2O6F
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![BU of 2o6f by Molmil](/molmil-images/mine/2o6f) | Structure of metal- free rTp34 from Treponema pallidum | 分子名称: | 1,2-ETHANEDIOL, 34 kDa membrane antigen, CHLORIDE ION, ... | 著者 | Machius, M, Brautigam, C.A, Deka, R.K, Tomchick, D.R, Lumpkins, S.B, Norgard, M.V. | 登録日 | 2006-12-07 | 公開日 | 2006-12-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Crystal structure of the Tp34 (TP0971) lipoprotein of treponema pallidum: implications of its metal-bound state and affinity for human lactoferrin. J.Biol.Chem., 282, 2007
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2O6D
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![BU of 2o6d by Molmil](/molmil-images/mine/2o6d) | Structure of native rTp34 from Treponema pallidum | 分子名称: | 1,2-ETHANEDIOL, 34 kDa membrane antigen, CHLORIDE ION, ... | 著者 | Machius, M, Brautigam, C.A, Deka, R.K, Tomchick, D.R, Lumpkins, S.B, Norgard, M.V. | 登録日 | 2006-12-07 | 公開日 | 2006-12-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Crystal structure of the Tp34 (TP0971) lipoprotein of treponema pallidum: implications of its metal-bound state and affinity for human lactoferrin. J.Biol.Chem., 282, 2007
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2O6C
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![BU of 2o6c by Molmil](/molmil-images/mine/2o6c) | Structure of selenomethionyl rTp34 from Treponema pallidum | 分子名称: | 1,2-ETHANEDIOL, 34 kDa membrane antigen, CHLORIDE ION, ... | 著者 | Machius, M, Brautigam, C.A, Deka, R.K, Tomchick, D.R, Lumpkins, S.B, Norgard, M.V. | 登録日 | 2006-12-07 | 公開日 | 2006-12-26 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of the Tp34 (TP0971) lipoprotein of treponema pallidum: implications of its metal-bound state and affinity for human lactoferrin. J.Biol.Chem., 282, 2007
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2O6E
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![BU of 2o6e by Molmil](/molmil-images/mine/2o6e) | Structure of native rTp34 from Treponema pallidum from zinc-soaked crystals | 分子名称: | 1,2-ETHANEDIOL, 34 kDa membrane antigen, CHLORIDE ION, ... | 著者 | Machius, M, Brautigam, C.A, Deka, R.K, Tomchick, D.R, Lumpkins, S.B, Norgard, M.V. | 登録日 | 2006-12-07 | 公開日 | 2006-12-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of the Tp34 (TP0971) lipoprotein of treponema pallidum: implications of its metal-bound state and affinity for human lactoferrin. J.Biol.Chem., 282, 2007
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1N11
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![BU of 1n11 by Molmil](/molmil-images/mine/1n11) | D34 REGION OF HUMAN ANKYRIN-R AND LINKER | 分子名称: | Ankyrin, BROMIDE ION, CHLORIDE ION | 著者 | Michaely, P, Tomchick, D.R, Machius, M, Anderson, R.G.W. | 登録日 | 2002-10-16 | 公開日 | 2002-12-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal structure of a 12 ANK repeat stack from human ankyrinR Embo J., 21, 2002
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1W15
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![BU of 1w15 by Molmil](/molmil-images/mine/1w15) | rat synaptotagmin 4 C2B domain in the presence of calcium | 分子名称: | CALCIUM ION, CHLORIDE ION, SODIUM ION, ... | 著者 | Dai, H, Shin, O.-H, Machius, M, Tomchick, D.R, Sudhof, T.C, Rizo, J. | 登録日 | 2004-06-16 | 公開日 | 2004-08-13 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.93 Å) | 主引用文献 | Structural Basis for the Evolutionary Inactivation of Ca2+ Binding to Synaptotagmin 4 Nat.Struct.Mol.Biol., 11, 2004
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1W16
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![BU of 1w16 by Molmil](/molmil-images/mine/1w16) | rat synaptotagmin 4 C2B domain in the absence of calcium | 分子名称: | CHLORIDE ION, SODIUM ION, SYNAPTOTAGMIN IV | 著者 | Dai, H, Shin, O.-H, Machius, M, Tomchick, D.R, Sudhof, T.C, Rizo, J. | 登録日 | 2004-06-16 | 公開日 | 2004-08-13 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural Basis for the Evolutionary Inactivation of Ca2+ Binding to Synaptotagmin 4 Nat.Struct.Mol.Biol., 11, 2004
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6NYC
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![BU of 6nyc by Molmil](/molmil-images/mine/6nyc) | Munc13-1 C2B-domain, calcium free | 分子名称: | 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, Munc13-1 | 著者 | Tomchick, D.R, Rizo, J, Machius, M, Lu, J. | 登録日 | 2019-02-11 | 公開日 | 2019-02-20 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.893 Å) | 主引用文献 | Munc13 C2B domain is an activity-dependent Ca2+ regulator of synaptic exocytosis. Nat. Struct. Mol. Biol., 17, 2010
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3V1A
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![BU of 3v1a by Molmil](/molmil-images/mine/3v1a) | Crystal structure of de novo designed MID1-apo1 | 分子名称: | Computational design, MID1-apo1 | 著者 | Der, B.S, Machius, M, Miley, M.J, Kuhlman, B. | 登録日 | 2011-12-09 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (0.98 Å) | 主引用文献 | Metal-mediated affinity and orientation specificity in a computationally designed protein homodimer. J.Am.Chem.Soc., 134, 2012
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3V1E
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![BU of 3v1e by Molmil](/molmil-images/mine/3v1e) | Crystal structure of de novo designed MID1-zinc H12E mutant | 分子名称: | Computational design, MID1-zinc H12E mutant, ZINC ION | 著者 | Der, B.S, Machius, M, Miley, M.J, Kuhlman, B. | 登録日 | 2011-12-09 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.073 Å) | 主引用文献 | Metal-mediated affinity and orientation specificity in a computationally designed protein homodimer. J.Am.Chem.Soc., 134, 2012
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3V1C
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![BU of 3v1c by Molmil](/molmil-images/mine/3v1c) | Crystal structure of de novo designed MID1-zinc | 分子名称: | Computational design, MID1-zinc, L(+)-TARTARIC ACID, ... | 著者 | Der, B.S, Machius, M, Miley, M.J, Kuhlman, B. | 登録日 | 2011-12-09 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.129 Å) | 主引用文献 | Metal-mediated affinity and orientation specificity in a computationally designed protein homodimer. J.Am.Chem.Soc., 134, 2012
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2FQW
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![BU of 2fqw by Molmil](/molmil-images/mine/2fqw) | PnrA from Treponema pallidum as purified from E. coli (bound to inosine) | 分子名称: | INOSINE, Membrane lipoprotein tmpC | 著者 | Brautigam, C.A, Deka, R.K, Tomchick, D.R, Machius, M, Norgard, M.V. | 登録日 | 2006-01-18 | 公開日 | 2006-02-14 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | The PnrA (Tp0319; TmpC) lipoprotein represents a new family of bacterial purine nucleoside receptor encoded within an ATP-binding cassette (ABC)-like operon in Treponema pallidum J.Biol.Chem., 281, 2006
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2FQY
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![BU of 2fqy by Molmil](/molmil-images/mine/2fqy) | PnrA from Treponema pallidum complexed with adenosine. | 分子名称: | ADENOSINE, Membrane lipoprotein tmpC | 著者 | Brautigam, C.A, Deka, R.K, Tomchick, D.R, Machius, M, Norgard, M.V. | 登録日 | 2006-01-18 | 公開日 | 2006-02-14 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | The PnrA (Tp0319; TmpC) lipoprotein represents a new family of bacterial purine nucleoside receptor encoded within an ATP-binding cassette (ABC)-like operon in Treponema pallidum J.Biol.Chem., 281, 2006
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2XNS
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![BU of 2xns by Molmil](/molmil-images/mine/2xns) | Crystal Structure Of Human G alpha i1 Bound To A Designed Helical Peptide Derived From The Goloco Motif Of RGS14 | 分子名称: | GUANINE NUCLEOTIDE-BINDING PROTEIN G(I) SUBUNIT ALPHA-1, GUANOSINE-5'-DIPHOSPHATE, REGULATOR OF G-PROTEIN SIGNALING 14, ... | 著者 | Bosch, D, Sammond, D.W, Butterfoss, G.L, Machius, M, Siderovski, D.P, Kuhlman, B. | 登録日 | 2010-08-05 | 公開日 | 2011-06-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.41 Å) | 主引用文献 | Computational Design of the Sequence and Structure of a Protein-Binding Peptide. J.Am.Chem.Soc., 133, 2011
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2XTZ
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![BU of 2xtz by Molmil](/molmil-images/mine/2xtz) | Crystal structure of the G alpha protein AtGPA1 from Arabidopsis thaliana | 分子名称: | 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, CHLORIDE ION, GUANINE NUCLEOTIDE-BINDING PROTEIN ALPHA-1 SUBUNIT, ... | 著者 | Jones, J.C, Duffy, J.W, Machius, M, Temple, B.R.S, Dohlman, H.G, Jones, A.M. | 登録日 | 2010-10-13 | 公開日 | 2011-02-16 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | The Crystal Structure of a Self-Activating G Protein Alpha Subunit Reveals its Distinct Mechanism of Signal Initiation Sci.Signal., 159, 2011
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5VPB
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![BU of 5vpb by Molmil](/molmil-images/mine/5vpb) | Transcription factor FosB/JunD bZIP domain in its oxidized form, type-I crystal | 分子名称: | CHLORIDE ION, Protein fosB, Transcription factor jun-D | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.691 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
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5VPD
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![BU of 5vpd by Molmil](/molmil-images/mine/5vpd) | Transcription factor FosB/JunD bZIP domain in its oxidized form, type-III crystal | 分子名称: | CHLORIDE ION, Protein fosB, SODIUM ION, ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
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5VPA
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![BU of 5vpa by Molmil](/molmil-images/mine/5vpa) | Transcription factor FosB/JunD bZIP domain | 分子名称: | CHLORIDE ION, Protein fosB, SODIUM ION, ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.83 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
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5VPF
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![BU of 5vpf by Molmil](/molmil-images/mine/5vpf) | Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-II crystal | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ... | 著者 | Yin, Z, Rudenko, G, Machius, M. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.694 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
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3KY9
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![BU of 3ky9 by Molmil](/molmil-images/mine/3ky9) | Autoinhibited Vav1 | 分子名称: | Proto-oncogene vav, ZINC ION | 著者 | Tomchick, D.R, Rosen, M.K, Machius, M, Yu, B. | 登録日 | 2009-12-04 | 公開日 | 2010-02-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.731 Å) | 主引用文献 | Structural and Energetic Mechanisms of Cooperative Autoinhibition and Activation of Vav1 Cell(Cambridge,Mass.), 140, 2010
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5VPE
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![BU of 5vpe by Molmil](/molmil-images/mine/5vpe) | Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-I crystal | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.053 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
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6NYT
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![BU of 6nyt by Molmil](/molmil-images/mine/6nyt) | Munc13-1 C2B-domain, calcium bound | 分子名称: | CALCIUM ION, CHLORIDE ION, GLYCEROL, ... | 著者 | Tomchick, D.R, Rizo, J, Machius, M, Lu, J. | 登録日 | 2019-02-12 | 公開日 | 2019-02-20 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.369 Å) | 主引用文献 | Munc13 C2B domain is an activity-dependent Ca2+ regulator of synaptic exocytosis. Nat. Struct. Mol. Biol., 17, 2010
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5K0K
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![BU of 5k0k by Molmil](/molmil-images/mine/5k0k) | Crystal structure of the catalytic domain of the proto-oncogene tyrosine-protein kinase MER in complex with inhibitor UNC2434 | 分子名称: | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]te traazacyclotetradecin-8(3H)-one, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Wang, X, Liu, J, Zhang, W, Stashko, M.A, Nichols, J, DeRyckere, D, Miley, M.J, Norris-Drouin, J, Chen, Z, Machius, M, Wood, E, Graham, D.K, Earp, H.S, Graham, K, Kireev, D, Frye, S.V. | 登録日 | 2016-05-17 | 公開日 | 2017-01-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.545 Å) | 主引用文献 | Design and Synthesis of Novel Macrocyclic Mer Tyrosine Kinase Inhibitors. ACS Med Chem Lett, 7, 2016
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5K0X
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![BU of 5k0x by Molmil](/molmil-images/mine/5k0x) | Crystal structure of the catalytic domain of the proto-oncogene tyrosine-protein kinase MER in complex with inhibitor UNC2541 | 分子名称: | (7S)-7-amino-N-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide, CHLORIDE ION, Tyrosine-protein kinase Mer | 著者 | McIver, A.L, Zhang, W, Liu, Q, Jiang, X, Stashko, M.A, Nichols, J, Miley, M.J, Norris-Drouin, J, Machius, M, DeRyckere, D, Wood, E, Graham, D.K, Earp, H.S, Kireev, D, Frye, S.V, Wang, X. | 登録日 | 2016-05-17 | 公開日 | 2017-02-22 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.231 Å) | 主引用文献 | Discovery of Macrocyclic Pyrimidines as MerTK-Specific Inhibitors. ChemMedChem, 12, 2017
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2J9F
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![BU of 2j9f by Molmil](/molmil-images/mine/2j9f) | Human branched-chain alpha-ketoacid dehydrogenase-decarboxylase E1b | 分子名称: | 2-OXOISOVALERATE DEHYDROGENASE ALPHA SUBUNIT, 2-OXOISOVALERATE DEHYDROGENASE BETA SUBUNIT, C2-1-HYDROXY-3-METHYL-PROPYL-THIAMIN DIPHOSPHATE, ... | 著者 | Jun, L, Machius, M, Chuang, J.L, Wynn, R.M, Chuang, D.T. | 登録日 | 2006-11-07 | 公開日 | 2007-02-27 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | The Two Active Sites in Human Branched-Chain Alpha- Keto Acid Dehydrogenase Operate Independently without an Obligatory Alternating-Site Mechanism. J.Biol.Chem., 282, 2007
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