4GP7
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![BU of 4gp7 by Molmil](/molmil-images/mine/4gp7) | Polynucleotide kinase | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, CITRIC ACID, MAGNESIUM ION, ... | 著者 | Wang, L.K, Das, U, Smith, P, Shuman, S. | 登録日 | 2012-08-20 | 公開日 | 2012-11-14 | 最終更新日 | 2017-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure and mechanism of the polynucleotide kinase component of the bacterial Pnkp-Hen1 RNA repair system. Rna, 18, 2012
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4GQR
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![BU of 4gqr by Molmil](/molmil-images/mine/4gqr) | Human Pancreatic alpha-amylase in complex with myricetin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 3,5,7-TRIHYDROXY-2-(3,4,5-TRIHYDROXYPHENYL)-4H-CHROMEN-4-ONE, CALCIUM ION, ... | 著者 | Williams, L.K, Brayer, G.D. | 登録日 | 2012-08-23 | 公開日 | 2012-10-24 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Order and disorder: differential structural impacts of myricetin and ethyl caffeate on human amylase, an antidiabetic target. J.Med.Chem., 55, 2012
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2AQU
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![BU of 2aqu by Molmil](/molmil-images/mine/2aqu) | Structure of HIV-1 protease bound to atazanavir | 分子名称: | (3S,8S,9S,12S)-3,12-BIS(1,1-DIMETHYLETHYL)-8-HYDROXY-4,11-DIOXO-9-(PHENYLMETHYL)-6-[[4-(2-PYRIDINYL)PHENYL]METHYL]-2,5, 6,10,13-PENTAAZATETRADECANEDIOIC ACID DIMETHYL ESTER, HIV-1 Protease | 著者 | Clemente, J.C, Coman, R.M, Thiaville, M.M, Janka, L.K, Jeung, J.A, Nukoolkarn, S, Govindasamy, L, Agbandje-McKenna, M, McKenna, R, Leelamanit, W, Goodenow, M.M, Dunn, B.M. | 登録日 | 2005-08-18 | 公開日 | 2006-08-29 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Analysis of HIV-1 CRF_01 A/E protease inhibitor resistance: structural determinants for maintaining sensitivity and developing resistance to atazanavir. Biochemistry, 45, 2006
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4GP6
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![BU of 4gp6 by Molmil](/molmil-images/mine/4gp6) | Polynucleotide kinase | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Metallophosphoesterase | 著者 | Wang, L.K, Das, U, Smith, P, Shuman, S. | 登録日 | 2012-08-20 | 公開日 | 2012-11-14 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure and mechanism of the polynucleotide kinase component of the bacterial Pnkp-Hen1 RNA repair system. Rna, 18, 2012
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1D4L
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![BU of 1d4l by Molmil](/molmil-images/mine/1d4l) | HIV-1 PROTEASE COMPLEXED WITH A MACROCYCLIC PEPTIDOMIMETIC INHIBITOR | 分子名称: | (10S,13S,1'R)-13-[1'-HYDROXY-2'-(N-P-AMINOBENZENESULFONYL-1''-AMINO-3''-METHYLBUTYL)ETHYL]-8,11-DIOXO-10-ISOPROPYL-2-OXA-9,12-DIAZABICYCLO [13.2.2]NONADECA-15,17,18-TRIENE, HIV-1 PROTEASE, SULFATE ION | 著者 | Tyndall, J.D, Reid, R.C, Tyssen, D.P, Jardine, D.K, Todd, B, Passmore, M, March, D.R, Pattenden, L.K, Alewood, D, Hu, S.H, Alewood, P.F, Birch, C.J, Martin, J.L, Fairlie, D.P. | 登録日 | 1999-10-04 | 公開日 | 2000-10-11 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease. J.Med.Chem., 43, 2000
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4GQQ
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1MVY
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![BU of 1mvy by Molmil](/molmil-images/mine/1mvy) | Amylosucrase mutant E328Q co-crystallized with maltoheptaose. | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, ... | 著者 | Skov, L.K, Mirza, O, Sprogoe, D, Dar, I, Remaud-Simeon, M, Albenne, C, Monsan, P, Gajhede, M. | 登録日 | 2002-09-27 | 公開日 | 2002-12-18 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Oligosaccharide and Sucrose Complexes of Amylosucrase. STRUCTURAL IMPLICATIONS FOR THE POLYMERASE ACTIVITY J.BIOL.CHEM., 277, 2002
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1MW1
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![BU of 1mw1 by Molmil](/molmil-images/mine/1mw1) | Amylosucrase soaked with 14mM sucrose. | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, amylosucrase, beta-D-fructofuranose-(2-1)-alpha-D-glucopyranose | 著者 | Skov, L.K, Mirza, O, Sprogoe, D, Dar, I, Remaud-Simeon, M, Albenne, C, Monsan, P, Gajhede, M. | 登録日 | 2002-09-27 | 公開日 | 2002-12-18 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Oligosaccharide and Sucrose Complexes of Amylosucrase. STRUCTURAL IMPLICATIONS FOR THE POLYMERASE ACTIVITY J.BIOL.CHEM., 277, 2002
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1D4K
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![BU of 1d4k by Molmil](/molmil-images/mine/1d4k) | HIV-1 PROTEASE COMPLEXED WITH A MACROCYCLIC PEPTIDOMIMETIC INHIBITOR | 分子名称: | HIV-1 PROTEASE, N-13-[(10S,13S)-9,12-DIOXO-10-(2-BUTYL)-2-OXA-8,11-DIAZABICYCLO [13.2.2] NONADECA-15,17,18-TRIENE] (2R)-BENZYL-(4S)-HYDROXY-5-AMINOPENTANOIC (1R)-HYDROXY-(2S)-INDANEAMIDE, SULFATE ION | 著者 | Tyndall, J.D, Reid, R.C, Tyssen, D.P, Jardine, D.K, Todd, B, Passmore, M, March, D.R, Pattenden, L.K, Alewood, D, Hu, S.H, Alewood, P.F, Birch, C.J, Martin, J.L, Fairlie, D.P. | 登録日 | 1999-10-04 | 公開日 | 2000-10-11 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease. J.Med.Chem., 43, 2000
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2B7Z
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![BU of 2b7z by Molmil](/molmil-images/mine/2b7z) | Structure of HIV-1 protease mutant bound to indinavir | 分子名称: | HIV-1 protease, N-[2(R)-HYDROXY-1(S)-INDANYL]-5-[(2(S)-TERTIARY BUTYLAMINOCARBONYL)-4(3-PYRIDYLMETHYL)PIPERAZINO]-4(S)-HYDROXY-2(R)-PHENYLMETHYLPENTANAMIDE | 著者 | Clemente, J.C, Stow, L.R, Janka, L.K, Jeung, J.A, Desai, K.A, Govindasamy, L, Agbandje-McKenna, M, McKenna, R, Goodenow, M.M, Dunn, B.M. | 登録日 | 2005-10-05 | 公開日 | 2006-11-14 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | In vivo, kinetic, and structural analysis of the development of ritonavir resistance To be Published
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2B60
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![BU of 2b60 by Molmil](/molmil-images/mine/2b60) | Structure of HIV-1 protease mutant bound to Ritonavir | 分子名称: | GLYCEROL, Gag-Pol polyprotein, RITONAVIR | 著者 | Clemente, J.C, Stow, L.R, Janka, L.K, Jeung, J.A, Desai, K.A, Govindasamy, L, Agbandje-McKenna, M, McKenna, R, Goodenow, M.M, Dunn, B.M. | 登録日 | 2005-09-29 | 公開日 | 2006-11-14 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | In vivo, kinetic, and structural analysis of the development of ritonavir resistance To be Published
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2ATM
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![BU of 2atm by Molmil](/molmil-images/mine/2atm) | Crystal structure of the recombinant allergen Ves v 2 | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Hyaluronoglucosaminidase, SULFATE ION | 著者 | Skov, L.K, Seppala, U, Coen, J.J.F, Crickmore, N, King, T.P, Monsalve, R, Kastrup, J.S, Spangfort, M.D, Gajhede, M. | 登録日 | 2005-08-25 | 公開日 | 2006-05-23 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of recombinant Ves v 2 at 2.0 Angstrom resolution: structural analysis of an allergenic hyaluronidase from wasp venom. Acta Crystallogr.,Sect.D, 62, 2006
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4JT2
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![BU of 4jt2 by Molmil](/molmil-images/mine/4jt2) | Structure of Clostridium thermocellum polynucleotide kinase bound to CTP | 分子名称: | CYTIDINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Metallophosphoesterase | 著者 | Das, U, Wang, L.K, Smith, P, Shuman, S. | 登録日 | 2013-03-22 | 公開日 | 2013-08-28 | 最終更新日 | 2013-12-18 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Structural and biochemical analysis of the phosphate donor specificity of the polynucleotide kinase component of the bacterial pnkphen1 RNA repair system. Biochemistry, 52, 2013
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2FAQ
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![BU of 2faq by Molmil](/molmil-images/mine/2faq) | Crystal Structure of Pseudomonas aeruginosa LigD polymerase domain with ATP and Manganese | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, SULFATE ION, ... | 著者 | Zhu, H, Nandakumar, J, Aniukwu, J, Wang, L.K, Glickman, M.S, Lima, C.D, Shuman, S. | 登録日 | 2005-12-07 | 公開日 | 2006-05-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Atomic structure and nonhomologous end-joining function of the polymerase component of bacterial DNA ligase D Proc.Natl.Acad.Sci.USA, 103, 2006
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2FAO
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![BU of 2fao by Molmil](/molmil-images/mine/2fao) | Crystal Structure of Pseudomonas aeruginosa LigD polymerase domain | 分子名称: | SULFATE ION, probable ATP-dependent DNA ligase | 著者 | Zhu, H, Nandakumar, J, Aniukwu, J, Wang, L.K, Glickman, M.S, Lima, C.D, Shuman, S. | 登録日 | 2005-12-07 | 公開日 | 2006-05-23 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Atomic structure and nonhomologous end-joining function of the polymerase component of bacterial DNA ligase D Proc.Natl.Acad.Sci.USA, 103, 2006
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1QP1
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![BU of 1qp1 by Molmil](/molmil-images/mine/1qp1) | KAPPA VARIABLE LIGHT CHAIN | 分子名称: | BENCE-JONES KAPPA I ANTIBODY BRE (LIGHT CHAIN) | 著者 | Steinrauf, L.K. | 登録日 | 1999-05-30 | 公開日 | 1999-06-17 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Molecular structure of the amyloid-forming protein kappa I Bre. J.Biochem.(Tokyo), 125, 1999
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4JT4
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![BU of 4jt4 by Molmil](/molmil-images/mine/4jt4) | Structure of Clostridium thermocellum polynucleotide kinase bound to dATP | 分子名称: | 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, MAGNESIUM ION, Metallophosphoesterase, ... | 著者 | Das, U, Wang, L.K, Smith, P, Shuman, S. | 登録日 | 2013-03-22 | 公開日 | 2013-08-28 | 最終更新日 | 2013-12-18 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Structural and biochemical analysis of the phosphate donor specificity of the polynucleotide kinase component of the bacterial pnkphen1 RNA repair system. Biochemistry, 52, 2013
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4JSY
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![BU of 4jsy by Molmil](/molmil-images/mine/4jsy) | Structure of Clostridium thermocellum polynucleotide kinase bound to GTP | 分子名称: | GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Metallophosphoesterase | 著者 | Das, U, Wang, L.K, Smith, P, Shuman, S. | 登録日 | 2013-03-22 | 公開日 | 2013-08-28 | 最終更新日 | 2013-12-18 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Structural and biochemical analysis of the phosphate donor specificity of the polynucleotide kinase component of the bacterial pnkphen1 RNA repair system. Biochemistry, 52, 2013
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2FAR
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![BU of 2far by Molmil](/molmil-images/mine/2far) | Crystal Structure of Pseudomonas aeruginosa LigD polymerase domain with dATP and Manganese | 分子名称: | 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, MANGANESE (II) ION, SULFATE ION, ... | 著者 | Zhu, H, Nandakumar, J, Aniukwu, J, Wang, L.K, Glickman, M.S, Lima, C.D, Shuman, S. | 登録日 | 2005-12-07 | 公開日 | 2006-05-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Atomic structure and nonhomologous end-joining function of the polymerase component of bacterial DNA ligase D Proc.Natl.Acad.Sci.USA, 103, 2006
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4C7A
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![BU of 4c7a by Molmil](/molmil-images/mine/4c7a) | Crystal structure of the Smoothened CRD, selenomethionine-labeled | 分子名称: | SMOOTHENED, SODIUM ION, ZINC ION | 著者 | Nachtergaele, S, Whalen, D.M, Mydock, L.K, Zhao, Z, Malinauskas, T, Krishnan, K, Ingham, P.W, Covey, D.F, Rohatgi, R, Siebold, C. | 登録日 | 2013-09-20 | 公開日 | 2013-11-06 | 最終更新日 | 2013-11-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure and Function of the Smoothened Extracellular Domain in Vertebrate Hedgehog Signaling Elife, 2, 2013
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2R2J
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![BU of 2r2j by Molmil](/molmil-images/mine/2r2j) | crystal structure of human ERp44 | 分子名称: | FORMIC ACID, SUCCINIC ACID, Thioredoxin domain-containing protein 4 | 著者 | Wang, L.K, Li, S.J, Sun, F, Wang, C.C. | 登録日 | 2007-08-25 | 公開日 | 2008-07-08 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of human ERp44 shows a dynamic functional modulation by its carboxy-terminal tail. Embo Rep., 2008
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4OQY
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![BU of 4oqy by Molmil](/molmil-images/mine/4oqy) | Streptomyces sp. GF3546 imine reductase | 分子名称: | (S)-imine reductase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Schneider, L.K, Huber, T, Gerhardt, S, Muller, M, Einsle, O. | 登録日 | 2014-02-10 | 公開日 | 2014-10-22 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Direct Reductive Amination of Ketones: Structure and Activity of S-Selective Imine Reductases from Streptomyces. CHEMCATCHEM, 2014
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2LCZ
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4CPF
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![BU of 4cpf by Molmil](/molmil-images/mine/4cpf) | Wild-type streptavidin in complex with love-hate ligand 3 (LH3) | 分子名称: | STREPTAVIDIN, methyl 4-(2-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H- thieno[3,4-d]imidazolidin-4-yl]pentanehydrazido}-3- [4-(methoxycarbonyl)phenyl]phenyl)benzoate | 著者 | Fairhead, M, Shen, D, Chan, L.K.M, Lowe, E.D, Donohoe, T.J, Howarth, M. | 登録日 | 2014-02-06 | 公開日 | 2014-08-06 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | Love-Hate Ligands for High Resolution Analysis of Strain in Ultra-Stable Protein/Small Molecule Interaction. Bioorg.Med.Chem., 22, 2014
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2M8R
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![BU of 2m8r by Molmil](/molmil-images/mine/2m8r) | |