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PDB: 2 results

7U4C
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BU of 7u4c by Molmil
Borrelia burgdorferi HtpG N-terminal domain (1-228) in complex with BX-2819
Descriptor: Chaperone protein HtpG, ethyl (4-{3-[2,4-dihydroxy-5-(1-methylethyl)phenyl]-5-sulfanyl-4H-1,2,4-triazol-4-yl}benzyl)carbamate
Authors:Kowalewski, M.E, Lietzan, A, Haystead, T, Redinbo, M.R.
Deposit date:2022-02-28
Release date:2023-03-08
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.28 Å)
Cite:Targeting Borrelia burgdorferi HtpG with a berserker molecule, a strategy for anti-microbial development.
Cell Chem Biol, 2023
5VJA
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BU of 5vja by Molmil
Crystal Structure of human zipper-interacting protein kinase (ZIPK, alias DAPK3) in complex with a pyrazolo[3,4-d]pyrimidinone ligand (HS38)
Descriptor: (2R)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide, DIMETHYL SULFOXIDE, Death-associated protein kinase 3, ...
Authors:Carlson, D.A, Singer, M.R, Sutherland, C, Redondo, C, Alexander, L, Hughes, P.F, Knapp, S, MacDonald, J.A, Haystead, T.A.J.
Deposit date:2017-04-19
Release date:2018-08-08
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.46 Å)
Cite:Targeting Pim Kinases and DAPK3 to Control Hypertension.
Cell Chem Biol, 25, 2018

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