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PDB: 2 results

4YOA
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BU of 4yoa by Molmil
Crsystal structure HIV-1 Protease MDR769 L33F Complexed with darunavir
Descriptor: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, HIV-1 Protease
Authors:Kuiper, B.D, Keusch, B, Dewdney, T.G, Chordia, P, Brunzelle, J.S, Ross, K, Kovari, I.A, MacArthur, R, Salimnia, H, Kovari, L.C.
Deposit date:2015-03-11
Release date:2015-07-08
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.697 Å)
Cite:The L33F darunavir resistance mutation acts as a molecular anchor reducing the flexibility of the HIV-1 protease 30s and 80s loops.
Biochem Biophys Rep, 2, 2015
4YOB
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BU of 4yob by Molmil
Crystal Structure of Apo HIV-1 Protease MDR769 L33F
Descriptor: HIV-1 Protease
Authors:Kuiper, B.D, Keusch, B, Dewdney, T.G, Chordia, P, Ross, K, Brunzelle, J.S, Kovari, I.A, MacArthur, R, Salimnia, H, Kovari, L.C.
Deposit date:2015-03-11
Release date:2015-07-08
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.504 Å)
Cite:The L33F darunavir resistance mutation acts as a molecular anchor reducing the flexibility of the HIV-1 protease 30s and 80s loops.
Biochem Biophys Rep, 2, 2015

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