6SC8
dAb3/HOIP-RBR-Ligand4
Summary for 6SC8
Entry DOI | 10.2210/pdb6sc8/pdb |
Descriptor | E3 ubiquitin-protein ligase RNF31, Single domain antibody, [2-(methylamino)-2-oxidanylidene-ethyl] (~{E})-4-[(2-oxidanylidene-5,6,7,8-tetrahydro-1~{H}-quinolin-3-yl)carbonylamino]but-2-enoate, ... (7 entities in total) |
Functional Keywords | human single domain antibody, hoip, rbr, inhibitor, ligase |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 3 |
Total formula weight | 70623.27 |
Authors | Tsai, Y.-C.I.,Johansson, H.,House, D.,Rittinger, K. (deposition date: 2019-07-23, release date: 2019-11-27, Last modification date: 2024-05-01) |
Primary citation | Tsai, Y.I.,Johansson, H.,Dixon, D.,Martin, S.,Chung, C.W.,Clarkson, J.,House, D.,Rittinger, K. Single-Domain Antibodies as Crystallization Chaperones to Enable Structure-Based Inhibitor Development for RBR E3 Ubiquitin Ligases. Cell Chem Biol, 27:83-, 2020 Cited by PubMed: 31813847DOI: 10.1016/j.chembiol.2019.11.007 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.106 Å) |
Structure validation
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