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PDB: 51630 件

6W5E
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Class D beta-lactamase BSU-2
分子名称: 1,2-ETHANEDIOL, BSU-2 beta-lactamase, MALONATE ION
著者Smith, C.A, Vakulenko, S.B, Stewart, N.K, Toth, M.
登録日2020-03-13
公開日2020-06-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献A surface loop modulates activity of the Bacillus class D beta-lactamases.
J.Struct.Biol., 211, 2020
7AEN
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Galectin-8 N-terminal carbohydrate recognition domain in complex with methyl 3-O-((7-carboxy)quinolin-2-yl)-methoxy)-beta-D-galactopyranoside
分子名称: CHLORIDE ION, GLYCEROL, Isoform 2 of Galectin-8, ...
著者Hassan, M, Klavern, V.S, Hakansson, M, Anderluh, M, Tomasic, T, Jakopin, Z, Nilsson, J.U, Kovacic, R, Walse, B, Diehl, C.
登録日2020-09-17
公開日2021-07-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure-Guided Design of d-Galactal Derivatives with High Affinity and Selectivity for the Galectin-8 N-Terminal Domain
Acs Med.Chem.Lett., 12, 2021
5NX2
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Crystal structure of thermostabilised full-length GLP-1R in complex with a truncated peptide agonist at 3.7 A resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Glucagon-like peptide 1 receptor, ...
著者Rappas, M, Jazayeri, A, Brown, A.J.H, Kean, J, Errey, J.C, Robertson, N, Fiez-Vandal, C, Andrews, S.P, Congreve, M, Bortolato, A, Mason, J.S, Baig, A.H, Teobald, I, Dore, A.S, Weir, M, Cooke, R.M, Marshall, F.H.
登録日2017-05-09
公開日2017-06-14
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3.7 Å)
主引用文献Crystal structure of the GLP-1 receptor bound to a peptide agonist.
Nature, 546, 2017
5DQU
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Crystal Structure of Cas-DNA-10 complex
分子名称: CRISPR-associated endonuclease Cas1, CRISPR-associated endoribonuclease Cas2, DNA (5'-D(*GP*AP*GP*TP*CP*GP*AP*TP*GP*CP*TP*TP*TP*TP*T)-3'), ...
著者Wang, J, Li, J, Zhao, H, Sheng, G, Wang, M, Yin, M, Wang, Y.
登録日2015-09-15
公開日2015-11-11
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (4.5 Å)
主引用文献Structural and Mechanistic Basis of PAM-Dependent Spacer Acquisition in CRISPR-Cas Systems.
Cell, 163, 2015
8JXF
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rat megalin RAP complex bodyA
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-2-macroglobulin receptor-associated protein, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8JUT
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rat megalin RAP complex
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-27
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
7JX4
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Crystal Structure of N-Lysine Peptoid-modified Collagen Triple Helix
分子名称: Collagen mimetic peptide with N-Lysine guest
著者Yu, M.S, Whitby, F.G, Hill, C.P, Kessler, J.L, Yang, L.D.
登録日2020-08-26
公開日2021-07-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (0.95 Å)
主引用文献Peptoid Residues Make Diverse, Hyperstable Collagen Triple-Helices.
J.Am.Chem.Soc., 143, 2021
7JX5
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Crystal Structure of N-Phenylalanine Peptoid-modified Collagen Triple Helix
分子名称: Collagen mimetic peptide with N-Phenylalanine guest
著者Yu, M.S, Whitby, F.G, Hill, C.P, Kessler, J.L, Yang, L.D.
登録日2020-08-26
公開日2021-07-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Peptoid Residues Make Diverse, Hyperstable Collagen Triple-Helices
J.Am.Chem.Soc., 143, 2021
8JXI
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rat megalin RAP complex wingB
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8JXH
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rat megalin RAP complex wingA
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8JXA
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cryo-EM structure of rat megalin bodyB
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
6GE0
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Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2
分子名称: 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{H}-isoindol-2-yl]-~{N}-[(1~{R})-1-(3-methoxyphenyl)ethyl]ethanamide, DIMETHYL SULFOXIDE, Mitogen-activated protein kinase 1, ...
著者O'Reilly, M.
登録日2018-04-25
公開日2018-05-30
最終更新日2018-06-27
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2.
J. Med. Chem., 61, 2018
8JXB
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BU of 8jxb by Molmil
Cryo-EM structure of rat megalin wingAc
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8CXP
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Characterisation of a Seneca Valley Virus Thermostable Mutant
分子名称: Capsid protein VP1, Capsid protein VP3, VP2, ...
著者Jayawardena, N, Bostina, M, Strauss, M.
登録日2022-05-22
公開日2022-09-28
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (2.47 Å)
主引用文献Characterisation of a Seneca Valley virus thermostable mutant.
Virology, 575, 2022
8JXG
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rat megalin RAP complex bodyB
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
6FTK
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Gp36-MPER
分子名称: Envelope protein
著者D'Ursi, A.M, Grimaldi, M.
登録日2018-02-22
公開日2019-03-20
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献NMR Structure of the FIV gp36 C-Terminal Heptad Repeat and Membrane-Proximal External Region.
Int J Mol Sci, 21, 2020
7REF
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BU of 7ref by Molmil
Structure of MS3494 from Mycobacterium smegmatis
分子名称: BROMIDE ION, MS3494
著者Kent, J.E, Aleshin, A.E, Zhang, L, Niederweis, M, Marassi, F.M.
登録日2021-07-12
公開日2021-08-18
最終更新日2022-06-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A periplasmic cinched protein is required for siderophore secretion and virulence of Mycobacterium tuberculosis.
Nat Commun, 13, 2022
6G81
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Solution structure of the Ni metallochaperone HypA from Helicobacter pylori
分子名称: Hydrogenase maturation factor HypA, ZINC ION
著者Spronk, C.A.E.M, Zerko, S, Gorka, M, Kozminski, W, Bardiaux, B, Zambelli, B, Musiani, F, Piccioli, M, Hu, H, Maroney, M, Ciurli, S.
登録日2018-04-07
公開日2018-10-10
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献Structure and dynamics of Helicobacter pylori nickel-chaperone HypA: an integrated approach using NMR spectroscopy, functional assays and computational tools.
J. Biol. Inorg. Chem., 23, 2018
8JXJ
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rat megalin RAP complex leg
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, LDL receptor related protein 2, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8JX9
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rat megalin bodyA
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
8JXE
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rat megalin RAP complex head
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Goto, S, Tsutsumi, A, Lee, Y, Hosojima, M, Kabasawa, H, Komochi, K, Yun-san, L, Nagatoshi, S, Tsumoto, K, Nishizawa, T, Kikkawa, M, Saito, A.
登録日2023-06-30
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-EM structures elucidate the multiligand receptor nature of megalin.
Proc.Natl.Acad.Sci.USA, 121, 2024
6W7B
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K2P2.1 (TREK-1), 0 mM K+
分子名称: CADMIUM ION, DECANE, DODECANE, ...
著者Lolicato, M, Minor, D.L.
登録日2020-03-19
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.88 Å)
主引用文献K 2P channel C-type gating involves asymmetric selectivity filter order-disorder transitions.
Sci Adv, 6, 2020
6W84
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K2P2.1 (TREK-1), 200 mM K+
分子名称: CADMIUM ION, DODECANE, N-OCTANE, ...
著者Lolicato, M, Minor, D.L.
登録日2020-03-20
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.7 Å)
主引用文献K 2P channel C-type gating involves asymmetric selectivity filter order-disorder transitions.
Sci Adv, 6, 2020
6W8A
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K2P2.1 (TREK-1):ML335 complex, 10 mM K+
分子名称: CADMIUM ION, DODECANE, HEXADECANE, ...
著者Lolicato, M, Minor, D.L.
登録日2020-03-20
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.002 Å)
主引用文献K 2P channel C-type gating involves asymmetric selectivity filter order-disorder transitions.
Sci Adv, 6, 2020
6W8F
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K2P2.1 (TREK-1):ML335 complex, 0 mM K+
分子名称: CADMIUM ION, DODECANE, HEXADECANE, ...
著者Lolicato, M, Minor, D.L.
登録日2020-03-20
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献K 2P channel C-type gating involves asymmetric selectivity filter order-disorder transitions.
Sci Adv, 6, 2020

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