3RO6
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![BU of 3ro6 by Molmil](/molmil-images/mine/3ro6) | Crystal structure of Dipeptide Epimerase from Methylococcus capsulatus complexed with Mg ion | 分子名称: | GLYCEROL, MAGNESIUM ION, Putative chloromuconate cycloisomerase, ... | 著者 | Lukk, T, Sakai, A, Song, L, Gerlt, J.A, Nair, S.K. | 登録日 | 2011-04-25 | 公開日 | 2011-05-11 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Homology models guide discovery of diverse enzyme specificities among dipeptide epimerases in the enolase superfamily. Proc.Natl.Acad.Sci.USA, 109, 2012
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3R10
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![BU of 3r10 by Molmil](/molmil-images/mine/3r10) | Crystal structure of NYSGRC enolase target 200555, a putative dipeptide epimerase from Francisella philomiragia : Mg complex | 分子名称: | Enzyme of enolase superfamily, GLYCEROL, MAGNESIUM ION, ... | 著者 | Vetting, M.W, Hillerich, B, Seidel, R.D, Zencheck, W.D, Toro, R, Imker, H.J, Gerlt, J.A, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC) | 登録日 | 2011-03-09 | 公開日 | 2011-04-20 | 最終更新日 | 2012-03-28 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Homology models guide discovery of diverse enzyme specificities among dipeptide epimerases in the enolase superfamily. Proc.Natl.Acad.Sci.USA, 109, 2012
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3OTU
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![BU of 3otu by Molmil](/molmil-images/mine/3otu) | PDK1 mutant bound to allosteric disulfide fragment activator JS30 | 分子名称: | 3-(1H-INDOL-3-YL)-4-{1-[2-(1-METHYLPYRROLIDIN-2-YL)ETHYL]-1H-INDOL-3-YL}-1H-PYRROLE-2,5-DIONE, 3-phosphoinositide-dependent protein kinase 1, 4-[4-(naphthalen-1-ylmethyl)piperazin-1-yl]-4-oxobutane-1-thiol, ... | 著者 | Sadowsky, J.D, Wells, J.A. | 登録日 | 2010-09-13 | 公開日 | 2011-03-23 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.1013 Å) | 主引用文献 | Turning a protein kinase on or off from a single allosteric site via disulfide trapping. Proc.Natl.Acad.Sci.USA, 108, 2011
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3OW1
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![BU of 3ow1 by Molmil](/molmil-images/mine/3ow1) | Crystal structure of D-mannonate dehydratase from Chromohalobacter salexigens complexed with MG | 分子名称: | GLYCEROL, MAGNESIUM ION, Mandelate racemase/muconate lactonizing enzyme, ... | 著者 | Fedorov, A.A, Fedorov, E.V, Wichelecki, D, Gerlt, J.A, Almo, S.C. | 登録日 | 2010-09-17 | 公開日 | 2011-09-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.798 Å) | 主引用文献 | CRYSTAL STRUCTURE OF D-MANNONATE DEHYDRATASE FROM CHROMOHALOBACTER SALEXIGENS complexed with MG To be Published
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1Q41
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![BU of 1q41 by Molmil](/molmil-images/mine/1q41) | GSK-3 Beta complexed with Indirubin-3'-monoxime | 分子名称: | (Z)-1H,1'H-[2,3']BIINDOLYLIDENE-3,2'-DIONE-3-OXIME, GLYCOGEN SYNTHASE KINASE-3 BETA | 著者 | Bertrand, J.A, Thieffine, S, Vulpetti, A, Cristiani, C, Valsasina, B, Knapp, S, Kalisz, H.M, Flocco, M. | 登録日 | 2003-08-01 | 公開日 | 2003-10-21 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural Characterization of the Gsk-3Beta Active Site Using Selective and Non-selective ATP-Mimetic Inhibitors J.Mol.Biol., 333, 2003
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3P0W
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![BU of 3p0w by Molmil](/molmil-images/mine/3p0w) | Crystal structure of D-Glucarate dehydratase from Ralstonia solanacearum complexed with Mg and D-glucarate | 分子名称: | D-GLUCARATE, MAGNESIUM ION, Mandelate racemase/muconate lactonizing protein | 著者 | Fedorov, A.A, Fedorov, E.V, Gerlt, J.A, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC) | 登録日 | 2010-09-29 | 公開日 | 2010-10-13 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.71 Å) | 主引用文献 | Crystal structure of D-Glucarate dehydratase from Ralstonia solanacearum complexed with Mg and D-glucarate To be Published
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1PRM
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![BU of 1prm by Molmil](/molmil-images/mine/1prm) | TWO BINDING ORIENTATIONS FOR PEPTIDES TO SRC SH3 DOMAIN: DEVELOPMENT OF A GENERAL MODEL FOR SH3-LIGAND INTERACTIONS | 分子名称: | C-SRC TYROSINE KINASE SH3 DOMAIN, PROLINE-RICH LIGAND PLR1 (AFAPPLPRR) | 著者 | Feng, S, Chen, J.K, Yu, H, Simon, J.A, Schreiber, S.L. | 登録日 | 1994-10-10 | 公開日 | 1995-02-07 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Two binding orientations for peptides to the Src SH3 domain: development of a general model for SH3-ligand interactions. Science, 266, 1994
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1PRL
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![BU of 1prl by Molmil](/molmil-images/mine/1prl) | TWO BINDING ORIENTATIONS FOR PEPTIDES TO SRC SH3 DOMAIN: DEVELOPMENT OF A GENERAL MODEL FOR SH3-LIGAND INTERACTIONS | 分子名称: | C-SRC TYROSINE KINASE SH3 DOMAIN, PROLINE-RICH LIGAND PLR1 (AFAPPLPRR) | 著者 | Feng, S, Chen, J.K, Yu, H, Simon, J.A, Schreiber, S.L. | 登録日 | 1994-10-10 | 公開日 | 1995-02-07 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Two binding orientations for peptides to the Src SH3 domain: development of a general model for SH3-ligand interactions. Science, 266, 1994
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3P60
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![BU of 3p60 by Molmil](/molmil-images/mine/3p60) | Crystal structure of the mutant T159V of orotidine 5'-monophosphate decarboxylase from Methanobacterium thermoautotrophicum complexed with inhibitor BMP | 分子名称: | 6-HYDROXYURIDINE-5'-PHOSPHATE, Orotidine 5'-monophosphate decarboxylase | 著者 | Fedorov, A.A, Fedorov, E.V, Wood, B.M, Gerlt, J.A, Almo, S.C. | 登録日 | 2010-10-11 | 公開日 | 2011-09-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Conformational changes in orotidine 5'-monophosphate decarboxylase: a structure-based explanation for how the 5'-phosphate group activates the enzyme. Biochemistry, 51, 2012
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1PJR
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3P3I
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![BU of 3p3i by Molmil](/molmil-images/mine/3p3i) | Crystal structure of the F36A mutant of the fluoroacetyl-CoA-specific thioesterase FlK in complex with fluoroacetate and CoA | 分子名称: | COENZYME A, Fluoroacetyl coenzyme A thioesterase, fluoroacetic acid | 著者 | Weeks, A.M, Coyle, S.M, Jinek, M, Doudna, J.A, Chang, M.C.Y. | 登録日 | 2010-10-04 | 公開日 | 2010-10-20 | 最終更新日 | 2011-11-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural and biochemical studies of a fluoroacetyl-CoA-specific thioesterase reveal a molecular basis for fluorine selectivity. Biochemistry, 49, 2010
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3P5Y
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![BU of 3p5y by Molmil](/molmil-images/mine/3p5y) | Crystal structure of the mutant T159A of orotidine 5'-monophosphate decarboxylase from Methanobacterium thermoautotrophicum complexed with inhibitor BMP | 分子名称: | 6-HYDROXYURIDINE-5'-PHOSPHATE, GLYCEROL, Orotidine 5'-phosphate decarboxylase | 著者 | Fedorov, A.A, Fedorov, E.V, Wood, B.M, Gerlt, J.A, Almo, S.C. | 登録日 | 2010-10-11 | 公開日 | 2011-09-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Conformational changes in orotidine 5'-monophosphate decarboxylase: a structure-based explanation for how the 5'-phosphate group activates the enzyme. Biochemistry, 51, 2012
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1QMP
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![BU of 1qmp by Molmil](/molmil-images/mine/1qmp) | Phosphorylated aspartate in the crystal structure of the sporulation response regulator, Spo0A | 分子名称: | CALCIUM ION, Stage 0 sporulation protein A | 著者 | Lewis, R.J, Brannigan, J.A, Muchova, K, Barak, I, Wilkinson, A.J. | 登録日 | 1999-10-04 | 公開日 | 1999-11-14 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Phosphorylated aspartate in the structure of a response regulator protein. J. Mol. Biol., 294, 1999
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1QDD
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![BU of 1qdd by Molmil](/molmil-images/mine/1qdd) | CRYSTAL STRUCTURE OF HUMAN LITHOSTATHINE TO 1.3 A RESOLUTION | 分子名称: | LITHOSTATHINE, beta-D-galactopyranose-(1-3)-[N-acetyl-alpha-neuraminic acid-(2-6)]2-acetamido-2-deoxy-alpha-D-glucopyranose | 著者 | Gerbaud, V, Pignol, D, Loret, E, Bertrand, J.A, Berland, Y, Fontecilla-Camps, J.C, Canselier, J.P, Gabas, N, Verdier, J.M. | 登録日 | 1999-05-20 | 公開日 | 1999-05-28 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Mechanism of calcite crystal growth inhibition by the N-terminal undecapeptide of lithostathine. J.Biol.Chem., 275, 2000
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1QGY
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![BU of 1qgy by Molmil](/molmil-images/mine/1qgy) | Ferredoxin:NADP+ reductase mutant with Lys 75 replaced by Glu (K75E) | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, Ferredoxin--NADP+ reductase, SULFATE ION | 著者 | Hermoso, J.A, Mayoral, T, Medina, M, Martinez-Ripoll, M, Martinez-Julvez, M, Sanz-Aparicio, J, Gomez-Moreno, C. | 登録日 | 1999-05-10 | 公開日 | 2004-03-09 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural analysis of interactions for complex formation between Ferredoxin-NADP+ reductase and its protein partners Proteins, 59, 2005
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3RR1
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![BU of 3rr1 by Molmil](/molmil-images/mine/3rr1) | Crystal structure of enolase PRK14017 (target EFI-500653) from Ralstonia pickettii 12J | 分子名称: | CHLORIDE ION, D-MALATE, Putative D-galactonate dehydratase | 著者 | Patskovsky, Y, Hillerich, B, Seidel, R.D, Zencheck, W.D, Toro, R, Imker, H.J, Gerlt, J.A, Almo, S.C, Enzyme Function Initiative (EFI) | 登録日 | 2011-04-28 | 公開日 | 2011-05-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Crystal structure of enolase PRK14017 from Ralstonia pickettii To be Published
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1QO5
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1QVL
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![BU of 1qvl by Molmil](/molmil-images/mine/1qvl) | Structure of the antimicrobial hexapeptide cyc-(RRWWRF) bound to SDS micelles | 分子名称: | c-RW | 著者 | Appelt, C, Soderhall, J.A, Bienert, M, Dathe, M, Schmieder, P. | 登録日 | 2003-08-28 | 公開日 | 2004-09-28 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of the Antimicrobial, Cationic Hexapeptide Cyclo(RRWWRF) and Its Analogues in Solution and Bound to Detergent Micelles Chembiochem, 6, 2005
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1SO4
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![BU of 1so4 by Molmil](/molmil-images/mine/1so4) | Crystal structure of K64A mutant of 3-keto-L-gulonate 6-phosphate decarboxylase with bound L-threonohydroxamate 4-phosphate | 分子名称: | 3-keto-L-gulonate 6-phosphate decarboxylase, L-THREONOHYDROXAMATE 4-PHOSPHATE, MAGNESIUM ION | 著者 | Wise, E.L, Yew, W.S, Gerlt, J.A, Rayment, I. | 登録日 | 2004-03-12 | 公開日 | 2004-06-08 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Evolution of Enzymatic Activities in the Orotidine 5'-Monophosphate Decarboxylase Suprafamily: Crystallographic Evidence for a Proton Relay System in the Active Site of 3-Keto-l-gulonate 6-Phosphate Decarboxylase(,) Biochemistry, 43, 2004
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1SJ4
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![BU of 1sj4 by Molmil](/molmil-images/mine/1sj4) | Crystal structure of a C75U mutant Hepatitis Delta Virus ribozyme precursor, in Cu2+ solution | 分子名称: | precursor form of the Hepatitis Delta virus ribozyme, small nuclear ribonucleoprotein A | 著者 | Ke, A, Zhou, K, Ding, F, Cate, J.H, Doudna, J.A. | 登録日 | 2004-03-02 | 公開日 | 2004-05-18 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | A Conformational Switch controls hepatitis delta virus ribozyme
catalysis Nature, 429, 2004
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1SJB
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![BU of 1sjb by Molmil](/molmil-images/mine/1sjb) | X-ray structure of o-succinylbenzoate synthase complexed with o-succinylbenzoic acid | 分子名称: | 2-SUCCINYLBENZOATE, MAGNESIUM ION, N-acylamino acid racemase | 著者 | Thoden, J.B, Taylor-Ringia, E.A, Garrett, J.B, Gerlt, J.A, Holden, H.M, Rayment, I. | 登録日 | 2004-03-03 | 公開日 | 2004-06-01 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Evolution of Enzymatic Activity in the Enolase Superfamily: Structural Studies of the Promiscuous o-Succinylbenzoate Synthase from Amycolatopsis Biochemistry, 43, 2004
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1SKL
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![BU of 1skl by Molmil](/molmil-images/mine/1skl) | Structure of the antimicrobial hexapeptide cyc-(RRNalNalRF) bound to DPC micelles | 分子名称: | cyclic hexapeptide RR(NAL)(NAL)RF | 著者 | Appelt, C, Soderhall, J.A, Bienert, M, Dathe, M, Schmieder, P. | 登録日 | 2004-03-05 | 公開日 | 2005-03-15 | 最終更新日 | 2012-12-12 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of the antimicrobial, cationic hexapeptide cyclo(RRWWRF) and its analogues in solution and bound to detergent micelles. Chembiochem, 6, 2005
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3RR3
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![BU of 3rr3 by Molmil](/molmil-images/mine/3rr3) | Structure of (R)-flurbiprofen bound to mCOX-2 | 分子名称: | (2R)-2-(3-fluoro-4-phenyl-phenyl)propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Duggan, K.C, Hermanson, D.J, Musee, J, Prusakiewicz, J.J, Scheib, J, Carter, B.D, Banerjee, S, Oates, J.A, Marnett, L.J. | 登録日 | 2011-04-28 | 公開日 | 2011-11-09 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.842 Å) | 主引用文献 | (R)-Profens are substrate-selective inhibitors of endocannabinoid oxygenation by COX-2. Nat.Chem.Biol., 7, 2011
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3RUV
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![BU of 3ruv by Molmil](/molmil-images/mine/3ruv) | Crystal structure of Cpn-rls in complex with ATP analogue from Methanococcus maripaludis | 分子名称: | Chaperonin, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Pereira, J.H, Ralston, C.Y, Douglas, N.R, Kumar, R, McAndrew, R.P, Knee, K.M, King, J.A, Frydman, J, Adams, P.D. | 登録日 | 2011-05-05 | 公開日 | 2012-01-04 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.242 Å) | 主引用文献 | Mechanism of nucleotide sensing in group II chaperonins. Embo J., 31, 2012
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1SPD
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![BU of 1spd by Molmil](/molmil-images/mine/1spd) | |