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PDB: 4 results

6OPJ
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BU of 6opj by Molmil
Menin in complex with peptide inhibitor 25
Descriptor: DIMETHYL SULFOXIDE, Menin, Peptide inhibitor 25, ...
Authors:Linhares, B.M, Fortuna, P, Cierpicki, T, Grembecka, J, Berlicki, L.
Deposit date:2019-04-25
Release date:2020-09-02
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.5006572 Å)
Cite:Covalent and noncovalent constraints yield a figure eight-like conformation of a peptide inhibiting the menin-MLL interaction.
Eur.J.Med.Chem., 207, 2020
7AD0
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BU of 7ad0 by Molmil
X-ray structure of Mdm2 with modified p53 peptide
Descriptor: E3 ubiquitin-protein ligase Mdm2, Modified p53 peptide
Authors:Twarda-Clapa, A, Fortuna, P, Grudnik, P, Dubin, G, Berlicki, L, Holak, T.A.
Deposit date:2020-09-13
Release date:2020-10-28
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.07 Å)
Cite:Systematic ""foldamerization"" of peptide inhibiting p53-MDM2/X interactions by the incorporation of trans- or cis-2-aminocyclopentanecarboxylic acid residues
Eur.J.Med.Chem., 208, 2020
7ARR
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BU of 7arr by Molmil
The de novo designed hybrid alpha/beta-miniprotein
Descriptor: CHLORIDE ION, MAGNESIUM ION, alpha/beta-peptide, ...
Authors:Bejger, M, Fortuna, P, Drewniak-Switalska, M, Rypniewski, W, Berlicki, L.
Deposit date:2020-10-26
Release date:2021-07-14
Method:X-RAY DIFFRACTION (1.1 Å)
Cite:A computationally designed beta-amino acid-containing miniprotein.
Chem.Commun.(Camb.), 57, 2021
7ARS
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BU of 7ars by Molmil
The de novo designed hybrid alpha/beta-miniprotein (with Se-Methionine)
Descriptor: MAGNESIUM ION, alpha/beta-peptide, trifluoroacetic acid
Authors:Bejger, M, Fortuna, P, Drewniak-Switalska, M, Rypniewski, W, Berlicki, L.
Deposit date:2020-10-26
Release date:2021-07-14
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:A computationally designed beta-amino acid-containing miniprotein.
Chem.Commun.(Camb.), 57, 2021

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