6LUE
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![BU of 6lue by Molmil](/molmil-images/mine/6lue) | Crystal structure of mouse Cryptochrome 1 in complex with compound KL201 | 分子名称: | 2-bromanyl-N-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)benzamide, Cryptochrome-1 | 著者 | Miller, S, Aikawa, Y, Hirota, T. | 登録日 | 2020-01-27 | 公開日 | 2020-06-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | An Isoform-Selective Modulator of Cryptochrome 1 Regulates Circadian Rhythms in Mammals. Cell Chem Biol, 27, 2020
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7DLI
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![BU of 7dli by Molmil](/molmil-images/mine/7dli) | Crystal structure of mouse CRY1 in complex with KL001 compound | 分子名称: | 1,2-ETHANEDIOL, Cryptochrome-1, N-[(2R)-3-carbazol-9-yl-2-oxidanyl-propyl]-N-(furan-2-ylmethyl)methanesulfonamide | 著者 | Miller, S.A, Aikawa, Y, Hirota, T. | 登録日 | 2020-11-27 | 公開日 | 2021-06-23 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural differences in the FAD-binding pockets and lid loops of mammalian CRY1 and CRY2 for isoform-selective regulation. Proc.Natl.Acad.Sci.USA, 118, 2021
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7D0N
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7D0M
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7WVA
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![BU of 7wva by Molmil](/molmil-images/mine/7wva) | |
7V8Y
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![BU of 7v8y by Molmil](/molmil-images/mine/7v8y) | |
7V8Z
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![BU of 7v8z by Molmil](/molmil-images/mine/7v8z) | |
7EJ9
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![BU of 7ej9 by Molmil](/molmil-images/mine/7ej9) | |
7D1C
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![BU of 7d1c by Molmil](/molmil-images/mine/7d1c) | |
7D19
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1HXS
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![BU of 1hxs by Molmil](/molmil-images/mine/1hxs) | CRYSTAL STRUCTURE OF MAHONEY STRAIN OF POLIOVIRUS AT 2.2A RESOLUTION | 分子名称: | GENOME POLYPROTEIN, COAT PROTEIN VP1, COAT PROTEIN VP2, ... | 著者 | Miller, S.T, Hogle, J.M, Filman, D.J. | 登録日 | 2001-01-16 | 公開日 | 2002-01-16 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Ab initio phasing of high-symmetry macromolecular complexes: successful phasing of authentic poliovirus data to 3.0 A resolution. J.Mol.Biol., 307, 2001
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6KX8
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![BU of 6kx8 by Molmil](/molmil-images/mine/6kx8) | Crystal structure of mouse Cryptochrome 2 in complex with TH301 compound | 分子名称: | 1-(4-chlorophenyl)-N-[2-(4-methoxyphenyl)-5,5-bis(oxidanylidene)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]cyclopentane-1-carboxamide, Cryptochrome-2 | 著者 | Miller, S.A, Aikawa, Y, Hirota, T. | 登録日 | 2019-09-10 | 公開日 | 2020-04-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Isoform-selective regulation of mammalian cryptochromes. Nat.Chem.Biol., 16, 2020
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6KX7
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![BU of 6kx7 by Molmil](/molmil-images/mine/6kx7) | Crystal structure of mouse Cryptochrome 1 in complex with TH301 compound | 分子名称: | 1-(4-chlorophenyl)-N-[2-(4-methoxyphenyl)-5,5-bis(oxidanylidene)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]cyclopentane-1-carboxamide, Cryptochrome-1 | 著者 | Miller, S.A, Aikawa, Y, Hirota, T. | 登録日 | 2019-09-10 | 公開日 | 2020-04-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Isoform-selective regulation of mammalian cryptochromes. Nat.Chem.Biol., 16, 2020
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6KX5
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6KX6
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![BU of 6kx6 by Molmil](/molmil-images/mine/6kx6) | Crystal structure of mouse Cryptochrome 1 in complex with KL101 compound | 分子名称: | Cryptochrome-1, ~{N}-[2-(2,4-dimethylphenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]-3,4-dimethyl-benzamide | 著者 | Miller, S.A, Aikawa, Y, Hirota, T. | 登録日 | 2019-09-10 | 公開日 | 2020-04-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Isoform-selective regulation of mammalian cryptochromes. Nat.Chem.Biol., 16, 2020
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6KX4
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4BNP
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![BU of 4bnp by Molmil](/molmil-images/mine/4bnp) | 3D structure of E. coli Isocitrate Dehydrogenase K100M mutant in complex with isocitrate and magnesium(II) | 分子名称: | ISOCITRATE DEHYDROGENASE [NADP], ISOCITRIC ACID, MAGNESIUM ION, ... | 著者 | Miller, S.P, Goncalves, S, Matias, P.M, Dean, A.M. | 登録日 | 2013-05-16 | 公開日 | 2014-05-21 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Evolution of a Transition State: Role of Lys100 in the Active Site of Isocitrate Dehydrogenase. Chembiochem, 15, 2014
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3ZYK
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![BU of 3zyk by Molmil](/molmil-images/mine/3zyk) | Structure of CALM (PICALM) ANTH domain | 分子名称: | PHOSPHATIDYLINOSITOL-BINDING CLATHRIN ASSEMBLY PROTEIN | 著者 | Miller, S.E, Sahlender, D.A, Graham, S.C, Honing, S, Robinson, M.S, Peden, A.A, Owen, D.J. | 登録日 | 2011-08-23 | 公開日 | 2011-12-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The molecular basis for the endocytosis of small R-SNAREs by the clathrin adaptor CALM. Cell, 147, 2011
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3ZYM
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![BU of 3zym by Molmil](/molmil-images/mine/3zym) | Structure of CALM (PICALM) in complex with VAMP8 | 分子名称: | GLYCEROL, PHOSPHATE ION, PHOSPHATIDYLINOSITOL-BINDING CLATHRIN ASSEMBLY PROTEIN, ... | 著者 | Miller, S.E, Sahlender, D.A, Graham, S.C, Honing, S, Robinson, M.S, Peden, A.A, Owen, D.J. | 登録日 | 2011-08-23 | 公開日 | 2011-12-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | The molecular basis for the endocytosis of small R-SNAREs by the clathrin adaptor CALM. Cell, 147, 2011
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3ZYL
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![BU of 3zyl by Molmil](/molmil-images/mine/3zyl) | Structure of a truncated CALM (PICALM) ANTH domain | 分子名称: | PHOSPHATIDYLINOSITOL-BINDING CLATHRIN ASSEMBLY PROTEIN | 著者 | Miller, S.E, Sahlender, D.A, Graham, S.C, Honing, S, Robinson, M.S, Peden, A.A, Owen, D.J. | 登録日 | 2011-08-23 | 公開日 | 2011-12-07 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The molecular basis for the endocytosis of small R-SNAREs by the clathrin adaptor CALM. Cell, 147, 2011
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8G6Z
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![BU of 8g6z by Molmil](/molmil-images/mine/8g6z) | JAK2 crystal structure in complex with Compound 13 | 分子名称: | (3R)-3-cyclopentyl-3-[(4M)-4-{5-methyl-2-[(1-methyl-1H-pyrazol-4-yl)amino]pyrimidin-4-yl}-1H-pyrazol-1-yl]propanenitrile, 1,2-ETHANEDIOL, Tyrosine-protein kinase JAK2 | 著者 | Miller, S.T, Ellis, D.A. | 登録日 | 2023-02-16 | 公開日 | 2023-06-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Eyes on Topical Ocular Disposition: The Considered Design of a Lead Janus Kinase (JAK) Inhibitor That Utilizes a Unique Azetidin-3-Amino Bridging Scaffold to Attenuate Off-Target Kinase Activity, While Driving Potency and Aqueous Solubility. J.Med.Chem., 66, 2023
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8G8O
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![BU of 8g8o by Molmil](/molmil-images/mine/8g8o) | The crystal structure of JAK2 in complex with Compound 31 | 分子名称: | 1,2-ETHANEDIOL, DIMETHYL SULFOXIDE, Tyrosine-protein kinase JAK2, ... | 著者 | Miller, S.T, Ellis, D.A. | 登録日 | 2023-02-18 | 公開日 | 2023-06-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Eyes on Topical Ocular Disposition: The Considered Design of a Lead Janus Kinase (JAK) Inhibitor That Utilizes a Unique Azetidin-3-Amino Bridging Scaffold to Attenuate Off-Target Kinase Activity, While Driving Potency and Aqueous Solubility. J.Med.Chem., 66, 2023
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8G8X
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![BU of 8g8x by Molmil](/molmil-images/mine/8g8x) | X-ray co-crystal structure of compound 27 in with complex JAK2 | 分子名称: | 3-cyclopropyl-1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}azetidin-3-ol, Tyrosine-protein kinase JAK2 | 著者 | Miller, S.T, Ellis, D.A. | 登録日 | 2023-02-20 | 公開日 | 2023-06-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Eyes on Topical Ocular Disposition: The Considered Design of a Lead Janus Kinase (JAK) Inhibitor That Utilizes a Unique Azetidin-3-Amino Bridging Scaffold to Attenuate Off-Target Kinase Activity, While Driving Potency and Aqueous Solubility. J.Med.Chem., 66, 2023
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2QYW
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![BU of 2qyw by Molmil](/molmil-images/mine/2qyw) | Crystal structure of mouse vti1b Habc domain | 分子名称: | Vesicle transport through interaction with t-SNAREs 1B homolog | 著者 | Miller, S.E, Collins, B.M, McCoy, A.J, Robinson, M.S, Owen, D.J. | 登録日 | 2007-08-15 | 公開日 | 2007-11-27 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | A SNARE-adaptor interaction is a new mode of cargo recognition in clathrin-coated vesicles. Nature, 450, 2007
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2QY7
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![BU of 2qy7 by Molmil](/molmil-images/mine/2qy7) | Crystal structure of human epsinR ENTH domain | 分子名称: | Clathrin interactor 1 | 著者 | Miller, S.E, Collins, B.M, McCoy, A.J, Robinson, M.S, Owen, D.J. | 登録日 | 2007-08-13 | 公開日 | 2007-11-27 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | A SNARE-adaptor interaction is a new mode of cargo recognition in clathrin-coated vesicles. Nature, 450, 2007
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