6OPJ
Menin in complex with peptide inhibitor 25
Summary for 6OPJ
Entry DOI | 10.2210/pdb6opj/pdb |
Descriptor | Menin, Peptide inhibitor 25, DIMETHYL SULFOXIDE, ... (6 entities in total) |
Functional Keywords | protein-protein interaction inhibitor, protein binding-inhibitor complex, protein binding/inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 56878.96 |
Authors | Linhares, B.M.,Fortuna, P.,Cierpicki, T.,Grembecka, J.,Berlicki, L. (deposition date: 2019-04-25, release date: 2020-09-02, Last modification date: 2023-11-15) |
Primary citation | Fortuna, P.,Linhares, B.M.,Purohit, T.,Pollock, J.,Cierpicki, T.,Grembecka, J.,Berlicki, L. Covalent and noncovalent constraints yield a figure eight-like conformation of a peptide inhibiting the menin-MLL interaction. Eur.J.Med.Chem., 207:112748-112748, 2020 Cited by PubMed: 32882610DOI: 10.1016/j.ejmech.2020.112748 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.50065718427 Å) |
Structure validation
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