4GH6
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![BU of 4gh6 by Molmil](/molmil-images/mine/4gh6) | Crystal structure of the PDE9A catalytic domain in complex with inhibitor 28 | 分子名称: | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, MAGNESIUM ION, N-(4-methoxyphenyl)-N~2~-[1-(2-methylphenyl)-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl]-L-alaninamide, ... | 著者 | Hou, J, Ke, H. | 登録日 | 2012-08-07 | 公開日 | 2012-10-03 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structure-Based Discovery of Highly Selective Phosphodiesterase-9A Inhibitors and Implications for Inhibitor Design. J.Med.Chem., 55, 2012
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1ZKN
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![BU of 1zkn by Molmil](/molmil-images/mine/1zkn) | Structure of PDE4D2-IBMX | 分子名称: | 3-ISOBUTYL-1-METHYLXANTHINE, MAGNESIUM ION, ZINC ION, ... | 著者 | Huai, Q, Liu, Y, Francis, S.H, Corbin, J.D, Ke, H. | 登録日 | 2005-05-03 | 公開日 | 2005-05-17 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal Structures of Phosphodiesterases 4 and 5 in Complex with Inhibitor 3-Isobutyl-1-Methylxanthine Suggest a Conformation Determinant of Inhibitor Selectivity J.Biol.Chem., 279, 2004
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1ZKL
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![BU of 1zkl by Molmil](/molmil-images/mine/1zkl) | Multiple Determinants for Inhibitor Selectivity of Cyclic Nucleotide Phosphodiesterases | 分子名称: | 3-ISOBUTYL-1-METHYLXANTHINE, High-affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A, MAGNESIUM ION, ... | 著者 | Wang, H, Liu, Y, Chen, Y, Robinson, H, Ke, H. | 登録日 | 2005-05-03 | 公開日 | 2005-07-05 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Multiple elements jointly determine inhibitor selectivity of cyclic nucleotide phosphodiesterases 4 and 7 J.Biol.Chem., 280, 2005
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1IAY
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![BU of 1iay by Molmil](/molmil-images/mine/1iay) | CRYSTAL STRUCTURE OF ACC SYNTHASE COMPLEXED WITH COFACTOR PLP AND INHIBITOR AVG | 分子名称: | 1-AMINOCYCLOPROPANE-1-CARBOXYLATE SYNTHASE 2, 2-AMINO-4-(2-AMINO-ETHOXY)-BUTYRIC ACID, PYRIDOXAL-5'-PHOSPHATE | 著者 | Huai, Q, Xia, Y, Chen, Y, Callahan, B, Li, N, Ke, H. | 登録日 | 2001-03-24 | 公開日 | 2001-04-04 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal structures of 1-aminocyclopropane-1-carboxylate (ACC) synthase in complex with aminoethoxyvinylglycine and pyridoxal-5'-phosphate provide new insight into catalytic mechanisms J.Biol.Chem., 276, 2001
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6CFE
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![BU of 6cfe by Molmil](/molmil-images/mine/6cfe) | |
6CBU
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![BU of 6cbu by Molmil](/molmil-images/mine/6cbu) | Crystal structure of C4S3: A computationally designed immunogen to target Carbohydrate-Occluded Epitopes on the HIV envelope | 分子名称: | Acylphosphatase-1, SULFATE ION | 著者 | Zhu, C, Ke, H.M, Swanstrom, R, Dokholyan, N.V. | 登録日 | 2018-02-05 | 公開日 | 2019-02-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Rationally designed carbohydrate-occluded epitopes elicit HIV-1 Env-specific antibodies. Nat Commun, 10, 2019
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4CYH
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5CYH
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![BU of 5cyh by Molmil](/molmil-images/mine/5cyh) | |
1FGL
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![BU of 1fgl by Molmil](/molmil-images/mine/1fgl) | Cyclophilin A complexed with a fragment of HIV-1 GAG protein | 分子名称: | CYCLOPHILIN A, HIV-1 GAG PROTEIN | 著者 | Zhao, Y, Chen, Y, Schutkowski, M, Fischer, G, Ke, H. | 登録日 | 1996-11-18 | 公開日 | 1997-04-01 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Cyclophilin A complexed with a fragment of HIV-1 gag protein: insights into HIV-1 infectious activity. Structure, 5, 1997
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4EL1
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![BU of 4el1 by Molmil](/molmil-images/mine/4el1) | Crystal structure of oxidized hPDI (abb'xa') | 分子名称: | Protein disulfide-isomerase | 著者 | Wang, C, Li, W, Ren, J, Ke, H, Gong, W, Feng, W, Wang, C.-C. | 登録日 | 2012-04-10 | 公開日 | 2013-04-10 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.883 Å) | 主引用文献 | Structural insights into the redox-regulated dynamic conformations of human protein disulfide isomerase Antioxid Redox Signal, 19, 2013
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4EKZ
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![BU of 4ekz by Molmil](/molmil-images/mine/4ekz) | Crystal structure of reduced hPDI (abb'xa') | 分子名称: | Protein disulfide-isomerase | 著者 | Wang, C, Li, W, Ren, J, Ke, H, Gong, W, Feng, W, Wang, C.-C. | 登録日 | 2012-04-10 | 公開日 | 2013-04-10 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Structural insights into the redox-regulated dynamic conformations of human protein disulfide isomerase Antioxid Redox Signal, 19, 2013
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1RMH
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![BU of 1rmh by Molmil](/molmil-images/mine/1rmh) | RECOMBINANT CYCLOPHILIN A FROM HUMAN T CELL | 分子名称: | AAPF PEPTIDE SUBSTRATE, CYCLOPHILIN A | 著者 | Zhao, Y, Ke, H. | 登録日 | 1995-07-31 | 公開日 | 1996-10-14 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structure implies that cyclophilin predominantly catalyzes the trans to cis isomerization. Biochemistry, 35, 1996
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1VBT
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![BU of 1vbt by Molmil](/molmil-images/mine/1vbt) | Structure of cyclophilin complexed with sulfur-substituted tetrapeptide AAPF | 分子名称: | CYCLOPHILIN A, SULFUR-SUBSTITUTED TETRAPEPTIDE | 著者 | Zhao, Y, Chen, Y, Schutkowski, M, Fischer, G, Ke, H. | 登録日 | 1998-06-16 | 公開日 | 1999-01-13 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Insight Into Conversion of Substrate to Inhibitor To be Published
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7ELE
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7ELD
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1VBS
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![BU of 1vbs by Molmil](/molmil-images/mine/1vbs) | STRUCTURE OF CYCLOPHILIN COMPLEXED WITH (D)ALA CONTAINING TETRAPEPTIDE | 分子名称: | CYCLOPHILIN A, TETRAPEPTIDE | 著者 | Zhao, Y, Chen, Y, Schutkowski, M, Fischer, G, Ke, H. | 登録日 | 1998-06-16 | 公開日 | 1999-01-13 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Mapping the stereospecificity of peptidyl prolyl cis/trans isomerases. FEBS Lett., 432, 1998
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