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PDB: 42550 件

2XI5
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N-terminal endonuclease domain of La Crosse virus L-protein
分子名称: MANGANESE (II) ION, RNA POLYMERASE L
著者Reguera, J, Weber, F, Cusack, S.
登録日2010-06-28
公開日2010-10-06
最終更新日2012-07-18
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Bunyaviridae RNA Polymerases (L-Protein) Have an N-Terminal, Influenza-Like Endonuclease Domain, Essential for Viral CAP-Dependent Transcription.
Plos Pathog., 6, 2010
2XJH
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Structure and Copper-binding Properties of Methanobactins from Methylosinus trichosporium OB3b
分子名称: COPPER (II) ION, METHANOBACTIN MB-OB3B, SODIUM ION
著者El-Ghazouani, A, Basle, A, Firbank, S.J, Knapp, C.W, Gray, J, Graham, D.W, Dennison, C.
登録日2010-07-06
公開日2011-02-02
最終更新日2019-05-22
実験手法X-RAY DIFFRACTION (0.92 Å)
主引用文献Copper-Binding Properties and Structures of Methanobactins from Methylosinus Trichosporium Ob3B.
Inorg.Chem., 50, 2011
2XF6
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Crystal structure of Bacillus subtilis SPP1 phage gp23.1, a putative chaperone.
分子名称: GP23.1
著者Veesler, D, Blangy, S, Lichiere, J, Ortiz-Lombardia, M, Tavares, P, Campanacci, V, Cambillau, C.
登録日2010-05-20
公開日2010-08-11
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Crystal Structure of Bacillus Subtilis Spp1 Phage Gp23.1, A Putative Chaperone.
Protein Sci., 19, 2010
2XJ0
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Protein kinase Pim-1 in complex with fragment-4 from crystallographic fragment screen
分子名称: (E)-3-(2-AMINO-PYRIDINE-5YL)-ACRYLIC ACID, PROTO-ONCOGENE SERINE/THREONINE PROTEIN KINASE PIM-1
著者Schulz, M.N, Fanghanel, J, Schafer, M, Badock, V, Briem, H, Boemer, U, Nguyen, D, Husemann, M, Hillig, R.C.
登録日2010-07-01
公開日2011-02-23
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystallographic Fragment Screen Identifies Cinnamic Acid Derivatives as Starting Points for Potent Pim-1 Inhibitors
Acta Crystallogr.,Sect.D, 67, 2011
2XF7
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Crystal structure of Bacillus subtilis SPP1 phage gp23.1, a putative chaperone. High-resolution structure.
分子名称: GP23.1
著者Veesler, D, Blangy, S, Lichiere, J, Ortiz-Lombardia, M, Tavares, P, Campanacci, V, Cambillau, C.
登録日2010-05-20
公開日2010-08-11
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Crystal Structure of Bacillus Subtilis Spp1 Phage Gp23.1, A Putative Chaperone.
Protein Sci., 19, 2010
4CT8
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Competence or damage-inducible protein CinA from Thermus thermophilus
分子名称: CINA-LIKE PROTEIN, GLYCEROL, SODIUM ION, ...
著者Derrick, J, Karuppiah, V.
登録日2014-03-12
公開日2014-10-15
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.16 Å)
主引用文献Structure and Mechanism of the Bifunctional Cina Enzyme from Thermus Thermophilus
J.Biol.Chem., 289, 2014
2XBM
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Crystal structure of the dengue virus methyltransferase bound to a 5'- capped octameric RNA
分子名称: 5'-(*G3AP*GP*AP*AP*CP*CP*UP*GP*A)-3', GLYCEROL, NONSTRUCTURAL PROTEIN NS5, ...
著者Yap, L.J, Luo, D.H, Chung, K.Y, Lim, S.P, Bodenreider, C, Noble, C, Shi, P.Y, Lescar, J.
登録日2010-04-13
公開日2010-09-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal Structure of the Dengue Virus Methyltransferase Bound to a 5'-Capped Octameric RNA
Plos One, 5, 2010
2PQZ
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HIV-1 Protease in complex with a pyrrolidine-based inhibitor
分子名称: CHLORIDE ION, N,N'-(3S,4S)-PYRROLIDINE-3,4-DIYLBIS(N-BENZYLBENZENESULFONAMIDE), Protease
著者Boettcher, J, Blum, A, Heine, A, Diederich, W.E, Klebe, G.
登録日2007-05-03
公開日2008-04-15
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structure-Guided Design of C2-Symmetric HIV-1 Protease Inhibitors Based on a Pyrrolidine Scaffold.
J.Med.Chem., 51, 2008
2XF5
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Crystal structure of Bacillus subtilis SPP1 phage gp23.1, a putative chaperone.
分子名称: GP23.1
著者Veesler, D, Blangy, S, Lichiere, J, Ortiz-Lombardia, M, Tavares, P, Campanacci, V, Cambillau, C.
登録日2010-05-20
公開日2010-08-11
最終更新日2017-07-12
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure of Bacillus Subtilis Spp1 Phage Gp23.1, A Putative Chaperone.
Protein Sci., 19, 2010
1IFY
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Solution Structure of the Internal UBA Domain of HHR23A
分子名称: UV EXCISION REPAIR PROTEIN RAD23 HOMOLOG A
著者Mueller, T.D, Feigon, J.
登録日2001-04-13
公開日2002-07-03
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structures of UBA domains reveal a conserved hydrophobic surface for protein-protein interactions.
J.Mol.Biol., 319, 2002
2XRF
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Crystal structure of human uridine phosphorylase 2
分子名称: GLYCEROL, MAGNESIUM ION, URACIL, ...
著者Welin, M, Moche, M, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Karlberg, T, Kol, S, Kotenyova, T, Kouznetsova, E, Nyman, T, Persson, C, Schuler, H, Schutz, P, Siponen, M.I, Thorsell, A.G, Tresaugues, L, Van Der Berg, S, Wahlberg, E, Weigelt, J, Nordlund, P.
登録日2010-09-14
公開日2010-09-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of Human Uridine Phosphorylase 2
To be Published
1CQ7
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ASPARTATE AMINOTRANSFERASE (E.C. 2.6.1.1) COMPLEXED WITH C5-PYRIDOXAL-5P-PHOSPHATE
分子名称: 2-[O-PHOSPHONOPYRIDOXYL]-AMINO-PENTANOIC ACID, ASPARTATE AMINOTRANSFERASE
著者Ishijima, J, Nakai, T, Kawaguchi, S, Hirotsu, K, Kuramitsu, S.
登録日1999-08-06
公開日2000-12-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Free energy requirement for domain movement of an enzyme
J.Biol.Chem., 275, 2000
2XMQ
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Crystal structure of human NDRG2 protein provides insight into its role as a tumor suppressor
分子名称: ACETATE ION, PROTEIN NDRG2
著者Hwang, J, Kim, Y, Lee, H, Kim, M.H.
登録日2010-07-29
公開日2011-01-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.81 Å)
主引用文献Crystal Structure of Human Ndrg2 Protein Provides Insight Into its Role as a Tumor Suppressor.
J.Biol.Chem., 286, 2011
2XP1
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Structure of the tandem SH2 domains from Antonospora locustae transcription elongation factor Spt6
分子名称: CHLORIDE ION, SPT6, SULFATE ION
著者Diebold, M.-L, Koch, M, Cavarelli, J, Romier, C.
登録日2010-08-24
公開日2010-09-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Noncanonical Tandem Sh2 Enables Interaction of Elongation Factor Spt6 with RNA Polymerase II.
J.Biol.Chem., 285, 2010
2XRI
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Crystal structure of human ERI1 exoribonuclease 3
分子名称: ERI1 EXORIBONUCLEASE 3, GLYCEROL, MAGNESIUM ION
著者Welin, M, Siponen, M.I, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Karlberg, T, Kol, S, Kotenyova, T, Kouznetsova, E, Moche, M, Nyman, T, Persson, C, Schuler, H, Schutz, P, Thorsell, A.G, Tresaugues, L, Van Der Berg, S, Wahlberg, E, Weigelt, J, Nordlund, P.
登録日2010-09-15
公開日2010-09-29
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal Structure of Human Eri1 Exoribonuclease 3
To be Published
2XKJ
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CRYSTAL STRUCTURE OF CATALYTIC CORE OF A. BAUMANNII TOPO IV (PARE- PARC FUSION TRUNCATE)
分子名称: GLYCEROL, SULFATE ION, TOPOISOMERASE IV
著者Wohlkonig, A, Chan, P.F, Fosberry, A.P, Homes, P, Huang, J, Kranz, M, Leydon, V.R, Miles, T.J, Pearson, N.D, Perera, R.L, Shillings, A.J, Gwynn, M.N, Bax, B.D.
登録日2010-07-08
公開日2010-09-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Basis of Quinolone Inhibition of Type Iia Topoisomerases and Target-Mediated Resistance
Nat.Struct.Mol.Biol., 17, 2010
1GZM
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Structure of Bovine Rhodopsin in a Trigonal Crystal Form
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, DI-PALMITOYL-3-SN-PHOSPHATIDYLETHANOLAMINE, LAURYL DIMETHYLAMINE-N-OXIDE, ...
著者Li, J.
登録日2002-05-24
公開日2003-11-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Structure of Bovine Rhodopsin in a Trigonal Crystal Form
J.Mol.Biol., 343, 2004
2XGJ
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Structure of Mtr4, a DExH helicase involved in nuclear RNA processing and surveillance
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATP-DEPENDENT RNA HELICASE DOB1, RNA (5'-(*AP*AP*AP*AP*A)-3')
著者Weir, J.R, Bonneau, F, Hentschel, J, Conti, E.
登録日2010-06-04
公開日2010-06-23
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural Analysis Reveals the Characteristic Features of Mtr4, a Dexh Helicase Involved in Nuclear RNA Processing and Surveillance.
Proc.Natl.Acad.Sci.USA, 107, 2010
2XIZ
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Protein kinase Pim-1 in complex with fragment-3 from crystallographic fragment screen
分子名称: (E)-PYRIDIN-4-YL-ACRYLIC ACID, PROTO-ONCOGENE SERINE/THREONINE PROTEIN KINASE PIM-1
著者Schulz, M.N, Fanghanel, J, Schafer, M, Badock, V, Briem, H, Boemer, U, Nguyen, D, Husemann, M, Hillig, R.C.
登録日2010-07-01
公開日2011-02-23
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献Crystallographic Fragment Screen Identifies Cinnamic Acid Derivatives as Starting Points for Potent Pim-1 Inhibitors
Acta Crystallogr.,Sect.D, 67, 2011
2XTD
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Structure of the TBL1 tetramerisation domain
分子名称: TBL1 F-BOX-LIKE/WD REPEAT-CONTAINING PROTEIN TBL1X
著者Oberoi, J, Fairall, L, Watson, P.J, Greenwood, J.A, Schwabe, J.W.R.
登録日2010-10-06
公開日2011-01-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural Basis for the Assembly of the Smrt/Ncor Core Transcriptional Repression Machinery.
Nat.Struct.Mol.Biol., 18, 2011
2XJI
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Structure and Copper-binding Properties of Methanobactins from Methylosinus trichosporium OB3b
分子名称: COPPER (II) ION, METHANOBACTIN MB-OB3B
著者El-Ghazouani, A, Basle, A, Firbank, S.J, Knapp, C.W, Gray, J, Graham, D.W, Dennison, C.
登録日2010-07-06
公開日2011-02-02
最終更新日2019-07-10
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献Copper-Binding Properties and Structures of Methanobactins from Methylosinus Trichosporium Ob3B.
Inorg.Chem., 50, 2011
2XRG
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Crystal structure of Autotaxin (ENPP2) in complex with the HA155 boronic acid inhibitor
分子名称: CALCIUM ION, ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE FAMILY MEMBER 2, IODIDE ION, ...
著者Hausmann, J, Albers, H.M.H.G, Perrakis, A.
登録日2010-09-14
公開日2011-01-19
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural Basis of Substrate Discrimination and Integrin Binding by Autotaxin.
Nat.Struct.Mol.Biol., 18, 2011
2XBK
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X-ray structure of the substrate-bound cytochrome P450 PimD - a polyene macrolide antibiotic pimaricin epoxidase
分子名称: 4,5-DE-EPOXYPIMARICIN, PIMD PROTEIN, PROTOPORPHYRIN IX CONTAINING FE
著者Kells, P.M, Ouellet, H, Santos-Aberturas, J, Aparicio, J.F, Podust, L.M.
登録日2010-04-12
公開日2010-08-04
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of Cytochrome P450 Pimd Suggests Epoxidation of the Polyene Macrolide Pimaricin Occurs Via a Hydroperoxoferric Intermediate.
Chem.Biol., 17, 2010
2XI7
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N-terminal endonuclease domain of La Crosse virus L-protein
分子名称: 2-4-DIOXO-4-PHENYLBUTANOIC ACID, MANGANESE (II) ION, RNA POLYMERASE L
著者Reguera, J, Weber, F, Cusack, S.
登録日2010-06-28
公開日2010-10-06
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Bunyaviridae RNA Polymerases (L-Protein) Have an N-Terminal, Influenza-Like Endonuclease Domain, Essential for Viral CAP-Dependent Transcription.
Plos Pathog., 6, 2010
2XKK
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CRYSTAL STRUCTURE OF MOXIFLOXACIN, DNA, and A. BAUMANNII TOPO IV (PARE-PARC FUSION TRUNCATE)
分子名称: 1-cyclopropyl-6-fluoro-8-methoxy-7-[(4aS,7aS)-octahydro-6H-pyrrolo[3,4-b]pyridin-6-yl]-4-oxo-1,4-dihydroquinoline-3-carboxylic acid, DNA, MAGNESIUM ION, ...
著者Wohlkonig, A, Chan, P.F, Fosberry, A.P, Homes, P, Huang, J, Kranz, M, Leydon, V.R, Miles, T.J, Pearson, N.D, Perera, R.L, Shillings, A.J, Gwynn, M.N, Bax, B.D.
登録日2010-07-08
公開日2010-09-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Structural Basis of Quinolone Inhibition of Type Iia Topoisomerases and Target-Mediated Resistance
Nat.Struct.Mol.Biol., 17, 2010

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