6LUE
Crystal structure of mouse Cryptochrome 1 in complex with compound KL201
Summary for 6LUE
Entry DOI | 10.2210/pdb6lue/pdb |
Descriptor | Cryptochrome-1, 2-bromanyl-N-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)benzamide (3 entities in total) |
Functional Keywords | cryptochrome, cry, circadian clock, kl201, circadian clock protein |
Biological source | Mus musculus (Mouse) |
Total number of polymer chains | 2 |
Total formula weight | 115520.03 |
Authors | Miller, S.,Aikawa, Y.,Hirota, T. (deposition date: 2020-01-27, release date: 2020-06-10, Last modification date: 2023-11-29) |
Primary citation | Miller, S.,Aikawa, Y.,Sugiyama, A.,Nagai, Y.,Hara, A.,Oshima, T.,Amaike, K.,Kay, S.A.,Itami, K.,Hirota, T. An Isoform-Selective Modulator of Cryptochrome 1 Regulates Circadian Rhythms in Mammals. Cell Chem Biol, 27:1192-1198.e5, 2020 Cited by PubMed: 32502390DOI: 10.1016/j.chembiol.2020.05.008 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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