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PDB: 51630 件

5ZWE
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Covalent bond formation between histidine of Vitamin D receptor (VDR) and a full agonist having a vinyl ketone group via conjugate addition reaction
分子名称: (6R)-6-[(1R,3aS,4E,7aR)-7a-methyl-4-[2-[(3R,5R)-4-methylidene-3,5-bis(oxidanyl)cyclohexylidene]ethylidene]-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]hept-1-en-3-one, 13-meric peptide from DRIP205 NR2 BOX peptide, Vitamin D3 receptor
著者Yoshizawa, M, Itoh, T, Anami, Y, Kato, A, Yoshimoto, N, Yamamoto, K.
登録日2018-05-15
公開日2018-07-18
最終更新日2018-08-08
実験手法X-RAY DIFFRACTION (2.72 Å)
主引用文献Identification of the Histidine Residue in Vitamin D Receptor That Covalently Binds to Electrophilic Ligands
J. Med. Chem., 61, 2018
6AJA
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Crystal structure of Trypanosoma brucei glycosomal isocitrate dehydrogenase in complex with NADPH, alpha-ketoglutarate and ca2+
分子名称: 2-OXOGLUTARIC ACID, CALCIUM ION, GLYCEROL, ...
著者Wang, X, Inaoka, D.K, Shiba, T, Balogun, E.O, Ziebart, N, Allman, S, Watanabe, Y, Nozaki, T, Boshart, M, Bringaud, F, Harada, S, Kita, K.
登録日2018-08-27
公開日2019-08-28
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Biochemical characterization of a novel Trypanosoma brucei glycosomal isocitrate dehydrogenase with dual coenzyme specificity (NADP+/NAD+)
To Be Published
5ZYP
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Structure of the Yeast Ctr9/Paf1 complex
分子名称: NICKEL (II) ION, RNA polymerase-associated protein CTR9,RNA polymerase II-associated protein 1
著者Xie, Y, Zheng, M, Zhou, H, Long, J.
登録日2018-05-28
公開日2018-09-26
最終更新日2019-05-22
実験手法X-RAY DIFFRACTION (2.532 Å)
主引用文献Paf1 and Ctr9 subcomplex formation is essential for Paf1 complex assembly and functional regulation.
Nat Commun, 9, 2018
5ZZ9
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Crystal structure of Homer2 EVH1/Drebrin PPXXF complex
分子名称: Homer protein homolog 2, Peptide from Drebrin
著者Li, Z, Liu, H, Li, J, Liu, W, Zhang, M.
登録日2018-05-31
公開日2018-12-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Homer Tetramer Promotes Actin Bundling Activity of Drebrin.
Structure, 27, 2019
6R8H
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Triosephosphate isomerase from liver fluke (Fasciola hepatica).
分子名称: SULFATE ION, Triosephosphate isomerase
著者Ferraro, F, Corvo, I, Bergalli, L, Ilarraz, A, Cabrera, M, Gil, J, Susuki, B, Caffrey, C, Timson, D.J, Robert, X, Guillon, C, Alvarez, G.
登録日2019-04-01
公開日2020-02-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Novel and selective inactivators of Triosephosphate isomerase with anti-trematode activity.
Sci Rep, 10, 2020
1A12
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REGULATOR OF CHROMOSOME CONDENSATION (RCC1) OF HUMAN
分子名称: REGULATOR OF CHROMOSOME CONDENSATION 1
著者Renault, L, Nassar, N, Vetter, I, Becker, J, Roth, M, Wittinghofer, A.
登録日1997-12-19
公開日1999-01-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The 1.7 A crystal structure of the regulator of chromosome condensation (RCC1) reveals a seven-bladed propeller.
Nature, 392, 1998
8TC1
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Cryo-EM Structure of Spike Glycoprotein from Civet Coronavirus 007 in Closed Conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, LINOLEIC ACID, ...
著者Bostina, M, Hills, F.R, Eruera, A.R.
登録日2023-06-29
公開日2024-05-01
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (1.92 Å)
主引用文献Variation in structural motifs within SARS-related coronavirus spike proteins.
Plos Pathog., 20, 2024
6AK1
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Crystal structure of DmoA from Hyphomicrobium sulfonivorans
分子名称: Dimethyl-sulfide monooxygenase
著者Cao, H.Y, Wang, P, Peng, M, Li, C.Y.
登録日2018-08-28
公開日2018-12-12
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.284 Å)
主引用文献Crystal structure of the dimethylsulfide monooxygenase DmoA from Hyphomicrobium sulfonivorans.
Acta Crystallogr.,Sect.F, 74, 2018
6AKO
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Crystal Structure of FOXC2 DBD Bound to DBE2 DNA
分子名称: DNA (5'-D(CP*AP*AP*AP*AP*TP*GP*TP*AP*AP*AP*CP*AP*AP*GP*A)-3'), DNA (5'-D(TP*CP*TP*TP*GP*TP*TP*TP*AP*CP*AP*TP*TP*TP*TP*G)-3'), Forkhead box protein C2, ...
著者Chen, X, Wei, H, Li, J, Liang, X, Dai, S, Jiang, L, Guo, M, Chen, Y.
登録日2018-09-03
公開日2019-02-06
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.396 Å)
主引用文献Structural basis for DNA recognition by FOXC2.
Nucleic Acids Res., 47, 2019
8TC0
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Cryo-EM Structure of Spike Glycoprotein from Bat Coronavirus WIV1 in Closed Conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bostina, M, Hills, F.R, Eruera, A.
登録日2023-06-29
公開日2024-05-01
最終更新日2024-06-26
実験手法ELECTRON MICROSCOPY (1.88 Å)
主引用文献Variation in structural motifs within SARS-related coronavirus spike proteins.
Plos Pathog., 20, 2024
6RBR
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BU of 6rbr by Molmil
Crystal structure of NAD kinase 1 from Listeria monocytogenes in complexe with an adenine derivative
分子名称: 8-bromanyl-9-ethyl-purin-6-amine, CITRIC ACID, NAD kinase 1
著者Gelin, M, Labesse, G.
登録日2019-04-11
公開日2020-02-19
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献From Substrate to Fragments to Inhibitor ActiveIn VivoagainstStaphylococcus aureus.
Acs Infect Dis., 6, 2020
6RC2
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BU of 6rc2 by Molmil
Crystal structure of NAD kinase 1 from Listeria monocytogenes in complexe with an adenine derivative
分子名称: 8-methyl-9-pent-4-ynyl-purin-6-amine, CITRIC ACID, NAD kinase 1
著者Gelin, M, Labesse, G.
登録日2019-04-11
公開日2020-02-19
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.048 Å)
主引用文献From Substrate to Fragments to Inhibitor ActiveIn VivoagainstStaphylococcus aureus.
Acs Infect Dis., 6, 2020
5ZUJ
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BU of 5zuj by Molmil
Binding and Enhanced Binding between Key Immunity Proteins TRAF6 and TIFA
分子名称: TNF receptor-associated factor 6, peptide 170-184 from TRAF-interacting protein with FHA domain-containing protein A
著者Huang, W.C, Maestre-Reyna, M, Hsiao, T.C, Tsai, M.D.
登録日2018-05-07
公開日2018-12-05
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Binding and Enhanced Binding between Key Immunity Proteins TRAF6 and TIFA.
Chembiochem, 20, 2019
6RD3
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BU of 6rd3 by Molmil
Crystal structure of the wild type OmpK36 from Klebsiella pneumonia
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, MAGNESIUM ION, OmpK36
著者Beis, K, Romano, M, Kwong, J.
登録日2019-04-12
公開日2019-09-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献OmpK36-mediated Carbapenem resistance attenuates ST258 Klebsiella pneumoniae in vivo.
Nat Commun, 10, 2019
165L
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BU of 165l by Molmil
CONTROL OF ENZYME ACTIVITY BY AN ENGINEERED DISULFIDE BOND
分子名称: BETA-MERCAPTOETHANOL, CHLORIDE ION, T4 LYSOZYME
著者Blaber, M, Matthews, B.W.
登録日1994-06-20
公開日1994-08-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Alanine scanning mutagenesis of the alpha-helix 115-123 of phage T4 lysozyme: effects on structure, stability and the binding of solvent.
J.Mol.Biol., 246, 1995
6AB9
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The crystal structure of the relaxed state of Nonlabens marinus Rhodopsin 3
分子名称: CHLORIDE ION, Chloride pumping rhodopsin, OLEIC ACID, ...
著者Yun, J.-H, Ohki, M, Park, J.-H, Jin, Z, Lee, W, Liu, H, Tame, J.R.H, Shibayama, N, Park, S.-Y.
登録日2018-07-20
公開日2019-07-31
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The pumping mechanism of NM-R3, a light-driven cyanobacterial chloride importer in the rhodopsin family
To Be Published
5ZUY
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Crystal structure of E134H mutant of phosphomannose isomerase from Salmonella typhimurium
分子名称: 1,2-ETHANEDIOL, Mannose-6-phosphate isomerase
著者Bangera, M, Murthy, M.R.N.
登録日2018-05-08
公開日2019-05-01
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and functional insights into phosphomannose isomerase: the role of zinc and catalytic residues.
Acta Crystallogr D Struct Biol, 75, 2019
6ABM
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Crystal structure of Methanosarcina mazei PylRS(Y306A/Y384F) complexed with pTmdZLys
分子名称: (2S)-2-azanyl-6-[[4-[3-(trifluoromethyl)-1,2-diazirin-3-yl]phenyl]methoxycarbonylamino]hexanoic acid, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Yanagisawa, T, Kuratani, M, Yokoyama, S.
登録日2018-07-22
公開日2019-04-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.368 Å)
主引用文献Structural Basis for Genetic-Code Expansion with Bulky Lysine Derivatives by an Engineered Pyrrolysyl-tRNA Synthetase.
Cell Chem Biol, 26, 2019
1A22
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BU of 1a22 by Molmil
HUMAN GROWTH HORMONE BOUND TO SINGLE RECEPTOR
分子名称: GROWTH HORMONE, GROWTH HORMONE RECEPTOR
著者De Vos, A.M, Ultsch, M.
登録日1998-01-15
公開日1998-04-29
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural and functional analysis of the 1:1 growth hormone:receptor complex reveals the molecular basis for receptor affinity.
J.Mol.Biol., 277, 1998
6ADE
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BU of 6ade by Molmil
Crystal structure of phosphorylated mutant of glyceraldehyde 3-phosphate dehydrogenase from human placenta at 3.15A resolution
分子名称: Glyceraldehyde-3-phosphate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Dilawari, R, Singh, P.K, Raje, M, Sharma, S, Singh, T.P.
登録日2018-07-31
公開日2018-08-22
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Crystal structure of phosphorylated mutant of glyceraldehyde 3-phosphate dehydrogenase from human placenta at 3.15A resolution
To Be Published
8TC5
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Cryo-EM Structure of Spike Glycoprotein from Civet Coronavirus SZ3 in Closed Conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Bostina, M, Hills, F.R, Eruera, A.
登録日2023-06-29
公開日2024-05-15
最終更新日2024-06-12
実験手法ELECTRON MICROSCOPY (2.11 Å)
主引用文献Variation in structural motifs within SARS-related coronavirus spike proteins.
Plos Pathog., 20, 2024
6RBX
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BU of 6rbx by Molmil
Crystal structure of NAD kinase 1 from Listeria monocytogenes in complexe with an adenine derivative
分子名称: 3-(6-azanyl-8-bromanyl-purin-9-yl)propan-1-ol, CITRIC ACID, NAD kinase 1
著者Gelin, M, Labesse, G.
登録日2019-04-11
公開日2020-02-19
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献From Substrate to Fragments to Inhibitor ActiveIn VivoagainstStaphylococcus aureus.
Acs Infect Dis., 6, 2020
6AKK
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Crystal structure of the second Coiled-coil domain of SIKE1
分子名称: GLYCEROL, Suppressor of IKBKE 1
著者Zhou, L, Chen, M, Zhou, Z.C.
登録日2018-09-02
公開日2019-01-16
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Architecture, substructures, and dynamic assembly of STRIPAK complexes in Hippo signaling.
Cell Discov, 5, 2019
8TI5
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Crystal structure of Tyr p 36.0101
分子名称: Profilin, SULFATE ION
著者O'Malley, A, Sankaran, S, Chruszcz, M.
登録日2023-07-19
公開日2024-05-08
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Structural homology of mite profilins to plant profilins is not indicative of allergic cross-reactivity.
Biol.Chem., 405, 2024
8TI6
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Crystal structure of Tyr p 36.0101
分子名称: Profilin, Proline-rich peptide, SULFATE ION
著者O'Malley, A, Sankaran, S, Chruszcz, M.
登録日2023-07-19
公開日2024-05-08
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Structural homology of mite profilins to plant profilins is not indicative of allergic cross-reactivity.
Biol.Chem., 405, 2024

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