6MBI
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7MZV
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![BU of 7mzv by Molmil](/molmil-images/mine/7mzv) | Structure of yeast pseudouridine synthase 7 (PUS7) | 分子名称: | Multisubstrate pseudouridine synthase 7, SULFATE ION | 著者 | Purchal, M, Koutmos, M. | 登録日 | 2021-05-24 | 公開日 | 2022-02-09 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Pseudouridine synthase 7 is an opportunistic enzyme that binds and modifies substrates with diverse sequences and structures. Proc.Natl.Acad.Sci.USA, 119, 2022
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5DJW
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5F7C
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5OVY
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![BU of 5ovy by Molmil](/molmil-images/mine/5ovy) | Crystal structure of MAB_4384 tetR | 分子名称: | Putative transcriptional regulator, TetR family | 著者 | Richard, M, Gutierrez, A.V, Viljoen, A, Ghigo, E, Blaise, M, Kremer, L. | 登録日 | 2017-08-30 | 公開日 | 2018-03-28 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Mechanistic and Structural Insights Into the Unique TetR-Dependent Regulation of a Drug Efflux Pump inMycobacterium abscessus. Front Microbiol, 9, 2018
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4Z66
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![BU of 4z66 by Molmil](/molmil-images/mine/4z66) | Nucleosome disassembly by RSC and SWI/SNF is enhanced by H3 acetylation near the nucleosome dyad axis | 分子名称: | DNA (147-MER), Histone H2A, Histone H2B 1.1, ... | 著者 | Dechassa, M.L, Luger, K, Chatterjee, N, North, J.A, Manohar, M, Prasad, R, Ottessen, J.J, Poirier, M.G, Bartholomew, B. | 登録日 | 2015-04-03 | 公開日 | 2015-10-14 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Histone Acetylation near the Nucleosome Dyad Axis Enhances Nucleosome Disassembly by RSC and SWI/SNF. Mol.Cell.Biol., 35, 2015
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6HHC
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![BU of 6hhc by Molmil](/molmil-images/mine/6hhc) | Allosteric Inhibition as a new mode of Action for BAY 1213790, a Neutralizing Antibody Targeting the Activated form of Coagulation Factor XI | 分子名称: | Coagulation factor XI, DIMETHYL SULFOXIDE, FXIA ANTIBODY FAB HEAVY CHAIN, ... | 著者 | Schaefer, M, Buchmueller, A, Dittmer, F, Strassburger, J, Wilmen, A. | 登録日 | 2018-08-27 | 公開日 | 2019-09-11 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Allosteric Inhibition as a New Mode of Action for BAY 1213790, a Neutralizing Antibody Targeting the Activated Form of Coagulation Factor XI. J.Mol.Biol., 431, 2019
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5G5R
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5ELX
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5G5X
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7FBY
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![BU of 7fby by Molmil](/molmil-images/mine/7fby) | Crystal Structure of PH0140 from Pyrococcus horikosii OT3 | 分子名称: | 1,2-ETHANEDIOL, ISOLEUCINE, Transcriptional regulatory protein | 著者 | Richard, M, Ahmad, M, Pal, R.K, Biswal, B.K, Jeyakanthan, J. | 登録日 | 2021-07-13 | 公開日 | 2022-07-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.001 Å) | 主引用文献 | Crystal Structure of PH0140 from Pyrococcus horikosii OT3 To Be Published
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5IG5
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5IG4
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![BU of 5ig4 by Molmil](/molmil-images/mine/5ig4) | Crystal structure of N. vectensis CaMKII-A hub | 分子名称: | GLYCEROL, Predicted protein | 著者 | Bhattacharyya, M, Pappireddi, N, Gee, C.L, Barros, T, Kuriyan, J. | 登録日 | 2016-02-26 | 公開日 | 2016-03-23 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Molecular mechanism of activation-triggered subunit exchange in Ca(2+)/calmodulin-dependent protein kinase II. Elife, 5, 2016
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5IG1
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![BU of 5ig1 by Molmil](/molmil-images/mine/5ig1) | Crystal structure of S. rosetta CaMKII kinase domain | 分子名称: | CAMK/CAMK2 protein kinase, PHOSPHATE ION | 著者 | Bhattacharyya, M, Gee, C.L, Barros, T, Kuriyan, J. | 登録日 | 2016-02-26 | 公開日 | 2016-03-23 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Molecular mechanism of activation-triggered subunit exchange in Ca(2+)/calmodulin-dependent protein kinase II. Elife, 5, 2016
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7Z90
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5IG0
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![BU of 5ig0 by Molmil](/molmil-images/mine/5ig0) | Crystal structure of S. rosetta CaMKII hub | 分子名称: | CAMK/CAMK2 protein kinase, GLYCEROL, SULFATE ION | 著者 | Bhattacharyya, M, Gee, C.L, Barros, T, Kuriyan, J. | 登録日 | 2016-02-26 | 公開日 | 2016-03-23 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Molecular mechanism of activation-triggered subunit exchange in Ca(2+)/calmodulin-dependent protein kinase II. Elife, 5, 2016
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5G2N
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![BU of 5g2n by Molmil](/molmil-images/mine/5g2n) | X-ray structure of PI3Kinase Gamma in complex with Copanlisib | 分子名称: | 2-azanyl-~{N}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamide, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM, SULFATE ION | 著者 | Schaefer, M, Scott, W.J, Hentemann, M.F, Rowley, R.B, Bull, C.O, Jenkins, S, Bullion, A.M, Johnson, J, Redman, A, Robbins, A.H, Esler, W, Fracasso, R.P, Garrison, T, Hamilton, M, Michels, M, Wood, J.E, Wilkie, D.P, Xiao, H, Levy, J, Liu, N, Stasik, E, Brands, M, Lefranc, J. | 登録日 | 2016-04-11 | 公開日 | 2016-04-20 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.68 Å) | 主引用文献 | Discovery and Sar of Novel 2,3-Dihydroimidazo(1,2-C)Quinazoline Pi3K Inhibitors: Identification of Copanlisib (Bay 80-6946) Chemmedchem, 11, 2016
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5G1X
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![BU of 5g1x by Molmil](/molmil-images/mine/5g1x) | Crystal structure of Aurora-A kinase in complex with N-Myc | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, AURORA KINASE A, MAGNESIUM ION, ... | 著者 | Richards, M.W, Burgess, S.G, Bayliss, R. | 登録日 | 2016-03-31 | 公開日 | 2016-11-16 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Structural Basis of N-Myc Binding by Aurora-A and its Destabilization by Kinase Inhibitors Proc.Natl.Acad.Sci.USA, 113, 2016
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5ID5
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5A0R
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![BU of 5a0r by Molmil](/molmil-images/mine/5a0r) | Product peptide-bound structure of metalloprotease Zmp1 variant E143A from Clostridium difficile | 分子名称: | GLYCEROL, PRODUCT PEPTIDE, ZINC ION, ... | 著者 | Schacherl, M, Pichlo, C, Neundorf, I, Baumann, U. | 登録日 | 2015-04-22 | 公開日 | 2015-08-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.251 Å) | 主引用文献 | Structural Basis of Proline-Proline Peptide Bond Specificity of the Metalloprotease Zmp1 Implicated in Motility of Clostridium Difficile. Structure, 23, 2015
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1M1L
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![BU of 1m1l by Molmil](/molmil-images/mine/1m1l) | Human Suppressor of Fused (N-terminal domain) | 分子名称: | Suppressor of Fused | 著者 | Merchant, M, Vajdos, F.F, Ultsch, M, Maun, H.R, Wendt, U, Cannon, J, Lazarus, R.A, de Vos, A.M, de Sauvage, F.J. | 登録日 | 2002-06-19 | 公開日 | 2004-02-03 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Suppressor of fused regulates Gli activity through a dual binding mechanism Mol.Cell.Biol., 24, 2004
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5A0P
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![BU of 5a0p by Molmil](/molmil-images/mine/5a0p) | Apo-structure of metalloprotease Zmp1 from Clostridium difficile | 分子名称: | ZINC ION, ZINC METALLOPROTEASE ZMP1 | 著者 | Schacherl, M, Pichlo, C, Neundorf, I, Baumann, U. | 登録日 | 2015-04-22 | 公開日 | 2015-08-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.398 Å) | 主引用文献 | Structural Basis of Proline-Proline Peptide Bond Specificity of the Metalloprotease Zmp1 Implicated in Motility of Clostridium Difficile. Structure, 23, 2015
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5A0X
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![BU of 5a0x by Molmil](/molmil-images/mine/5a0x) | Substrate peptide-bound structure of metalloprotease Zmp1 variant E143AY178F from Clostridium difficile | 分子名称: | SUBSTRATE PEPTIDE, ZINC ION, ZINC METALLOPROTEASE ZMP1 | 著者 | Schacherl, M, Pichlo, C, Neundorf, I, Baumann, U. | 登録日 | 2015-04-23 | 公開日 | 2015-08-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural Basis of Proline-Proline Peptide Bond Specificity of the Metalloprotease Zmp1 Implicated in Motility of Clostridium Difficile. Structure, 23, 2015
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3MG0
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![BU of 3mg0 by Molmil](/molmil-images/mine/3mg0) | Structure of yeast 20S proteasome with bortezomib | 分子名称: | N-[(1R)-1-(DIHYDROXYBORYL)-3-METHYLBUTYL]-N-(PYRAZIN-2-YLCARBONYL)-L-PHENYLALANINAMIDE, Proteasome component C1, Proteasome component C11, ... | 著者 | Sintchak, M.D. | 登録日 | 2010-04-05 | 公開日 | 2011-05-18 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.68 Å) | 主引用文献 | Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S beta5-subunit. Biochem.J., 430, 2010
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3MG4
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![BU of 3mg4 by Molmil](/molmil-images/mine/3mg4) | Structure of yeast 20S proteasome with Compound 1 | 分子名称: | (2S)-2-amino-N-[(1S)-1-({(1S)-1-[(4-methylbenzyl)carbamoyl]-3-phenylpropyl}carbamoyl)-3-phenylpropyl]-4-phenylbutanamide, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, MAGNESIUM ION, ... | 著者 | Sintchak, M.D. | 登録日 | 2010-04-05 | 公開日 | 2011-04-27 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.11 Å) | 主引用文献 | Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S beta5-subunit. Biochem.J., 430, 2010
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