7X4D
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![BU of 7x4d by Molmil](/molmil-images/mine/7x4d) | |
7X41
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![BU of 7x41 by Molmil](/molmil-images/mine/7x41) | |
7X43
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![BU of 7x43 by Molmil](/molmil-images/mine/7x43) | |
4R3K
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![BU of 4r3k by Molmil](/molmil-images/mine/4r3k) | |
4R3L
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![BU of 4r3l by Molmil](/molmil-images/mine/4r3l) | |
2CWB
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![BU of 2cwb by Molmil](/molmil-images/mine/2cwb) | Solution Structure of the Ubiquitin-Associated Domain of Human BMSC-UbP and its Complex with Ubiquitin | 分子名称: | Immunoglobulin G-binding protein G,Ubiquitin-like protein 7 | 著者 | Chang, Y.G, Song, A.X, Gao, Y.G, Shi, Y.H, Lin, X.J, Cao, X.T, Lin, D.H, Hu, H.Y. | 登録日 | 2005-06-17 | 公開日 | 2006-06-06 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the ubiquitin-associated domain of human BMSC-UbP and its complex with ubiquitin. Protein Sci., 15, 2006
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3MO0
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![BU of 3mo0 by Molmil](/molmil-images/mine/3mo0) | Human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E11 | 分子名称: | 1,2-ETHANEDIOL, Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, ... | 著者 | Chang, Y, Horton, J.R, Cheng, X. | 登録日 | 2010-04-22 | 公開日 | 2010-06-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Adding a lysine mimic in the design of potent inhibitors of histone lysine methyltransferases. J.Mol.Biol., 400, 2010
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4EM0
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![BU of 4em0 by Molmil](/molmil-images/mine/4em0) | |
4EM1
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3SVM
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![BU of 3svm by Molmil](/molmil-images/mine/3svm) | Human MPP8 - human DNMT3AK47me2 peptide | 分子名称: | DNA (cytosine-5)-methyltransferase 3A, M-phase phosphoprotein 8 | 著者 | Chang, Y, Horton, J.R, Zhang, X, Cheng, X. | 登録日 | 2011-07-12 | 公開日 | 2011-11-30 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a. Nat Commun, 2, 2011
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4EM2
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![BU of 4em2 by Molmil](/molmil-images/mine/4em2) | |
3SW9
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![BU of 3sw9 by Molmil](/molmil-images/mine/3sw9) | GLP (G9a-like protein) SET domain in complex with Dnmt3aK44me0 peptide | 分子名称: | DNA (cytosine-5)-methyltransferase 3A, Histone-lysine N-methyltransferase EHMT1, SINEFUNGIN, ... | 著者 | Chang, Y, Horton, J.R, Zhang, X, Cheng, X. | 登録日 | 2011-07-13 | 公開日 | 2011-12-07 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a. Nat Commun, 2, 2011
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3SWC
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![BU of 3swc by Molmil](/molmil-images/mine/3swc) | GLP (G9a-like protein) SET domain in complex with Dnmt3aK44me2 peptide | 分子名称: | DNA (cytosine-5)-methyltransferase 3A, Histone-lysine N-methyltransferase EHMT1, S-ADENOSYL-L-HOMOCYSTEINE, ... | 著者 | Chang, Y, Horton, J.R, Zhang, X, Cheng, X. | 登録日 | 2011-07-13 | 公開日 | 2011-11-30 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.332 Å) | 主引用文献 | MPP8 mediates the interactions between DNA methyltransferase Dnmt3a and H3K9 methyltransferase GLP/G9a. Nat Commun, 2, 2011
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3QXY
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![BU of 3qxy by Molmil](/molmil-images/mine/3qxy) | Human SETD6 in complex with RelA Lys310 | 分子名称: | 1,2-ETHANEDIOL, N-lysine methyltransferase SETD6, S-ADENOSYLMETHIONINE, ... | 著者 | Chang, Y, Levy, D, Horton, J.R, Peng, J, Zhang, X, Gozani, O, Cheng, X. | 登録日 | 2011-03-02 | 公開日 | 2011-05-25 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structural basis of SETD6-mediated regulation of the NF-kB network via methyl-lysine signaling. Nucleic Acids Res., 39, 2011
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3RC0
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![BU of 3rc0 by Molmil](/molmil-images/mine/3rc0) | Human SETD6 in complex with RelA Lys310 peptide | 分子名称: | 1,2-ETHANEDIOL, N-lysine methyltransferase SETD6, S-ADENOSYLMETHIONINE, ... | 著者 | Chang, Y, Levy, D, Horton, J.R, Peng, J, Zhang, X, Gozani, O, Cheng, X. | 登録日 | 2011-03-30 | 公開日 | 2011-05-25 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Structural basis of SETD6-mediated regulation of the NF-kB network via methyl-lysine signaling. Nucleic Acids Res., 39, 2011
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4LXO
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![BU of 4lxo by Molmil](/molmil-images/mine/4lxo) | |
3FPD
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![BU of 3fpd by Molmil](/molmil-images/mine/3fpd) | G9a-like protein lysine methyltransferase inhibition by BIX-01294 | 分子名称: | Histone-lysine N-methyltransferase, H3 lysine-9 specific 5, N-(1-benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amine, ... | 著者 | Chang, Y, Zhang, X, Horton, J.R, Cheng, X. | 登録日 | 2009-01-05 | 公開日 | 2009-02-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis for G9a-like protein lysine methyltransferase inhibition by BIX-01294. Nat.Struct.Mol.Biol., 16, 2009
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3OPT
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![BU of 3opt by Molmil](/molmil-images/mine/3opt) | Crystal structure of the Rph1 catalytic core with a-ketoglutarate | 分子名称: | 2-OXOGLUTARIC ACID, DNA damage-responsive transcriptional repressor RPH1, NICKEL (II) ION | 著者 | Chang, Y, Wu, J, Tong, X, Zhou, J, Ding, J. | 登録日 | 2010-09-02 | 公開日 | 2010-12-22 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal structure of the catalytic core of Saccharomyces cerevesiae histone demethylase Rph1: insights into the substrate specificity and catalytic mechanism Biochem.J., 433, 2011
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3OPW
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![BU of 3opw by Molmil](/molmil-images/mine/3opw) | Crystal Structure of the Rph1 catalytic core | 分子名称: | DNA damage-responsive transcriptional repressor RPH1 | 著者 | Chang, Y, Wu, J, Tong, X, Zhou, J, Ding, J. | 登録日 | 2010-09-02 | 公開日 | 2010-12-22 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of the catalytic core of Saccharomyces cerevesiae histone demethylase Rph1: insights into the substrate specificity and catalytic mechanism Biochem.J., 433, 2011
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3QO2
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![BU of 3qo2 by Molmil](/molmil-images/mine/3qo2) | Structural insights for MPP8 chromodomain interaction with histone H3 lysine 9 | 分子名称: | 1,2-ETHANEDIOL, Histone H3 peptide, M-phase phosphoprotein 8 | 著者 | Chang, Y, Horton, J.R, Bedford, M.T, Zhang, X, Cheng, X. | 登録日 | 2011-02-09 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Structural insights for MPP8 chromodomain interaction with histone H3 lysine 9: potential effect of phosphorylation on methyl-lysine binding. J.Mol.Biol., 408, 2011
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2Q9Q
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![BU of 2q9q by Molmil](/molmil-images/mine/2q9q) | The crystal structure of full length human GINS complex | 分子名称: | DNA replication complex GINS protein PSF1, DNA replication complex GINS protein PSF2, GINS complex subunit 3, ... | 著者 | Chang, Y.P, Wang, G, Chen, X.S. | 登録日 | 2007-06-13 | 公開日 | 2007-08-07 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.36 Å) | 主引用文献 | Crystal structure of the GINS complex and functional insights into its role in DNA replication. Proc.Natl.Acad.Sci.Usa, 104, 2007
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3UCI
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![BU of 3uci by Molmil](/molmil-images/mine/3uci) | Crystal structure of Rhodostomin ARLDDL mutant | 分子名称: | disintegrin | 著者 | Shiu, J.H, Chen, C.Y, Chen, Y.C, Chang, Y.T, Chang, Y.S, Huang, C.H, Chuang, W.J. | 登録日 | 2011-10-27 | 公開日 | 2012-11-21 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Design of Integrin AlphaVbeta3-Specific Disintegrin for Cancer Therapy To be Published
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1WKQ
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![BU of 1wkq by Molmil](/molmil-images/mine/1wkq) | |
6KPH
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![BU of 6kph by Molmil](/molmil-images/mine/6kph) | 343 K cryoEM structure of Sso-KARI in complex with Mg2+, NADH and CPD | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Ketol-acid reductoisomerase, MAGNESIUM ION, ... | 著者 | Chen, C.Y, Chang, Y.C, Lin, B.L, Huang, C.H, Tsai, M.D. | 登録日 | 2019-08-15 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (2.41 Å) | 主引用文献 | Temperature-Resolved Cryo-EM Uncovers Structural Bases of Temperature-Dependent Enzyme Functions. J.Am.Chem.Soc., 141, 2019
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6KQO
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![BU of 6kqo by Molmil](/molmil-images/mine/6kqo) | 328 K cryoEM structure of Sso-KARI in complex with Mg2+, NADH and CPD | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Ketol-acid reductoisomerase, MAGNESIUM ION, ... | 著者 | Chen, C.Y, Chang, Y.C, Lin, B.L, Huang, C.H, Tsai, M.D. | 登録日 | 2019-08-18 | 公開日 | 2020-03-25 | 最終更新日 | 2024-03-27 | 実験手法 | ELECTRON MICROSCOPY (2.52 Å) | 主引用文献 | Temperature-Resolved Cryo-EM Uncovers Structural Bases of Temperature-Dependent Enzyme Functions. J.Am.Chem.Soc., 141, 2019
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