5TSG
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![BU of 5tsg by Molmil](/molmil-images/mine/5tsg) | PilB from Geobacter metallireducens bound to ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, FORMIC ACID, MAGNESIUM ION, ... | 著者 | McCallum, M, Tammam, S, Khan, A, Burrows, L, Howell, P.L. | 登録日 | 2016-10-28 | 公開日 | 2017-05-17 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.4011 Å) | 主引用文献 | The molecular mechanism of the type IVa pilus motors. Nat Commun, 8, 2017
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5V8E
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![BU of 5v8e by Molmil](/molmil-images/mine/5v8e) | Structure of Bacillus cereus PatB1 | 分子名称: | Bacillus cereus PatB1, CITRIC ACID, DI(HYDROXYETHYL)ETHER, ... | 著者 | Sychantha, D, Little, D.J, Chapman, R.N, Boons, G.J, Robinson, H, Howell, P.L, Clarke, A.J. | 登録日 | 2017-03-21 | 公開日 | 2017-10-18 | 最終更新日 | 2017-12-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | PatB1 is an O-acetyltransferase that decorates secondary cell wall polysaccharides. Nat. Chem. Biol., 14, 2018
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5VDI
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![BU of 5vdi by Molmil](/molmil-images/mine/5vdi) | Crystal Structure of Human Glycine Receptor alpha-3 Mutant N38Q Bound to AM-3607, Glycine, and Ivermectin | 分子名称: | (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, (3S,3aS,9bS)-2-[(2H-1,3-benzodioxol-5-yl)sulfonyl]-3,5-dimethyl-1,2,3,3a,5,9b-hexahydro-4H-pyrrolo[3,4-c][1,6]naphthyridin-4-one, GLYCINE, ... | 著者 | Shaffer, P.L, Huang, X, Chen, H. | 登録日 | 2017-04-03 | 公開日 | 2017-05-24 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Crystal Structures of Human GlyR alpha 3 Bound to Ivermectin. Structure, 25, 2017
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5VDH
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![BU of 5vdh by Molmil](/molmil-images/mine/5vdh) | Crystal Structure of Human Glycine Receptor alpha-3 Bound to AM-3607, Glycine, and Ivermectin | 分子名称: | (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, (3S,3aS,9bS)-2-[(2H-1,3-benzodioxol-5-yl)sulfonyl]-3,5-dimethyl-1,2,3,3a,5,9b-hexahydro-4H-pyrrolo[3,4-c][1,6]naphthyridin-4-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Shaffer, P.L, Huang, X, Chen, H. | 登録日 | 2017-04-03 | 公開日 | 2017-05-24 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Crystal Structures of Human GlyR alpha 3 Bound to Ivermectin. Structure, 25, 2017
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5VJS
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![BU of 5vjs by Molmil](/molmil-images/mine/5vjs) | De Novo Photosynthetic Reaction Center Protein Equipped with Heme B, a synthetic Zn porphyrin, and Zn(II) cations | 分子名称: | CHLORIDE ION, PROTOPORPHYRIN IX CONTAINING FE, Reaction Center Maquette, ... | 著者 | Ennist, N.M, Dutton, P.L, Stayrook, S.E, Moser, C.C. | 登録日 | 2017-04-19 | 公開日 | 2018-04-25 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | De novo protein design of photochemical reaction centers. Nat Commun, 13, 2022
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5VJU
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![BU of 5vju by Molmil](/molmil-images/mine/5vju) | De Novo Photosynthetic Reaction Center Protein Variant Equipped with His-Tyr H-bond, Heme B, and Cd(II) ions | 分子名称: | CADMIUM ION, PROTOPORPHYRIN IX CONTAINING FE, Reaction Center Maquette Leu71His variant | 著者 | Ennist, N.M, Stayrook, S.E, Dutton, P.L, Moser, C.C. | 登録日 | 2017-04-19 | 公開日 | 2018-04-25 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | De novo protein design of photochemical reaction centers. Nat Commun, 13, 2022
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1B3C
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![BU of 1b3c by Molmil](/molmil-images/mine/1b3c) | SOLUTION STRUCTURE OF A BETA-NEUROTOXIN FROM THE NEW WORLD SCORPION CENTRUROIDES SCULPTURATUS EWING | 分子名称: | PROTEIN (NEUROTOXIN CSE-I) | 著者 | Jablonsky, M.J, Jackson, P.L, Trent, J.O, Watt, D.D, Krishna, N.R. | 登録日 | 1998-12-08 | 公開日 | 1998-12-16 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of a beta-neurotoxin from the New World scorpion Centruroides sculpturatus Ewing. Biochem.Biophys.Res.Commun., 254, 1999
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1DF0
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![BU of 1df0 by Molmil](/molmil-images/mine/1df0) | Crystal structure of M-Calpain | 分子名称: | CALPAIN, M-CALPAIN | 著者 | Hosfield, C.M, Elce, J.S, Davies, P.L, Jia, Z. | 登録日 | 1999-11-16 | 公開日 | 2000-06-21 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of calpain reveals the structural basis for Ca(2+)-dependent protease activity and a novel mode of enzyme activation. EMBO J., 18, 1999
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1DCN
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![BU of 1dcn by Molmil](/molmil-images/mine/1dcn) | INACTIVE MUTANT H162N OF DELTA 2 CRYSTALLIN WITH BOUND ARGININOSUCCINATE | 分子名称: | ARGININOSUCCINATE, DELTA 2 CRYSTALLIN | 著者 | Vallee, F, Turner, M.A, Lindley, P, Howell, P.L. | 登録日 | 1998-10-29 | 公開日 | 1999-04-27 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of an inactive duck delta II crystallin mutant with bound argininosuccinate. Biochemistry, 38, 1999
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5T10
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![BU of 5t10 by Molmil](/molmil-images/mine/5t10) | |
1DL2
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![BU of 1dl2 by Molmil](/molmil-images/mine/1dl2) | CRYSTAL STRUCTURE OF CLASS I ALPHA-1,2-MANNOSIDASE FROM SACCHAROMYCES CEREVISIAE AT 1.54 ANGSTROM RESOLUTION | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, CLASS I ALPHA-1,2-MANNOSIDASE, ... | 著者 | Vallee, F, Lipari, F, Yip, P, Herscovics, A, Howell, P.L. | 登録日 | 1999-12-08 | 公開日 | 2000-02-18 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Crystal structure of a class I alpha1,2-mannosidase involved in N-glycan processing and endoplasmic reticulum quality control. EMBO J., 19, 2000
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5VJT
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![BU of 5vjt by Molmil](/molmil-images/mine/5vjt) | De Novo Photosynthetic Reaction Center Protein Equipped with Heme B and Zn(II) cations | 分子名称: | CHLORIDE ION, PROTOPORPHYRIN IX CONTAINING FE, Reaction Center Maquette, ... | 著者 | Ennist, N.M, Stayrook, S.E, Dutton, P.L, Moser, C.C. | 登録日 | 2017-04-19 | 公開日 | 2018-04-25 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | De novo protein design of photochemical reaction centers. Nat Commun, 13, 2022
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1AUW
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![BU of 1auw by Molmil](/molmil-images/mine/1auw) | |
1CKW
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![BU of 1ckw by Molmil](/molmil-images/mine/1ckw) | CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR: SOLUTION STRUCTURES OF PEPTIDES BASED ON THE PHE508 REGION, THE MOST COMMON SITE OF DISEASE-CAUSING DELTA-F508 MUTATION | 分子名称: | PROTEIN (CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR (CFTR)) | 著者 | Massiah, M.A, Ko, Y.H, Pedersen, P.L, Mildvan, A.S. | 登録日 | 1999-04-26 | 公開日 | 1999-05-04 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Cystic fibrosis transmembrane conductance regulator: solution structures of peptides based on the Phe508 region, the most common site of disease-causing DeltaF508 mutation. Biochemistry, 38, 1999
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1CKZ
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![BU of 1ckz by Molmil](/molmil-images/mine/1ckz) | CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR: SOLUTION STRUCTURES OF PEPTIDES BASED ON THE PHE508 REGION, THE MOST COMMON SITE OF DISEASE-CAUSING DELTA-F508 MUTATION | 分子名称: | PROTEIN (CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR (CFTR)) | 著者 | Massiah, M.A, Ko, Y.H, Pedersen, P.L, Mildvan, A.S. | 登録日 | 1999-04-26 | 公開日 | 1999-05-04 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Cystic fibrosis transmembrane conductance regulator: solution structures of peptides based on the Phe508 region, the most common site of disease-causing DeltaF508 mutation. Biochemistry, 38, 1999
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1SD1
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![BU of 1sd1 by Molmil](/molmil-images/mine/1sd1) | STRUCTURE OF HUMAN 5'-DEOXY-5'-METHYLTHIOADENOSINE PHOSPHORYLASE COMPLEXED WITH FORMYCIN A | 分子名称: | (1S)-1-(7-amino-1H-pyrazolo[4,3-d]pyrimidin-3-yl)-1,4-anhydro-D-ribitol, 5'-methylthioadenosine phosphorylase | 著者 | Lee, J.E, Settembre, E.C, Cornell, K.A, Riscoe, M.K, Sufrin, J.R, Ealick, S.E, Howell, P.L. | 登録日 | 2004-02-12 | 公開日 | 2004-05-18 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Structural Comparison of MTA Phosphorylase and MTA/AdoHcy Nucleosidase Explains Substrate Preferences and Identifies Regions Exploitable for Inhibitor Design. Biochemistry, 43, 2004
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1SD2
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![BU of 1sd2 by Molmil](/molmil-images/mine/1sd2) | STRUCTURE OF HUMAN 5'-DEOXY-5'-METHYLTHIOADENOSINE PHOSPHORYLASE COMPLEXED WITH 5'-METHYLTHIOTUBERCIDIN | 分子名称: | 2-(4-AMINO-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-METHYLSULFANYLMETHYL-TETRAHYDRO-FURAN-3,4-DIOL, 5'-methylthioadenosine phosphorylase, SULFATE ION | 著者 | Lee, J.E, Settembre, E.C, Cornell, K.A, Riscoe, M.K, Sufrin, J.R, Ealick, S.E, Howell, P.L. | 登録日 | 2004-02-12 | 公開日 | 2004-05-18 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural Comparison of MTA Phosphorylase and MTA/AdoHcy Nucleosidase Explains Substrate Preferences and Identifies Regions Exploitable for Inhibitor Design. Biochemistry, 43, 2004
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1NC1
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![BU of 1nc1 by Molmil](/molmil-images/mine/1nc1) | Crystal structure of E. coli MTA/AdoHcy nucleosidase complexed with 5'-methylthiotubercidin (MTH) | 分子名称: | 2-(4-AMINO-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-METHYLSULFANYLMETHYL-TETRAHYDRO-FURAN-3,4-DIOL, MTA/SAH nucleosidase | 著者 | Lee, J.E, Cornell, K.A, Riscoe, M.K, Howell, P.L. | 登録日 | 2002-12-04 | 公開日 | 2003-11-25 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of Escherichia coli 5'-methylthioadenosine/ S-adenosylhomocysteine nucleosidase inhibitor complexes provide insight into the conformational changes required for substrate binding and catalysis. J.Biol.Chem., 278, 2003
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1U16
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![BU of 1u16 by Molmil](/molmil-images/mine/1u16) | Crystal structure of a duck-delta-crystallin-1 double loop mutant (DLM) in complex with sulfate | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORIDE ION, Delta crystallin I, ... | 著者 | Tsai, M, Sampaleanu, L.M, Greene, C, Creagh, L, Haynes, C, Howell, P.L. | 登録日 | 2004-07-14 | 公開日 | 2004-10-05 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | A duck delta1 crystallin double loop mutant provides insight into residues important for argininosuccinate lyase activity. Biochemistry, 43, 2004
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1S4P
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![BU of 1s4p by Molmil](/molmil-images/mine/1s4p) | Crystal structure of yeast alpha1,2-mannosyltransferase Kre2p/Mnt1p: ternary complex with GDP/Mn and methyl-alpha-mannoside acceptor | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CHLORIDE ION, ... | 著者 | Lobsanov, Y.D, Romero, P.A, Sleno, B, Yu, B, Yip, P, Herscovics, A, Howell, P.L. | 登録日 | 2004-01-16 | 公開日 | 2004-05-04 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Structure of Kre2p/Mnt1p: A YEAST {alpha}1,2-MANNOSYLTRANSFERASE INVOLVED IN MANNOPROTEIN BIOSYNTHESIS J.Biol.Chem., 279, 2004
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1R4I
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![BU of 1r4i by Molmil](/molmil-images/mine/1r4i) | Crystal Structure of Androgen Receptor DNA-Binding Domain Bound to a Direct Repeat Response Element | 分子名称: | 5'-D(*CP*CP*AP*GP*AP*AP*CP*AP*TP*CP*AP*AP*GP*AP*AP*CP*AP*G)-3', 5'-D(*CP*TP*GP*TP*TP*CP*TP*TP*GP*AP*TP*GP*TP*TP*CP*TP*GP*G)-3', Androgen receptor, ... | 著者 | Shaffer, P.L, Jivan, A, Dollins, D.E, Claessens, F, Gewirth, D.T. | 登録日 | 2003-10-06 | 公開日 | 2004-06-29 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural basis of androgen receptor binding to selective androgen response elements. Proc.Natl.Acad.Sci.USA, 101, 2004
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1P4O
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![BU of 1p4o by Molmil](/molmil-images/mine/1p4o) | Structure of Apo unactivated IGF-1R KInase domain at 1.5A resolution. | 分子名称: | Insulin-like growth factor I receptor protein | 著者 | Munshi, S, Kornienko, M, Hall, D.L, Darke, P.L, Waxman, L, Kuo, L.C. | 登録日 | 2003-04-23 | 公開日 | 2003-04-29 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structure of apo, unactivated insulin-like growth factor-1 receptor kinase at 1.5 A resolution. Acta Crystallogr.,Sect.D, 59, 2003
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1U15
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![BU of 1u15 by Molmil](/molmil-images/mine/1u15) | Crystal structure of a duck-delta-crystallin-1 double loop mutant (DLM) | 分子名称: | Delta crystallin I | 著者 | Tsai, M, Sampaleanu, L.M, Greene, C, Creagh, L, Haynes, C, Howell, P.L. | 登録日 | 2004-07-14 | 公開日 | 2004-10-05 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | A duck delta1 crystallin double loop mutant provides insight into residues important for argininosuccinate lyase activity. Biochemistry, 43, 2004
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1OQJ
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![BU of 1oqj by Molmil](/molmil-images/mine/1oqj) | Crystal structure of the SAND domain from glucocorticoid modulatory element binding protein-1 (GMEB1) | 分子名称: | Glucocorticoid Modulatory Element Binding protein-1, ZINC ION | 著者 | Surdo, P.L, Bottomley, M.J, Sattler, M, Scheffzek, K. | 登録日 | 2003-03-10 | 公開日 | 2003-11-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Crystal structure and nuclear magnetic resonance analyses of the SAND domain from glucocorticoid modulatory element binding protein-1 reveals deoxyribonucleic acid and zinc binding regions MOL.ENDOCRINOL., 17, 2003
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1RGQ
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![BU of 1rgq by Molmil](/molmil-images/mine/1rgq) | M9A HCV Protease complex with pentapeptide keto-amide inhibitor | 分子名称: | N-(PYRAZIN-2-YLCARBONYL)LEUCYLISOLEUCYL-N~1~-{1-[2-({1-CARBOXY-2-[4-(PHOSPHONOOXY)PHENYL]ETHYL}AMINO)-1,1-DIHYDROXY-2-OXOETHYL]BUT-3-ENYL}-3-CYCLOHEXYLALANINAMIDE, NS3 Protease, NS4A peptide, ... | 著者 | Liu, Y, Stoll, V.S, Richardson, P.L, Saldivar, A, Klaus, J.L, Molla, A, Kohlbrenner, W, Kati, W.M. | 登録日 | 2003-11-12 | 公開日 | 2004-10-19 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Hepatitis C NS3 protease inhibition by peptidyl-alpha-ketoamide inhibitors: kinetic mechanism and structure. Arch.Biochem.Biophys., 421, 2004
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