4USF
Human SLK with SB-440719
Summary for 4USF
Entry DOI | 10.2210/pdb4usf/pdb |
Related | 4USD 4USE |
Descriptor | STE20-LIKE SERINE/THREONINE-PROTEIN KINASE, 4-[4-(6-methoxynaphthalen-2-yl)-1H-imidazol-5-yl]pyridine (3 entities in total) |
Functional Keywords | transferase |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm : Q9H2G2 |
Total number of polymer chains | 2 |
Total formula weight | 69983.50 |
Authors | Elkins, J.M.,Salah, E.,Szklarz, M.,von Delft, F.,Bountra, C.,Edwards, A.M.,Knapp, S. (deposition date: 2014-07-07, release date: 2015-07-22, Last modification date: 2024-05-08) |
Primary citation | Elkins, J.M.,Fedele, V.,Szklarz, M.,Abdul Azeez, K.R.,Salah, E.,Mikolajczyk, J.,Romanov, S.,Sepetov, N.,Huang, X.P.,Roth, B.L.,Al Haj Zen, A.,Fourches, D.,Muratov, E.,Tropsha, A.,Morris, J.,Teicher, B.A.,Kunkel, M.,Polley, E.,Lackey, K.E.,Atkinson, F.L.,Overington, J.P.,Bamborough, P.,Moller, S.,Price, D.J.,Willson, T.M.,Drewry, D.H.,Knapp, S.,Zuercher, W.J. Comprehensive Characterization of the Published Kinase Inhibitor Set. Nat.Biotechnol., 34:95-, 2016 Cited by PubMed: 26501955DOI: 10.1038/NBT.3374 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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