3A99
Structure of PIM-1 kinase crystallized in the presence of P27KIP1 Carboxy-terminal peptide
Summary for 3A99
Entry DOI | 10.2210/pdb3a99/pdb |
Descriptor | Proto-oncogene serine/threonine-protein kinase pim-1, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... (4 entities in total) |
Functional Keywords | pim-1, p27kip1, peptide drug, prostate cancer, transferase |
Biological source | Homo sapiens (human) |
Cellular location | Isoform 2: Cytoplasm. Isoform 1: Cell membrane: P11309 |
Total number of polymer chains | 1 |
Total formula weight | 37013.89 |
Authors | Morishita, D.,Takami, M.,Yoshikawa, S.,Katayama, R.,Sato, S.,Kukimoto-Niino, M.,Umehara, T.,Shirouzu, M.,Sekimizu, K.,Yokoyama, S.,Fujita, N. (deposition date: 2009-10-22, release date: 2010-11-03, Last modification date: 2023-11-01) |
Primary citation | Morishita, D.,Takami, M.,Yoshikawa, S.,Katayama, R.,Sato, S.,Kukimoto-Niino, M.,Umehara, T.,Shirouzu, M.,Sekimizu, K.,Yokoyama, S.,Fujita, N. Cell-permeable carboxyl-terminal p27(Kip1) peptide exhibits anti-tumor activity by inhibiting Pim-1 kinase J.Biol.Chem., 286:2681-2688, 2011 Cited by PubMed: 21062737DOI: 10.1074/jbc.M109.092452 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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