2E0A
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![BU of 2e0a by Molmil](/molmil-images/mine/2e0a) | Crystal structure of human pyruvate dehydrogenase kinase 4 in complex with AMPPNP | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Pyruvate dehydrogenase kinase isozyme 4 | 著者 | Kukimoto-Niino, M, Tokmakov, A, Terada, T, Shiromizu, I, Kawamoto, M, Matsusue, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-10-03 | 公開日 | 2007-10-09 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr.,Sect.D, 67, 2011
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2DWG
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![BU of 2dwg by Molmil](/molmil-images/mine/2dwg) | RUN domain of Rap2 interacting protein x, crystallized in P2(1)2(1)2(1) space group | 分子名称: | Protein RUFY3 | 著者 | Kukimoto-Niino, M, Murayama, K, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-08-11 | 公開日 | 2006-10-24 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.22 Å) | 主引用文献 | Crystal Structure of the RUN Domain of the RAP2-interacting Protein x J.Biol.Chem., 281, 2006
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2E87
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![BU of 2e87 by Molmil](/molmil-images/mine/2e87) | Crystal structure of hypothetical GTP-binding protein PH1320 from Pyrococcus horikoshii OT3, in complex with GDP | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, Hypothetical protein PH1320, SULFATE ION | 著者 | Kukimoto-Niino, M, Bessho, Y, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2007-01-19 | 公開日 | 2007-07-24 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Crystal structure of hypothetical GTP-binding protein PH1320 from Pyrococcus horikoshii OT3, in complex with GDP To be Published
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2CXF
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![BU of 2cxf by Molmil](/molmil-images/mine/2cxf) | RUN domain of Rap2 interacting protein x, crystallized in C2 space group | 分子名称: | rap2 interacting protein x | 著者 | Kukimoto-Niino, M, Murayama, K, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-06-29 | 公開日 | 2005-12-29 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (3.07 Å) | 主引用文献 | Crystal Structure of the RUN Domain of the RAP2-interacting Protein x J.Biol.Chem., 281, 2006
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2CXL
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![BU of 2cxl by Molmil](/molmil-images/mine/2cxl) | RUN domain of Rap2 interacting protein x, crystallized in I422 space group | 分子名称: | rap2 interacting protein x | 著者 | Kukimoto-Niino, M, Umehara, T, Murayama, K, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-06-30 | 公開日 | 2005-12-30 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Crystal Structure of the RUN Domain of the RAP2-interacting Protein x J.Biol.Chem., 281, 2006
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2DWK
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![BU of 2dwk by Molmil](/molmil-images/mine/2dwk) | Crystal structure of the RUN domain of mouse Rap2 interacting protein x | 分子名称: | Protein RUFY3 | 著者 | Kukimoto-Niino, M, Murayama, K, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-08-15 | 公開日 | 2006-08-29 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structure of the RUN Domain of the RAP2-interacting Protein x J.Biol.Chem., 281, 2006
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2CXX
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2DBY
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![BU of 2dby by Molmil](/molmil-images/mine/2dby) | Crystal structure of the GTP-binding protein YchF in complexed with GDP | 分子名称: | FORMIC ACID, GTP-binding protein, GUANOSINE-5'-DIPHOSPHATE | 著者 | Kukimoto-Niino, M, Murayama, K, Shirouzu, M, Kuramitsu, S, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-12-16 | 公開日 | 2006-06-16 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Crystal structure of the GTP-binding protein YchF in complexed with GDP To be Published
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2DWQ
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![BU of 2dwq by Molmil](/molmil-images/mine/2dwq) | Thermus thermophilus YchF GTP-binding protein | 分子名称: | GTP-binding protein | 著者 | Kukimoto-Niino, M, Murayama, K, Shorouzu, M, Kuramitsu, S, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-08-16 | 公開日 | 2007-02-16 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Thermus thermophilus YchF GTP-binding protein To be Published
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2DYL
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![BU of 2dyl by Molmil](/molmil-images/mine/2dyl) | Crystal structure of human mitogen-activated protein kinase kinase 7 activated mutant (S287D, T291D) | 分子名称: | Dual specificity mitogen-activated protein kinase kinase 7 | 著者 | Kukimoto-Niino, M, Takagi, T, Kaminishi, T, Uchikubo-Kamo, T, Terada, T, Matsuzaki, O, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-09-15 | 公開日 | 2007-08-28 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of human mitogen-activated protein kinase kinase 7 activated mutant (S287D, T291D) To be Published
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2DWB
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![BU of 2dwb by Molmil](/molmil-images/mine/2dwb) | Aurora-A kinase complexed with AMPPNP | 分子名称: | PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, SULFATE ION, Serine/threonine-protein kinase 6 | 著者 | Kukimoto-Niino, M, Murayama, K, Shirouzu, S, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2006-08-10 | 公開日 | 2007-07-31 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Aurora-A kinase complexed with AMPPNP To be Published
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3WU4
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![BU of 3wu4 by Molmil](/molmil-images/mine/3wu4) | Oxidized-form structure of E.coli Lon Proteolytic domain | 分子名称: | Lon protease, SULFATE ION | 著者 | Nishii, W, Kukimoto-Niino, M, Terada, T, Shirouzu, M, Muramatsu, T, Yokoyama, S. | 登録日 | 2014-04-22 | 公開日 | 2014-11-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A redox switch shapes the Lon protease exit pore to facultatively regulate proteolysis. Nat. Chem. Biol., 11, 2015
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5CWZ
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5GV3
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![BU of 5gv3 by Molmil](/molmil-images/mine/5gv3) | Crystal structure of the membrane-distal domain of mouse lysosome-associated membrane protein 2 (LAMP-2) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Lysosome-associated membrane glycoprotein 2, ZINC ION | 著者 | Tomabechi, Y, Ehara, H, Kukimoto-Niino, M, Shirouzu, M. | 登録日 | 2016-09-01 | 公開日 | 2017-09-06 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.096 Å) | 主引用文献 | Lysosome-associated membrane proteins-1 and -2 (LAMP-1 and LAMP-2) assemble via distinct modes. Biochem. Biophys. Res. Commun., 479, 2016
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6JPP
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7Y4A
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![BU of 7y4a by Molmil](/molmil-images/mine/7y4a) | Crystal structure of human ELMO1 RBD-RhoG complex | 分子名称: | Engulfment and cell motility protein 1, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Tsuda, K, Kukimoto-Niino, M, Shirouzu, M. | 登録日 | 2022-06-14 | 公開日 | 2023-03-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Targeting Ras-binding domain of ELMO1 by computational nanobody design. Commun Biol, 6, 2023
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7XN1
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![BU of 7xn1 by Molmil](/molmil-images/mine/7xn1) | Crystal structure of human acetylcholinesterase in complex with tacrine | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, Acetylcholinesterase, ... | 著者 | Dileep, K.V, Ihara, K, Mishima-Tsumagari, C, Kukimoto-Niino, M, Yonemochi, M, Hanada, K, Shirouzu, M, Zhang, K.Y.J. | 登録日 | 2022-04-27 | 公開日 | 2023-03-01 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery Int.J.Biol.Macromol., 210, 2022
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2PSM
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![BU of 2psm by Molmil](/molmil-images/mine/2psm) | Crystal structure of Interleukin 15 in complex with Interleukin 15 receptor alpha | 分子名称: | BENZAMIDINE, Interleukin-15, Interleukin-15 receptor alpha chain | 著者 | Olsen, S.K, Murayama, K, Kishishita, S, Kukimoto-Niino, M, Terada, T, Shirouzu, M, Ota, N, Kanagawa, O, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2007-05-07 | 公開日 | 2007-11-06 | 最終更新日 | 2021-08-18 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Crystal Structure of the Interleukin-15{middle dot}Interleukin-15 Receptor {alpha} Complex: INSIGHTS INTO TRANS AND CIS PRESENTATION J.Biol.Chem., 282, 2007
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5AX9
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![BU of 5ax9 by Molmil](/molmil-images/mine/5ax9) | Crystal structure of the kinase domain of human TRAF2 and NCK-interacting protein kinase in complex with compund 9 | 分子名称: | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile, SULFATE ION, TRAF2 and NCK-interacting protein kinase | 著者 | Ohbayashi, N, Kukimoto-Niino, M, Yamada, T, Shirouzu, M. | 登録日 | 2015-07-21 | 公開日 | 2016-07-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | TNIK inhibition abrogates colorectal cancer stemness Nat Commun, 7, 2016
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5D7A
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![BU of 5d7a by Molmil](/molmil-images/mine/5d7a) | Crystal structure of the kinase domain of TRAF2 and NCK-interacting protein kinase with NCB-0846 | 分子名称: | SULFATE ION, TRAF2 and NCK-interacting protein kinase, cis-4-{[2-(1H-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | 著者 | Ohbayashi, N, Kukimoto-Niino, M, Yamada, T, Shirouzu, M. | 登録日 | 2015-08-13 | 公開日 | 2016-08-17 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | TNIK inhibition abrogates colorectal cancer stemness Nat Commun, 7, 2016
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5ZJ6
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![BU of 5zj6 by Molmil](/molmil-images/mine/5zj6) | Crystal structure of HCK kinase complexed with a pyrrolo-pyrimidine inhibitor 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine | 分子名称: | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine, Tyrosine-protein kinase HCK | 著者 | Tomabechi, Y, Kukimoto-Niino, M, Shirouzu, M. | 登録日 | 2018-03-19 | 公開日 | 2018-06-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.696 Å) | 主引用文献 | Phosphorylated and non-phosphorylated HCK kinase domains produced by cell-free protein expression. Protein Expr. Purif., 150, 2018
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7E3H
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![BU of 7e3h by Molmil](/molmil-images/mine/7e3h) | Crystal structure of human acetylcholinesterase in complex with donepezil | 分子名称: | 1-BENZYL-4-[(5,6-DIMETHOXY-1-INDANON-2-YL)METHYL]PIPERIDINE, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholinesterase | 著者 | Dileep, K.V, Ihara, K, Mishima-Tsumagari, C, Kukimoto-Niino, M, Yonemochi, M, Hanada, K, Shirouzu, M, Zhang, K.Y.J. | 登録日 | 2021-02-08 | 公開日 | 2022-02-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery Int.J.Biol.Macromol., 210, 2022
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7E3D
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![BU of 7e3d by Molmil](/molmil-images/mine/7e3d) | Crystal structure of human acetylcholinesterase | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, Acetylcholinesterase | 著者 | Dileep, K.V, Ihara, K, Mishima-Tsumagari, C, Kukimoto-Niino, M, Yonemochi, M, Hanada, K, Shirouzu, M, Zhang, K.Y.J. | 登録日 | 2021-02-08 | 公開日 | 2022-02-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of human acetylcholinesterase in complex with tacrine: Implications for drug discovery Int.J.Biol.Macromol., 210, 2022
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5GV0
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![BU of 5gv0 by Molmil](/molmil-images/mine/5gv0) | Crystal structure of the membrane-proximal domain of mouse lysosome-associated membrane protein 1 (LAMP-1) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Lysosome-associated membrane glycoprotein 1, SULFATE ION | 著者 | Tomabechi, Y, Ehara, H, Kukimoto-Niino, M, Shirouzu, M. | 登録日 | 2016-09-01 | 公開日 | 2016-10-12 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Lysosome-associated membrane proteins-1 and -2 (LAMP-1 and LAMP-2) assemble via distinct modes Biochem.Biophys.Res.Commun., 479, 2016
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3A99
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![BU of 3a99 by Molmil](/molmil-images/mine/3a99) | Structure of PIM-1 kinase crystallized in the presence of P27KIP1 Carboxy-terminal peptide | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Proto-oncogene serine/threonine-protein kinase pim-1 | 著者 | Morishita, D, Takami, M, Yoshikawa, S, Katayama, R, Sato, S, Kukimoto-Niino, M, Umehara, T, Shirouzu, M, Sekimizu, K, Yokoyama, S, Fujita, N. | 登録日 | 2009-10-22 | 公開日 | 2010-11-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Cell-permeable carboxyl-terminal p27(Kip1) peptide exhibits anti-tumor activity by inhibiting Pim-1 kinase J.Biol.Chem., 286, 2011
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