIONE S-TRANSFERASE, S-HEXYLGLUTATHIONE
Authors:Sun, Y.-J, Kuan, C, Tam, M.F, Hsiao, C.-D.
Deposit date:1997-09-02
Release date:1998-03-04
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.94 Å)
Cite:The three-dimensional structure of an avian class-mu glutathione S-transferase, cGSTM1-1 at 1.94 A resolution.
J.Mol.Biol., 278, 1998
4QCI
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BU of 4qci by Molmil
PDGF-B blocking antibody bound to PDGF-BB
Descriptor: Platelet-derived growth factor subunit B, anti-PDGF-BB antibody - Light Chain, anti-PDGF-BB antibody - Heavy chain
Authors:Kuai, J, Mosyak, L, Tam, M, LaVallie, E, Pullen, N, Carven, G.
Deposit date:2014-05-12
Release date:2015-03-11
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Characterization of Binding Mode of Action of a Blocking Anti-Platelet-Derived Growth Factor (PDGF)-B Monoclonal Antibody, MOR8457, Reveals Conformational Flexibility and Avidity Needed for PDGF-BB To Bind PDGF Receptor-beta.
Biochemistry, 54, 2015
1VF1
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BU of 1vf1 by Molmil
cGSTA1-1 in complex with glutathione
Descriptor: GLUTATHIONE, Glutathione S-transferase 3
Authors:Lin, S.C, Lo, Y.C, Tam, M.F, Liaw, Y.C.
Deposit date:2004-04-07
Release date:2005-08-23
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.77 Å)
Cite:Crystal structures of chicken glutathione S-transferase A1-1
To be Published
1VF3
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BU of 1vf3 by Molmil
cGSTA1-1 in complex with glutathione conjugate of CDNB
Descriptor: ACETIC ACID, GLUTATHIONE S-(2,4 DINITROBENZENE), Glutathione S-transferase 3
Authors:Lin, S.C, Lo, Y.C, Tam, M.F, Liaw, Y.C.
Deposit date:2004-04-07
Release date:2005-08-23
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Crystal structures of chicken glutathione S-transferase A1-1
To be Published
1VF4
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BU of 1vf4 by Molmil
cGSTA1-1 apo form
Descriptor: ACETIC ACID, Glutathione S-transferase 3
Authors:Lin, S.C, Lo, Y.C, Tam, M.F, Liaw, Y.C.
Deposit date:2004-04-08
Release date:2005-08-23
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:Crystal structures of chicken glutathione S-transferase A1-1
To be Published
1VF2
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cGSTA1-1 in complex with S-hexyl-glutathione
Descriptor: Glutathione S-transferase 3, S-HEXYLGLUTATHIONE, ZINC ION
Authors:Lin, S.C, Lo, Y.C, Tam, M.F, Liaw, Y.C.
Deposit date:2004-04-07
Release date:2005-08-23
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Crystal structures of chicken glutathione S-transferase A1-1
To be Published

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