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1T5Z

Crystal Structure of the Androgen Receptor Ligand Binding Domain (LBD) with DHT and a peptide derived from its physiological coactivator ARA70

Summary for 1T5Z
Entry DOI10.2210/pdb1t5z/pdb
Related1T63 1T65
DescriptorAndrogen receptor, Nuclear receptor coactivator 4, 5-ALPHA-DIHYDROTESTOSTERONE, ... (4 entities in total)
Functional Keywordsandrogen receptor ligand binding domain ara70 crystal structure coactivators, hormone-growth factor complex, hormone/growth factor
Biological sourceHomo sapiens (human)
More
Cellular locationNucleus: P10275
Total number of polymer chains2
Total formula weight31460.90
Authors
Estebanez-Perpina, E.,Moore, J.M.R.,Mar, E.,Nguyen, P.,Delgado-Rodrigues, E.,Baxter, J.D.,Webb, P.,Fletterick, R.J.,Guy, R.K. (deposition date: 2004-05-05, release date: 2005-01-25, Last modification date: 2024-02-14)
Primary citationEstebanez-Perpina, E.,Moore, J.M.R.,Mar, E.,Delgado-Rodrigues, E.,Nguyen, P.,Baxter, J.D.,Buehrer, B.M.,Webb, P.,Fletterick, R.J.,Guy, R.K.
The Molecular Mechanisms of Coactivator Utilization in Ligand-dependent Transactivation by the Androgen Receptor.
J.Biol.Chem., 280:8060-8068, 2005
Cited by
PubMed: 15563469
DOI: 10.1074/jbc.M407046200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

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