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6OPJ

Menin in complex with peptide inhibitor 25

Summary for 6OPJ
Entry DOI10.2210/pdb6opj/pdb
DescriptorMenin, Peptide inhibitor 25, DIMETHYL SULFOXIDE, ... (6 entities in total)
Functional Keywordsprotein-protein interaction inhibitor, protein binding-inhibitor complex, protein binding/inhibitor
Biological sourceHomo sapiens (Human)
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Total number of polymer chains2
Total formula weight56878.96
Authors
Linhares, B.M.,Fortuna, P.,Cierpicki, T.,Grembecka, J.,Berlicki, L. (deposition date: 2019-04-25, release date: 2020-09-02, Last modification date: 2023-11-15)
Primary citationFortuna, P.,Linhares, B.M.,Purohit, T.,Pollock, J.,Cierpicki, T.,Grembecka, J.,Berlicki, L.
Covalent and noncovalent constraints yield a figure eight-like conformation of a peptide inhibiting the menin-MLL interaction.
Eur.J.Med.Chem., 207:112748-112748, 2020
Cited by
PubMed: 32882610
DOI: 10.1016/j.ejmech.2020.112748
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.50065718427 Å)
Structure validation

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