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PDB: 184 results

2RNF
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BU of 2rnf by Molmil
X-RAY CRYSTAL STRUCTURE OF HUMAN RIBONUCLEASE 4 IN COMPLEX WITH D(UP)
Descriptor: 2'-DEOXYURIDINE 3'-MONOPHOSPHATE, RIBONUCLEASE 4
Authors:Terzyan, S.S, Peracaula, R, De Llorens, R, Tsushima, Y, Yamada, H, Seno, M, Gomis-Ruth, F.X, Coll, M.
Deposit date:1998-11-03
Release date:1999-11-10
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:The three-dimensional structure of human RNase 4, unliganded and complexed with d(Up), reveals the basis for its uridine selectivity.
J.Mol.Biol., 285, 1999
3VOV
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Crystal Structure of ROK Hexokinase from Thermus thermophilus
Descriptor: GLYCEROL, Glucokinase, ZINC ION
Authors:Nakamura, T, Kashima, Y, Mine, S, Oku, T, Uegaki, K.
Deposit date:2012-02-21
Release date:2012-06-27
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.02 Å)
Cite:Characterization and crystal structure of the thermophilic ROK hexokinase from Thermus thermophilus
J.Biosci.Bioeng., 2012
7Q5X
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BU of 7q5x by Molmil
HIF PROLYL HYDROXYLASE 2 (PHD2/EGLN1) IN COMPLEX WITH 2-OXOGLUTARATE (2OG) AND HIF-2 ALPHA CODD (523-542)
Descriptor: 2-OXOGLUTARIC ACID, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Figg Jr, W.D, McDonough, M.A, Chowdhury, R, Nakashima, Y, Schofield, C.J.
Deposit date:2021-11-04
Release date:2022-11-16
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.21 Å)
Cite:Structural basis for binding of the renal carcinoma target hypoxia-inducible factor 2 alpha to prolyl hydroxylase domain 2.
Proteins, 91, 2023
7W9Q
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Crystal structure of V30M-TTR in complex with naringenin derivative-14
Descriptor: (2~{R})-2-(3-chloranyl-4-oxidanyl-phenyl)-5,7-bis(oxidanyl)-2,3-dihydrochromen-4-one, CALCIUM ION, Transthyretin
Authors:Katayama, W, Shimane, A, Nabeshima, Y, Yokoyama, T, Mizuguchi, M.
Deposit date:2021-12-10
Release date:2022-12-14
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (1.599 Å)
Cite:Chlorinated Naringenin Analogues as Potential Inhibitors of Transthyretin Amyloidogenesis.
J.Med.Chem., 65, 2022
7W9R
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Crystal structure of V30M-TTR in complex with naringenin derivative-18
Descriptor: (2~{R})-2-[3,5-bis(chloranyl)-4-oxidanyl-phenyl]-5,7-bis(oxidanyl)-2,3-dihydrochromen-4-one, Transthyretin
Authors:Katayama, W, Shimane, A, Nabeshima, Y, Yokoyama, T, Mizuguchi, M.
Deposit date:2021-12-10
Release date:2022-12-14
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (1.997 Å)
Cite:Chlorinated Naringenin Analogues as Potential Inhibitors of Transthyretin Amyloidogenesis.
J.Med.Chem., 65, 2022
7Q5V
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HIF PROLYL HYDROXYLASE 2 (PHD2/EGLN1) IN COMPLEX WITH N-OXALYLGLYCINE (NOG) AND HIF-2 ALPHA CODD (523-542)
Descriptor: CHLORIDE ION, DI(HYDROXYETHYL)ETHER, Egl nine homolog 1, ...
Authors:Figg Jr, W.D, McDonough, M.A, Chowdhury, R, Nakashima, Y, Schofield, C.J.
Deposit date:2021-11-04
Release date:2022-11-16
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.17 Å)
Cite:Structural basis for binding of the renal carcinoma target hypoxia-inducible factor 2 alpha to prolyl hydroxylase domain 2.
Proteins, 91, 2023
2MLQ
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Human CCR2 Membrane-Proximal C-Terminal Region (PRO-C) in a frount bound form
Descriptor: MCP-1 receptor
Authors:Esaki, K, Yoshinaga, S, Tsuji, T, Toda, E, Terashima, Y, Saitoh, T, Kohda, D, Kohno, T, Osawa, M, Ueda, T, Shimada, I, Matsushima, K, Terasawa, H.
Deposit date:2014-03-04
Release date:2014-10-08
Last modified:2024-05-15
Method:SOLUTION NMR
Cite:Structural basis for the binding of the membrane-proximal C-terminal region of chemokine receptor CCR2 with the cytosolic regulator FROUNT.
Febs J., 281, 2014
1A0A
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BU of 1a0a by Molmil
PHOSPHATE SYSTEM POSITIVE REGULATORY PROTEIN PHO4/DNA COMPLEX
Descriptor: DNA (5'-D(*CP*TP*AP*GP*TP*CP*CP*CP*AP*CP*GP*TP*GP*TP*GP*AP*G )-3'), DNA (5'-D(*CP*TP*CP*AP*CP*AP*CP*GP*TP*GP*GP*GP*AP*CP*TP*AP*G )-3'), PROTEIN (PHOSPHATE SYSTEM POSITIVE REGULATORY PROTEIN PHO4)
Authors:Shimizu, T, Toumoto, A, Ihara, K, Shimizu, M, Kyogoku, Y, Ogawa, N, Oshima, Y, Hakoshima, T.
Deposit date:1997-11-27
Release date:1998-03-18
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Crystal structure of PHO4 bHLH domain-DNA complex: flanking base recognition.
EMBO J., 16, 1997
1EWV
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BU of 1ewv by Molmil
CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 LIGAND FREE FORM II
Descriptor: METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1
Authors:Kunishima, N, Shimada, Y, Tsuji, Y, Jingami, H, Morikawa, K.
Deposit date:2000-04-27
Release date:2000-12-18
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (4 Å)
Cite:Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor.
Nature, 407, 2000
4TWY
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BU of 4twy by Molmil
Structure of SARS-3CL protease complex with a phenylbenzoyl (S,R)-N-decalin type inhibitor
Descriptor: (2S)-2-({[(3S,4aR,8aS)-2-(biphenyl-4-ylcarbonyl)decahydroisoquinolin-3-yl]methyl}amino)-3-(1H-imidazol-5-yl)propanal, 3C-like proteinase
Authors:Akaji, K, Teruya, K, Shimamoto, Y, Sanjho, A, Yamashita, E, Nakagawa, A.
Deposit date:2014-07-02
Release date:2015-02-18
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Fused-ring structure of decahydroisoquinolin as a novel scaffold for SARS 3CL protease inhibitors
Bioorg.Med.Chem., 23, 2015
2MLO
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BU of 2mlo by Molmil
Human CCR2 Membrane-Proximal C-Terminal Region (PRO-C) in a Membrane bound form
Descriptor: MCP-1 receptor
Authors:Esaki, K, Yoshinaga, S, Tsuji, T, Toda, E, Terashima, Y, Saitoh, T, Kohda, D, Kohno, T, Osawa, M, Ueda, T, Shimada, I, Matsushima, K, Terasawa, H.
Deposit date:2014-03-04
Release date:2014-10-08
Last modified:2024-05-15
Method:SOLUTION NMR
Cite:Structural basis for the binding of the membrane-proximal C-terminal region of chemokine receptor CCR2 with the cytosolic regulator FROUNT.
Febs J., 281, 2014
1EWK
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BU of 1ewk by Molmil
CRYSTAL STRUCTURE OF METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 1 COMPLEXED WITH GLUTAMATE
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLUTAMIC ACID, ...
Authors:Kunishima, N, Shimada, Y, Jingami, H, Morikawa, K.
Deposit date:2000-04-26
Release date:2000-12-18
Last modified:2020-07-29
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor.
Nature, 407, 2000
7FFC
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BU of 7ffc by Molmil
Diarylpentanoid-producing polyketide synthase (A210E mutant)
Descriptor: GLYCEROL, Type III polyketide synthase
Authors:Morita, H, Wong, C.P, Liu, Q, Kodama, T, Lee, Y, Nakashima, Y.
Deposit date:2021-07-23
Release date:2022-01-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.61 Å)
Cite:Identification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood.
Nat Commun, 13, 2022
5X9S
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BU of 5x9s by Molmil
Crystal structure of fully modified H-Ras-GppNHp
Descriptor: CALCIUM ION, GTPase HRas, MAGNESIUM ION, ...
Authors:Matsumoto, S, Ke, H, Murashima, Y, Taniguchi-Tamura, H, Miyamoto, R, Yoshikawa, Y, Kumasaka, T, Mizohata, E, Edamatsu, H, Kataoka, T.
Deposit date:2017-03-09
Release date:2017-08-30
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural basis for intramolecular interaction of post-translationally modified H-RasGTP prepared by protein ligation
FEBS Lett., 591, 2017
5H0Q
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BU of 5h0q by Molmil
Crystal structure of lipid binding protein Nakanori at 1.5A
Descriptor: Lipid binding protein
Authors:Makino, A, Abe, M, Ishitsuka, R, Murate, M, Kishimoto, T, Sakai, S, Hullin-Matsuda, F, Shimada, Y, Inaba, T, Miyatake, H, Tanaka, H, Kurahashi, A, Pack, C.G, Kasai, R.S, Kubo, S, Schieber, N.L, Dohmae, N, Tochio, N, Hagiwara, K, Sasaki, Y, Aida, Y, Fujimori, F, Kigawa, T, Nishikori, K, Parton, R.G, Kusumi, A, Sako, Y, Anderluh, G, Yamashita, M, Kobayashi, T, Greimel, P, Kobayashi, T.
Deposit date:2016-10-06
Release date:2016-10-19
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (1.501 Å)
Cite:A novel sphingomyelin/cholesterol domain-specific probe reveals the dynamics of the membrane domains during virus release and in Niemann-Pick type C
FASEB J., 31, 2017
6ZBO
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BU of 6zbo by Molmil
HIF Prolyl Hydroxylase 2 (PHD2/EGLN1) in Complex with 1-(6-morpholinopyrimidin-4-yl)-4-(1H-1,2,3-triazol-1-yl)-1H-pyrazol-5-ol (Molidustat)
Descriptor: 2-(6-morpholin-4-ylpyrimidin-4-yl)-4-(1,2,3-triazol-1-yl)pyrazol-3-ol, CHLORIDE ION, Egl nine homolog 1, ...
Authors:Figg Jr, W.D, McDonough, M.A, Nakashima, Y, Holt-Martyn, J.P, Schofield, C.J.
Deposit date:2020-06-08
Release date:2021-04-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (1.79 Å)
Cite:Structural Basis of Prolyl Hydroxylase Domain Inhibition by Molidustat.
Chemmedchem, 16, 2021
6ZBN
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BU of 6zbn by Molmil
HIF Prolyl Hydroxylase 2 (PHD2/EGLN1) in complex with tert-butyl 6-(5-hydroxy-4-(1H-1,2,3-triazol-1-yl)-1H-pyrazol-1-yl)nicotinate (IOX4)
Descriptor: Egl nine homolog 1, GLYCEROL, MANGANESE (II) ION, ...
Authors:Figg Jr, W.D, McDonough, M.A, Nakashima, Y, Schofield, C.J.
Deposit date:2020-06-08
Release date:2021-04-07
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (2.01 Å)
Cite:Structural Basis of Prolyl Hydroxylase Domain Inhibition by Molidustat.
Chemmedchem, 16, 2021
8H8Q
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BU of 8h8q by Molmil
Fab-amyloid beta fragment complex at neutral pH
Descriptor: CHLORIDE ION, Fab, GLN-LYS-CYS-VAL-PHE-PHE-ALA-GLU-ASP-VAL-GLY-SER-ASN-CYS-GLY, ...
Authors:Kita, A, Irie, K, Irie, Y, Matsushima, Y, Miki, K.
Deposit date:2022-10-24
Release date:2023-10-25
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Fab-amyloid beta fragment complex at neutral pH
To Be Published
4TWW
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BU of 4tww by Molmil
Structure of SARS-3CL protease complex with a Bromobenzoyl (S,R)-N-decalin type inhibitor
Descriptor: (2S)-2-({[(3S,4aR,8aS)-2-(4-bromobenzoyl)decahydroisoquinolin-3-yl]methyl}amino)-3-(1H-imidazol-5-yl)propanal, 3C-like proteinase
Authors:Akaji, K, Teruya, K, Shimamoto, Y, Sanjho, A, Yamashita, E, Nakagawa, A.
Deposit date:2014-07-02
Release date:2015-02-18
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.42 Å)
Cite:Fused-ring structure of decahydroisoquinolin as a novel scaffold for SARS 3CL protease inhibitors
Bioorg.Med.Chem., 23, 2015
7FFI
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BU of 7ffi by Molmil
Diarylpentanoid-producing polyketide synthase (F340W mutant)
Descriptor: Type III polyketide synthase
Authors:Morita, H, Wong, C.P, Liu, Q, Kodama, T, Lee, Y, Nakashima, Y.
Deposit date:2021-07-23
Release date:2022-01-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Identification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood.
Nat Commun, 13, 2022
7FFG
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BU of 7ffg by Molmil
Diarylpentanoid-producing polyketide synthase (N199F mutant)
Descriptor: Type III polyketide synthase
Authors:Morita, H, Wong, C.P, Liu, Q, Kodama, T, Lee, Y, Nakashima, Y.
Deposit date:2021-07-23
Release date:2022-01-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Identification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood.
Nat Commun, 13, 2022
7FFA
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BU of 7ffa by Molmil
Diarylpentanoid-producing polyketide synthase from Aquilaria sinensis
Descriptor: Type III polyketide synthase
Authors:Morita, H, Wong, C.P, Liu, Q, Kodama, T, Lee, Y, Nakashima, Y.
Deposit date:2021-07-23
Release date:2022-01-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (1.98 Å)
Cite:Identification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood.
Nat Commun, 13, 2022
7FFH
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BU of 7ffh by Molmil
Diarylpentanoid-producing polyketide synthase (N199L mutant)
Descriptor: Type III polyketide synthase
Authors:Morita, H, Wong, C.P, Liu, Q, Takeshi, K, Lee, Y, Nakashima, Y.
Deposit date:2021-07-23
Release date:2022-01-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Identification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood.
Nat Commun, 13, 2022
6IN0
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BU of 6in0 by Molmil
Crystal structure of EphA3 in complex with 18-Crown-6
Descriptor: 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, CHLORIDE ION, Ephrin type-A receptor 3
Authors:Yokoyama, T, Kosaka, Y, Matsumoto, K, Kitakami, R, Nabeshima, Y, Mizuguchi, M.
Deposit date:2018-10-24
Release date:2019-10-30
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (1.501 Å)
Cite:Crown Ethers as Transthyretin Amyloidogenesis Inhibitor
To Be Published
6IMZ
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BU of 6imz by Molmil
Crystal structure of MTH1 in complex with 18-Crown-6
Descriptor: 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, 3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)pyridin-2-amine, 7,8-dihydro-8-oxoguanine triphosphatase, ...
Authors:Yokoyama, T, Kosaka, Y, Matsumoto, K, Kitakami, R, Nabeshima, Y, Mizuguchi, M.
Deposit date:2018-10-24
Release date:2019-10-30
Last modified:2024-03-27
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Crown Ethers as Transthyretin Amyloidogenesis Inhibitor
To Be Published

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