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PDB: 94 件

3F5C
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Structure of Dax-1:LRH-1 complex
分子名称: Nuclear receptor subfamily 0 group B member 1, Nuclear receptor subfamily 5 group A member 2
著者Fletterick, R.J, Sablin, E.P.
登録日2008-11-03
公開日2008-12-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The structure of corepressor Dax-1 bound to its target nuclear receptor LRH-1.
Proc.Natl.Acad.Sci.USA, 105, 2008
1AIM
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CRUZAIN INHIBITED BY BENZOYL-TYROSINE-ALANINE-FLUOROMETHYLKETONE
分子名称: BENZOYL-TYROSINE-ALANINE-FLUORO-METHYL KETONE, CRUZAIN
著者Fletterick, R, Gillmor, S.
登録日1997-04-21
公開日1997-10-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural determinants of specificity in the cysteine protease cruzain.
Protein Sci., 6, 1997
1ANC
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BU of 1anc by Molmil
ANIONIC TRYPSIN MUTANT WITH SER 214 REPLACED BY LYS
分子名称: ANIONIC TRYPSIN, BENZAMIDINE, CALCIUM ION
著者Fletterick, R.J, Mcgrath, M.E.
登録日1994-12-21
公開日1997-04-01
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Perturbing the polar environment of Asp102 in trypsin: consequences of replacing conserved Ser214.
Biochemistry, 31, 1992
1ANB
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ANIONIC TRYPSIN MUTANT WITH SER 214 REPLACED BY GLU
分子名称: ANIONIC TRYPSIN, BENZAMIDINE, CALCIUM ION
著者Fletterick, R.J, Mcgrath, M.E.
登録日1994-12-21
公開日1997-04-01
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Perturbing the polar environment of Asp102 in trypsin: consequences of replacing conserved Ser214.
Biochemistry, 31, 1992
1AND
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ANIONIC TRYPSIN MUTANT WITH ARG 96 REPLACED BY HIS
分子名称: ANIONIC TRYPSIN, BENZAMIDINE, COPPER (II) ION
著者Fletterick, R.J, Mcgrath, M.E.
登録日1994-12-21
公開日1997-04-01
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure of an engineered, metal-actuated switch in trypsin.
Biochemistry, 32, 1993
1ANE
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ANIONIC TRYPSIN WILD TYPE
分子名称: ANIONIC TRYPSIN, BENZAMIDINE
著者Fletterick, R.J, Mcgrath, M.E.
登録日1994-12-21
公開日1997-04-01
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of an engineered, metal-actuated switch in trypsin.
Biochemistry, 32, 1993
2NCD
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NCD (NON-CLARET DISJUNCTIONAL) DIMER FROM D. MELANOGASTER
分子名称: ADENOSINE-5'-DIPHOSPHATE, PROTEIN (Kinesin motor NCD), SULFATE ION
著者Sablin, E.P, Case, R.B, Dai, S.C, Hart, C.L, Ruby, A, Vale, R.D, Fletterick, R.J.
登録日1999-06-04
公開日1999-06-09
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Direction determination in the minus-end-directed kinesin motor ncd.
Nature, 395, 1998
6DDA
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Nurr1 Covalently Modified by a Dopamine Metabolite
分子名称: 5-hydroxy-1,2-dihydro-6H-indol-6-one, BROMIDE ION, Nuclear receptor subfamily 4 group A member 2, ...
著者Bruning, J.M, Wang, Y, Otrabella, F, Boxue, T, Liu, H, Bhattacharya, P, Guo, S, Holton, J.M, Fletterick, R.J, Jacobson, M.P, England, P.M.
登録日2018-05-09
公開日2019-03-20
最終更新日2019-11-06
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Covalent Modification and Regulation of the Nuclear Receptor Nurr1 by a Dopamine Metabolite.
Cell Chem Biol, 26, 2019
1T79
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Crystal structure of the androgen receptor ligand binding domain in complex with a FxxLW motif
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, FxxLW motif peptide
著者Hur, E, Pfaff, S.J, Payne, E.S, Gron, H, Buehrer, B.M, Fletterick, R.J.
登録日2004-05-08
公開日2004-08-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
1T7F
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Crystal structure of the androgen receptor ligand binding domain in complex with a LxxLL motif
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, LxxLL motif peptide
著者Hur, E, Pfaff, S.J, Payne, E.S, Gron, H, Buehrer, B.M, Fletterick, R.J.
登録日2004-05-10
公開日2004-08-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
1T7M
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Crystal structure of the androgen receptor ligand binding domain in complex with a FxxYF motif
分子名称: 1,2-ETHANEDIOL, 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, ...
著者Hur, E, Pfaff, S.J, Payne, E.S, Gron, H, Buehrer, B.M, Fletterick, R.J.
登録日2004-05-10
公開日2004-08-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
1T74
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Crystal structure of the androgen receptor ligand binding domain in complex with a WxxLF motif
分子名称: 1,2-ETHANEDIOL, 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, ...
著者Hur, E, Pfaff, S.J, Payne, E.S, Gron, H, Buehrer, B.M, Fletterick, R.J.
登録日2004-05-07
公開日2004-08-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
1T7T
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Crystal structure of the androgen receptor ligand binding domain in complex with 5-alpha dihydrotestosterone
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor
著者Hur, E, Pfaff, S.J, Payne, E.S, Gron, H, Buehrer, B.M, Fletterick, R.J.
登録日2004-05-10
公開日2004-08-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Recognition and accommodation at the androgen receptor coactivator binding interface.
Plos Biol., 2, 2004
2Z4J
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Crystal structure of AR LBD with SHP peptide NR Box 2
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, Nuclear receptor 0B2
著者Jouravel, N, Fletterick, R.J.
登録日2007-06-19
公開日2007-12-04
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Interaction between the androgen receptor and a segment of its corepressor SHP
Acta Crystallogr.,Sect.D, 63, 2007
3LVG
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Crystal structure of a clathrin heavy chain and clathrin light chain complex
分子名称: Clathrin heavy chain 1, Clathrin light chain B
著者Wilbur, J.D, Hwang, P.K, Ybe, J.A, Lane, M, Sellers, B.D, Jacobson, M.P, Fletterick, R.J, Brodsky, F.M.
登録日2010-02-20
公開日2010-06-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (7.94 Å)
主引用文献Conformation switching of clathrin light chain regulates clathrin lattice assembly.
Dev.Cell, 18, 2010
3LVH
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Crystal structure of a clathrin heavy chain and clathrin light chain complex
分子名称: Clathrin heavy chain 1, Clathrin light chain B
著者Wilbur, J.D, Hwang, P.K, Ybe, J.A, Lane, M, Sellers, B.D, Jacobson, M.P, Fletterick, R.J, Brodsky, F.M.
登録日2010-02-20
公開日2010-06-09
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (9 Å)
主引用文献Conformation switching of clathrin light chain regulates clathrin lattice assembly.
Dev.Cell, 18, 2010
3TX7
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Crystal structure of LRH-1/beta-catenin complex
分子名称: (2S)-3-{[{[(2S)-2,3-DIHYDROXYPROPYL]OXY}(HYDROXY)PHOSPHORYL]OXY}-2-[(6E)-HEXADEC-6-ENOYLOXY]PROPYL (8E)-OCTADEC-8-ENOATE, Catenin beta-1, Nuclear receptor subfamily 5 group A member 2
著者Yumoto, F, Fletterick, R.
登録日2011-09-22
公開日2011-12-14
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.76 Å)
主引用文献Structural basis of coactivation of liver receptor homolog-1 by beta-catenin.
Proc.Natl.Acad.Sci.USA, 109, 2012
3I00
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Crystal Structure of the huntingtin interacting protein 1 coiled coil domain
分子名称: Huntingtin-interacting protein 1
著者Wilbur, J.D, Hwang, P.K, Brodsky, F.M, Fletterick, R.J.
登録日2009-06-24
公開日2010-02-23
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Accommodation of structural rearrangements in the huntingtin-interacting protein 1 coiled-coil domain.
Acta Crystallogr.,Sect.D, 66, 2010
3BKI
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Crystal Structure of the GluR2 ligand binding core (S1S2J) in complex with FQX at 1.87 Angstroms
分子名称: Glutamate receptor 2, [1,2,5]oxadiazolo[3,4-g]quinoxaline-6,7(5H,8H)-dione 1-oxide
著者Cruz, L, Estebanez-Perpina, E, Pfaff, S, Borngraeber, S, Bao, N, Fletterick, R, England, P.
登録日2007-12-06
公開日2008-09-16
最終更新日2019-09-04
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione (ANQX) forms an irreversible bond to the active site of the GluR2 AMPA receptor.
J.Med.Chem., 51, 2008
1YGP
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PHOSPHORYLATED FORM OF YEAST GLYCOGEN PHOSPHORYLASE WITH PHOSPHATE BOUND IN THE ACTIVE SITE.
分子名称: PHOSPHATE ION, PYRIDOXAL-5'-PHOSPHATE, YEAST GLYCOGEN PHOSPHORYLASE
著者Lin, K, Rath, V.L, Dai, S.C, Fletterick, R.J, Hwang, P.K.
登録日1996-05-30
公開日1996-12-23
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A protein phosphorylation switch at the conserved allosteric site in GP.
Science, 273, 1996
1XZX
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Thyroxine-Thyroid Hormone Receptor Interactions
分子名称: 3,5,3'TRIIODOTHYRONINE, CACODYLATE ION, Thyroid hormone receptor beta-1
著者Sandler, B, Webb, P, Apriletti, J.W, Huber, B.R, Togashi, M, Cunha Lima, S.T, Juric, S, Nilsson, S, Wagner, R, Fletterick, R.J, Baxter, J.D.
登録日2004-11-12
公開日2004-12-07
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Thyroxine-thyroid hormone receptor interactions.
J.Biol.Chem., 279, 2004
3F7D
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SF-1 LBD bound by phosphatidylcholine
分子名称: (2S)-2-{[(1R)-1-hydroxyhexadecyl]oxy}-3-{[(1R)-1-hydroxyoctadecyl]oxy}propyl 2-(trimethylammonio)ethyl phosphate, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha, nuclear receptor SF-1
著者Sablin, E.P, Fletterick, R.J.
登録日2008-11-07
公開日2008-12-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of SF-1 bound by different phospholipids: evidence for regulatory ligands.
Mol.Endocrinol., 23, 2009
2AIM
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CRUZAIN INHIBITED WITH BENZOYL-ARGININE-ALANINE-FLUOROMETHYLKETONE
分子名称: BENZOYL-ARGININE-ALANINE-FLUORO-METHYL KETONE, CRUZAIN
著者Gillmor, S.A, Fletterick, R.J.
登録日1997-04-21
公開日1997-10-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural determinants of specificity in the cysteine protease cruzain.
Protein Sci., 6, 1997
1T5Z
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Crystal Structure of the Androgen Receptor Ligand Binding Domain (LBD) with DHT and a peptide derived from its physiological coactivator ARA70
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, Nuclear receptor coactivator 4
著者Estebanez-Perpina, E, Moore, J.M.R, Mar, E, Nguyen, P, Delgado-Rodrigues, E, Baxter, J.D, Webb, P, Fletterick, R.J, Guy, R.K.
登録日2004-05-05
公開日2005-01-25
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor.
J.Biol.Chem., 280, 2005
1T63
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Crystal Structure of the Androgen Receptor Ligand Binding Domain with DHT and a peptide derived from its physiological coactivator GRIP1 NR box3
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, Nuclear receptor coactivator 2
著者Estebanez-Perpina, E, Moore, J.M.R, Mar, E, Nguyen, P, Delgado-Rodrigues, E, Baxter, J.D, Webb, P, Fletterick, R.J, Guy, R.K.
登録日2004-05-05
公開日2005-01-25
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor.
J.Biol.Chem., 280, 2005

 

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