5J1I
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![BU of 5j1i by Molmil](/molmil-images/mine/5j1i) | |
5J1G
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![BU of 5j1g by Molmil](/molmil-images/mine/5j1g) | |
5J32
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![BU of 5j32 by Molmil](/molmil-images/mine/5j32) | Isopropylmalate dehydrogenase in complex with isopropylmalate | 分子名称: | 3-ISOPROPYLMALIC ACID, 3-isopropylmalate dehydrogenase 2, chloroplastic, ... | 著者 | Jez, J.M, Lee, S.G. | 登録日 | 2016-03-30 | 公開日 | 2016-05-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.933 Å) | 主引用文献 | Structure and Mechanism of Isopropylmalate Dehydrogenase from Arabidopsis thaliana: INSIGHTS ON LEUCINE AND ALIPHATIC GLUCOSINOLATE BIOSYNTHESIS. J.Biol.Chem., 291, 2016
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5JDV
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![BU of 5jdv by Molmil](/molmil-images/mine/5jdv) | Human carbonic anhydrase II (F131W) complexed with benzo[d]thiazole-2-sulfonamide | 分子名称: | 1,3-benzothiazole-2-sulfonamide, Carbonic anhydrase 2, ZINC ION | 著者 | Fox, J.M, Kang, K, Sastry, M, Sherman, W, Sankaran, B, Zwart, P.H, Whitesides, G.M. | 登録日 | 2016-04-17 | 公開日 | 2017-01-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Water-Restructuring Mutations Can Reverse the Thermodynamic Signature of Ligand Binding to Human Carbonic Anhydrase. Angew. Chem. Int. Ed. Engl., 56, 2017
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5J33
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![BU of 5j33 by Molmil](/molmil-images/mine/5j33) | Isopropylmalate dehydrogenase in complex with NAD+ | 分子名称: | 3-isopropylmalate dehydrogenase 2, chloroplastic, MAGNESIUM ION, ... | 著者 | Jez, J.M, Lee, S.G. | 登録日 | 2016-03-30 | 公開日 | 2016-05-18 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.492 Å) | 主引用文献 | Structure and Mechanism of Isopropylmalate Dehydrogenase from Arabidopsis thaliana: INSIGHTS ON LEUCINE AND ALIPHATIC GLUCOSINOLATE BIOSYNTHESIS. J.Biol.Chem., 291, 2016
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5J60
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![BU of 5j60 by Molmil](/molmil-images/mine/5j60) | Structure of a thioredoxin reductase from Gloeobacter violaceus | 分子名称: | CALCIUM ION, FLAVIN-ADENINE DINUCLEOTIDE, TETRAETHYLENE GLYCOL, ... | 著者 | Buey, R.M, de Pereda, J.M, Balsera, M. | 登録日 | 2016-04-04 | 公開日 | 2016-07-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A New Member of the Thioredoxin Reductase Family from Early Oxygenic Photosynthetic Organisms. Mol Plant, 10, 2017
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4N49
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![BU of 4n49 by Molmil](/molmil-images/mine/4n49) | Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1 Protein in complex with m7GpppG and SAM | 分子名称: | 7N-METHYL-8-HYDROGUANOSINE-5'-TRIPHOSPHATE, Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1, S-ADENOSYLMETHIONINE, ... | 著者 | Smietanski, M, Werener, M, Purta, E, Kaminska, K.H, Stepinski, J, Darzynkiewicz, E, Nowotny, M, Bujnicki, J.M. | 登録日 | 2013-10-08 | 公開日 | 2014-01-22 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural analysis of human 2'-O-ribose methyltransferases involved in mRNA cap structure formation. Nat Commun, 5, 2014
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4N5A
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![BU of 4n5a by Molmil](/molmil-images/mine/4n5a) | Crystal structure of Efr3 | 分子名称: | Protein EFR3 | 著者 | Wu, X, Chi, R.J, Baskin, J.M, Lucast, L, Burd, C.G, De Camilli, P, Reinisch, K.M. | 登録日 | 2013-10-09 | 公開日 | 2014-01-22 | 最終更新日 | 2014-03-19 | 実験手法 | X-RAY DIFFRACTION (3.204 Å) | 主引用文献 | Structural insights into assembly and regulation of the plasma membrane phosphatidylinositol 4-kinase complex. Dev.Cell, 28, 2014
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5XMH
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![BU of 5xmh by Molmil](/molmil-images/mine/5xmh) | Crystal structure of an IgM rheumatoid factor YES8c in complex with IgG1 Fc | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Immunoglobulin gamma-1 heavy chain, ... | 著者 | Shiroishi, M, Shimokawa, K, Lee, J.M, Kusakabe, M, Ueda, T. | 登録日 | 2017-05-15 | 公開日 | 2018-03-21 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure-function analyses of a stereotypic rheumatoid factor unravel the structural basis for germline-encoded antibody autoreactivity. J. Biol. Chem., 293, 2018
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4MX1
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![BU of 4mx1 by Molmil](/molmil-images/mine/4mx1) | Structure of ricin A chain bound with 2-amino-4-oxo-N-(2-(3-phenylureido)ethyl)-3,4-dihydropteridine-7-carboxamide | 分子名称: | 2-amino-4-oxo-N-{2-[(phenylcarbamoyl)amino]ethyl}-3,4-dihydropteridine-7-carboxamide, MALONIC ACID, Ricin A chain, ... | 著者 | Robertus, J.D, Wiget, P.A, Manzano, L.A, Pruet, J.M, Gao, G, Saito, R, Jasheway, K.R, Monzingo, A.F, Anslyn, E.V. | 登録日 | 2013-09-25 | 公開日 | 2014-01-15 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Sulfur incorporation generally improves Ricin inhibition in pterin-appended glycine-phenylalanine dipeptide mimics. Bioorg.Med.Chem.Lett., 23, 2013
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5JEH
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![BU of 5jeh by Molmil](/molmil-images/mine/5jeh) | Human carbonic anhydrase II (L198A) complexed with benzo[d]thiazole-2-sulfonamide | 分子名称: | 1,3-benzothiazole-2-sulfonamide, Carbonic anhydrase 2, ZINC ION | 著者 | Fox, J.M, Kang, K, Sastry, M, Sherman, W, Sankaran, B, Zwart, P.H, Whitesides, G.M. | 登録日 | 2016-04-18 | 公開日 | 2017-01-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | Water-Restructuring Mutations Can Reverse the Thermodynamic Signature of Ligand Binding to Human Carbonic Anhydrase. Angew. Chem. Int. Ed. Engl., 56, 2017
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4N4A
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![BU of 4n4a by Molmil](/molmil-images/mine/4n4a) | Cystal structure of Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1 | 分子名称: | Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1 | 著者 | Smietanski, M, Werener, M, Purta, E, Kaminska, K.H, Stepinski, J, Darzynkiewicz, E, Nowotny, M, Bujnicki, J.M. | 登録日 | 2013-10-08 | 公開日 | 2014-01-22 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structural analysis of human 2'-O-ribose methyltransferases involved in mRNA cap structure formation. Nat Commun, 5, 2014
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5JE7
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![BU of 5je7 by Molmil](/molmil-images/mine/5je7) | Human carbonic anhydrase II (F131Y) complexed with benzo[d]thiazole-2-sulfonamide | 分子名称: | 1,3-benzothiazole-2-sulfonamide, Carbonic anhydrase 2, ZINC ION | 著者 | Fox, J.M, Kang, K, Sastry, M, Sherman, W, Sankaran, B, Zwart, P.H, Whitesides, G.M. | 登録日 | 2016-04-17 | 公開日 | 2017-01-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Water-Restructuring Mutations Can Reverse the Thermodynamic Signature of Ligand Binding to Human Carbonic Anhydrase. Angew. Chem. Int. Ed. Engl., 56, 2017
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5XWB
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![BU of 5xwb by Molmil](/molmil-images/mine/5xwb) | Crystal Structure of 5-Enolpyruvulshikimate-3-phosphate Synthase from a Psychrophilic Bacterium, Colwellia psychrerythraea | 分子名称: | 3-phosphoshikimate 1-carboxyvinyltransferase | 著者 | Lee, J.H, Kim, H.J, Choi, J.M, Kim, D.-W, Seo, Y.-S. | 登録日 | 2017-06-29 | 公開日 | 2017-09-06 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structure of 5-enolpyruvylshikimate-3-phosphate synthase from a psychrophilic bacterium, Colwellia psychrerythraea 34H. Biochem. Biophys. Res. Commun., 492, 2017
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4N69
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![BU of 4n69 by Molmil](/molmil-images/mine/4n69) | Soybean Serine Acetyltransferase Complexed with Serine | 分子名称: | PHOSPHATE ION, SERINE, Serine Acetyltransferase Apoenzyme | 著者 | Yi, H, Dey, S, Kumaran, S, Krishnan, H.B, Jez, J.M. | 登録日 | 2013-10-11 | 公開日 | 2013-11-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure of soybean serine acetyltransferase and formation of the cysteine regulatory complex as a molecular chaperone. J.Biol.Chem., 288, 2013
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4NJ7
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![BU of 4nj7 by Molmil](/molmil-images/mine/4nj7) | PB1 Domain of AtARF7 - SeMet Derivative | 分子名称: | Auxin response factor 7 | 著者 | Korasick, D.A, Westfall, C.S, Lee, S.G, Nanao, M, Jez, J.M, Strader, L.C. | 登録日 | 2013-11-08 | 公開日 | 2014-03-26 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Molecular basis for AUXIN RESPONSE FACTOR protein interaction and the control of auxin response repression. Proc.Natl.Acad.Sci.USA, 111, 2014
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4NJ6
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![BU of 4nj6 by Molmil](/molmil-images/mine/4nj6) | PB1 Domain of AtARF7 | 分子名称: | Auxin response factor 7 | 著者 | Korasick, D.A, Westfall, C.S, Lee, S.G, Nanao, M, Jez, J.M, Strader, L.C. | 登録日 | 2013-11-08 | 公開日 | 2014-03-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Molecular basis for AUXIN RESPONSE FACTOR protein interaction and the control of auxin response repression. Proc.Natl.Acad.Sci.USA, 111, 2014
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4NMN
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![BU of 4nmn by Molmil](/molmil-images/mine/4nmn) | Aquifex aeolicus replicative helicase (DnaB) complexed with ADP, at 3.3 resolution | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Replicative DNA helicase, ... | 著者 | Lyubimov, A.Y, Strycharska, M.S, Erzberger, J.P, Berger, J.M. | 登録日 | 2013-11-15 | 公開日 | 2014-01-29 | 実験手法 | X-RAY DIFFRACTION (3.301 Å) | 主引用文献 | Nucleotide and partner-protein control of bacterial replicative helicase structure and function. Mol.Cell, 52, 2013
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4NQ5
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![BU of 4nq5 by Molmil](/molmil-images/mine/4nq5) | Bacillus cereus Zn-dependent metallo-beta-lactamase at pH 7 complexed with compound CS319 | 分子名称: | (3R,5R,7aS)-5-(sulfanylmethyl)tetrahydro[1,3]thiazolo[4,3-b][1,3]thiazole-3-carboxylic acid, Beta-lactamase 2, POTASSIUM ION, ... | 著者 | Gonzalez, J.M, Gonzalez, M.M, Vila, A.J. | 登録日 | 2013-11-23 | 公開日 | 2014-11-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Inhibition of metallo-lactamases with bicyclic compounds TO BE PUBLISHED
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4NDZ
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![BU of 4ndz by Molmil](/molmil-images/mine/4ndz) | Structure of Maltose Binding Protein fusion to 2-O-Sulfotransferase with bound heptasaccharide and PAP | 分子名称: | ADENOSINE-3'-5'-DIPHOSPHATE, Maltose-binding periplasmic protein, Heparan sulfate 2-O-sulfotransferase 1 fusion, ... | 著者 | Liu, C, Sheng, J, Krahn, J.M, Perera, L, Xu, Y, Hsieh, P, Liu, J, Pedersen, L.C. | 登録日 | 2013-10-28 | 公開日 | 2014-03-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.45 Å) | 主引用文献 | Deciphering the role of 2-O-sulfotransferase in regulating heparan sulfate biosynthesis To be Published
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5ZNI
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![BU of 5zni by Molmil](/molmil-images/mine/5zni) | |
6AFP
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![BU of 6afp by Molmil](/molmil-images/mine/6afp) | Crystal structure of class A b-lactamase, PenL, variant Asn136Asp, from Burkholderia thailandensis, in complex with ceftazidime-like boronic acid | 分子名称: | ACETATE ION, Beta-lactamase, PINACOL[[2-AMINO-ALPHA-(1-CARBOXY-1-METHYLETHOXYIMINO)-4-THIAZOLEACETYL]AMINO]METHANEBORONATE | 著者 | Cao, T.-P, Choi, J.M, Lee, S.H. | 登録日 | 2018-08-08 | 公開日 | 2020-01-15 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.398 Å) | 主引用文献 | Non-catalytic-Region Mutations Conferring Transition of Class A beta-Lactamases Into ESBLs. Front Mol Biosci, 2020
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6ALB
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![BU of 6alb by Molmil](/molmil-images/mine/6alb) | CREBBP bromodomain in complex with Cpd 30 (1-(3-(3-(1-methyl-1H-pyrazol-4-yl)isoquinolin-8-yl)-1-(tetrahydro-2H-pyran-4-yl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)ethan-1-one) | 分子名称: | 1-{3-[3-(1-methyl-1H-pyrazol-4-yl)isoquinolin-8-yl]-1-(oxan-4-yl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CREB-binding protein, ... | 著者 | Murray, J.M. | 登録日 | 2017-08-07 | 公開日 | 2018-10-17 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.053 Å) | 主引用文献 | Design and Synthesis of A Biaryl Series As Inhibitors for the Bromodomains of CBP/P300 To be published
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6AFO
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![BU of 6afo by Molmil](/molmil-images/mine/6afo) | |
1MM2
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![BU of 1mm2 by Molmil](/molmil-images/mine/1mm2) | Solution structure of the 2nd PHD domain from Mi2b | 分子名称: | Mi2-beta, ZINC ION | 著者 | Kwan, A.H.Y, Gell, D.A, Verger, A, Crossley, M, Matthews, J.M, Mackay, J.P. | 登録日 | 2002-09-02 | 公開日 | 2003-07-22 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Engineering a Protein Scaffold from a PHD Finger structure, 11, 2003
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