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PDB: 6 results

6GZY
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BU of 6gzy by Molmil
HOIP-fragment5 complex
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase RNF31, SODIUM ION, ...
Authors:Johansson, H, Tsai, Y.C.I, Fantom, K, Chung, C.W, Martino, L, House, D, Rittinger, K.
Deposit date:2018-07-05
Release date:2019-01-30
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Fragment-Based Covalent Ligand Screening Enables Rapid Discovery of Inhibitors for the RBR E3 Ubiquitin Ligase HOIP.
J. Am. Chem. Soc., 141, 2019
6SC9
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BU of 6sc9 by Molmil
dAb3/HOIP-RBR-HOIPIN-8
Descriptor: 2-[3-[2,6-bis(fluoranyl)-4-(1~{H}-pyrazol-4-yl)phenyl]-3-oxidanylidene-prop-1-enyl]-4-(1-methylpyrazol-4-yl)benzoic acid, CHLORIDE ION, E3 ubiquitin-protein ligase RNF31, ...
Authors:Tsai, Y.-C.I, Johansson, H, House, D, Rittinger, K.
Deposit date:2019-07-23
Release date:2019-11-27
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.47 Å)
Cite:Single-Domain Antibodies as Crystallization Chaperones to Enable Structure-Based Inhibitor Development for RBR E3 Ubiquitin Ligases.
Cell Chem Biol, 27, 2020
6SC8
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BU of 6sc8 by Molmil
dAb3/HOIP-RBR-Ligand4
Descriptor: CHLORIDE ION, E3 ubiquitin-protein ligase RNF31, SULFATE ION, ...
Authors:Tsai, Y.-C.I, Johansson, H, House, D, Rittinger, K.
Deposit date:2019-07-23
Release date:2019-11-27
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.106 Å)
Cite:Single-Domain Antibodies as Crystallization Chaperones to Enable Structure-Based Inhibitor Development for RBR E3 Ubiquitin Ligases.
Cell Chem Biol, 27, 2020
6SC7
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BU of 6sc7 by Molmil
dAb3/HOIP-RBR-Ligand3
Descriptor: CHLORIDE ION, E3 ubiquitin-protein ligase RNF31, SULFATE ION, ...
Authors:Tsai, Y.-C.I, Johansson, H, House, D, Rittinger, K.
Deposit date:2019-07-23
Release date:2019-11-27
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.56 Å)
Cite:Single-Domain Antibodies as Crystallization Chaperones to Enable Structure-Based Inhibitor Development for RBR E3 Ubiquitin Ligases.
Cell Chem Biol, 27, 2020
6SC5
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BU of 6sc5 by Molmil
dAb3/HOIP-RBR-Ligand2
Descriptor: CHLORIDE ION, E3 ubiquitin-protein ligase RNF31, SULFATE ION, ...
Authors:Tsai, Y.-C.I, Johansson, H, House, D, Rittinger, K.
Deposit date:2019-07-23
Release date:2019-11-27
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Single-Domain Antibodies as Crystallization Chaperones to Enable Structure-Based Inhibitor Development for RBR E3 Ubiquitin Ligases.
Cell Chem Biol, 27, 2020
2EW4
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BU of 2ew4 by Molmil
Solution structure of MrIA
Descriptor: MrIA
Authors:Nilsson, K.P, Lovelace, E.S, Caesar, C.E, Tynngard, N, Alewood, P.F, Johansson, H.M, Sharpe, I.A, Lewis, R.J, Daly, N.L, Craik, D.J.
Deposit date:2005-11-02
Release date:2005-11-15
Last modified:2020-06-24
Method:SOLUTION NMR
Cite:Solution structure of chi-conopeptide MrIA, a modulator of the human norepinephrine transporter
Biopolymers, 80, 2005

220113

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