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PDB: 274 件

5CB4
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Crystal structure of T2R-TTL-Tivantinib complex
分子名称: (3R,4R)-3-(5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl)-4-(1H-indol-3-yl)pyrrolidine-2,5-dione, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Wang, Y, Yu, Y, Chen, Q, Yang, J.
登録日2015-06-30
公開日2015-11-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.193 Å)
主引用文献Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283, 2016
5BMV
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CRYSTAL STRUCTURE OF TUBULIN-STATHMIN-TTL-Vinblastine COMPLEX
分子名称: (2ALPHA,2'BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLASTINE, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
著者Wang, Y, Chen, Q, Zhang, R.
登録日2015-05-23
公開日2016-07-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Insights into the Pharmacophore of Vinca Domain Inhibitors of Microtubules.
Mol.Pharmacol., 89, 2016
5GT9
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The X-ray structure of 7beta-hydroxysteroid dehydrogenase
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Oxidoreductase, short chain dehydrogenase/reductase family protein
著者Wang, F, Wang, R, Lv, Z, Chen, Q, Huo, X.
登録日2016-08-19
公開日2017-05-17
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of NADP(+)-bound 7 beta-hydroxysteroid dehydrogenase reveals two cofactor-binding modes
Acta Crystallogr F Struct Biol Commun, 73, 2017
1NT2
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CRYSTAL STRUCTURE OF FIBRILLARIN/NOP5P COMPLEX
分子名称: Fibrillarin-like pre-rRNA processing protein, S-ADENOSYLMETHIONINE, conserved hypothetical protein
著者Aittaleb, M, Rashid, R, Chen, Q, Palmer, J.R, Daniels, C.J, Li, H.
登録日2003-01-28
公開日2003-04-01
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structure and function of archaeal box C/D sRNP core proteins.
Nat.Struct.Biol., 10, 2003
6EC3
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Crystal Structure of EvdMO1
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Methyltransferase domain-containing protein, NICKEL (II) ION
著者McCulloch, K.M, Iverson, T.M, Starbird, C.A, Perry, N.A, Chen, Q, Berndt, S, Yamakawa, I, Loukachevitch, L.V.
登録日2018-08-07
公開日2018-12-26
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (3.35 Å)
主引用文献The Structure of the Bifunctional Everninomicin Biosynthetic Enzyme EvdMO1 Suggests Independent Activity of the Fused Methyltransferase-Oxidase Domains.
Biochemistry, 57, 2018
5E1J
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Structure of voltage-gated two-pore channel TPC1 from Arabidopsis thaliana
分子名称: BARIUM ION, CALCIUM ION, Two pore calcium channel protein 1
著者Guo, J, Zeng, W, Chen, Q, Lee, C, Chen, L, Yang, Y, Jiang, Y.
登録日2015-09-29
公開日2015-12-16
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.308 Å)
主引用文献Structure of the voltage-gated two-pore channel TPC1 from Arabidopsis thaliana.
Nature, 531, 2016
4B02
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The C-terminal Priming Domain is Strongly Associated with the Main Body of Bacteriophage phi6 RNA-Dependent RNA Polymerase
分子名称: MANGANESE (II) ION, RNA-DIRECTED RNA POLYMERASE
著者Sarin, L.P, Wright, S, Chen, Q, Degerth, L.H, Stuart, D.I, Grimes, J.M, Bamford, D.H, Poranen, M.M.
登録日2012-06-27
公開日2012-08-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献The C-Terminal Priming Domain is Strongly Associated with the Main Body of Bacteriophage Phi6 RNA-Dependent RNA Polymerase.
Virology, 432, 2012
7RPM
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Structures of the Intracellular Domain and Transmembrane Domain of the Human alpha7 Nicotinic Acetylcholine Receptors
分子名称: Neuronal acetylcholine receptor subunit alpha-7
著者Bondarenko, V, Chen, Q, Tang, P.
登録日2021-08-03
公開日2022-01-19
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structures of highly flexible intracellular domain of human alpha 7 nicotinic acetylcholine receptor.
Nat Commun, 13, 2022
5EZY
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Crystal structure of T2R-TTL-taccalonolide AJ complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
著者Wang, Y, Yu, Y, Chen, Q, Yang, J.
登録日2015-11-27
公開日2017-01-11
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Mechanism of microtubule stabilization by taccalonolide AJ
Nat Commun, 8, 2017
6KYB
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Crystal structure of Atg18 from Saccharomyces cerevisiae
分子名称: Autophagy-related protein 18
著者Tang, D, Lei, Y, Liao, G, Chen, Q, Xu, L, Lu, K, Qi, S.
登録日2019-09-17
公開日2020-09-09
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The crystal structure of Atg18 reveals a new binding site for Atg2 in Saccharomyces cerevisiae.
Cell.Mol.Life Sci., 78, 2021
6KYQ
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Crystal structure of DCLK1 Autoinhibited Kinase Domain
分子名称: BETA-MERCAPTOETHANOL, Serine/threonine-protein kinase DCLK1
著者Yu, Y, Chen, Q.
登録日2019-09-20
公開日2020-09-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.141 Å)
主引用文献DCLK1 Autoinhibition and Activation in Tumorigenesis
Innovation (N Y), 2021
6KYR
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Crystal structure of DCLK1 mutant (P675L) Autoinhibited Kinase Domain
分子名称: BETA-MERCAPTOETHANOL, Serine/threonine-protein kinase DCLK1
著者Yu, Y, Chen, Q.
登録日2019-09-20
公開日2020-09-23
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.206 Å)
主引用文献DCLK1 Autoinhibition and Activation in Tumorigenesis
Innovation (N Y), 2021
4XBK
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2-deoxyribose-5-phosphate aldolase from Lactobacillus brevis
分子名称: ACETIC ACID, Deoxyribose-phosphate aldolase
著者Jiao, X.-C, Pan, J, Xu, G.-C, Kong, X.-D, Chen, Q, Zhang, Z.-J, Xu, J.-H.
登録日2014-12-17
公開日2015-11-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.951 Å)
主引用文献Efficient synthesis of a statin precursor in high space-time yield by a new aldehyde-tolerant aldolase identified from Lactobacillus brevis
Catalysis Science And Technology, 5, 2015
8F4V
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Alpha7 nicotinic acetylcholine receptor intracellular and transmembrane domains bound to ivermectin in a desensitized state
分子名称: (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, Neuronal acetylcholine receptor subunit alpha-7
著者Bondarenko, V, Chen, Q, Tang, P.
登録日2022-11-11
公開日2023-02-22
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Elucidation of Ivermectin Binding to alpha 7nAChR and the Induced Channel Desensitization.
Acs Chem Neurosci, 14, 2023
4XBS
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2-deoxyribose-5-phosphate aldolase mutant - E78K
分子名称: Deoxyribose-phosphate aldolase
著者Jiao, X.-C, Pan, J, Xu, G.-C, Kong, X.-D, Chen, Q, Zhang, Z.-J, Xu, J.-H.
登録日2014-12-17
公開日2015-11-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Efficient synthesis of a statin precursor in high space-time yield by a new aldehyde-tolerant aldolase identified from Lactobacillus brevis
Catalysis Science And Technology, 5, 2015
4J0I
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Tannin acyl hydrolase in complex with 3,4-dihydroxybenzoate
分子名称: 3,4-DIHYDROXYBENZOIC ACID, DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-30
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0J
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Tannin acyl hydrolase in complex with ethyl 3,5-dihydroxybenzoate
分子名称: Tannase, ethyl 3,5-dihydroxybenzoate
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-31
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0G
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Tannin acyl hydrolase (mercury derivative)
分子名称: DI(HYDROXYETHYL)ETHER, MERCURY (II) ION, PENTAETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-30
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0C
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tannin acyl hydrolase from Lactobacillus plantarum (native structure)
分子名称: DI(HYDROXYETHYL)ETHER, PENTAETHYLENE GLYCOL, Tannase
著者Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-30
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0D
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tannin acyl hydrolase from Lactobacillus plantarum (Cadmium)
分子名称: CADMIUM ION, DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-30
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0H
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Tannin acyl hydrolase in complex with gallic acid
分子名称: 3,4,5-trihydroxybenzoic acid, DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-30
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4JUI
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crystal structure of tannase from from Lactobacillus plantarum
分子名称: DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, TRIETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, McKinstry, W.J, Chen, Q.
登録日2013-03-24
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
4J0K
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Tannin acyl hydrolase in complex with ethyl gallate
分子名称: DI(HYDROXYETHYL)ETHER, TETRAETHYLENE GLYCOL, TRIETHYLENE GLYCOL, ...
著者Ren, B, Wu, M, Wang, Q, Peng, X, Wen, H, Chen, Q, McKinstry, W.J.
登録日2013-01-31
公開日2013-05-22
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structure of tannase from Lactobacillus plantarum.
J.Mol.Biol., 425, 2013
5T38
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Crystal Structure of the N-terminal domain of EvdMO1 with SAH bound
分子名称: EvdMO1, S-ADENOSYL-L-HOMOCYSTEINE
著者McCulloch, K.M, Berndt, S, Yamakawa, I, Chen, Q, Loukachevitch, L.V, Starbird, C, Perry, N.A, Iverson, T.M.
登録日2016-08-25
公開日2017-09-06
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.1502 Å)
主引用文献The Structure of the Bifunctional Everninomicin Biosynthetic Enzyme EvdMO1 Suggests Independent Activity of the Fused Methyltransferase-Oxidase Domains.
Biochemistry, 57, 2018
5T39
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Crystal Structure of the N-terminal domain of EvdMO1 in the presence of SAH and D-fucose
分子名称: EvdMO1, S-ADENOSYL-L-HOMOCYSTEINE
著者McCulloch, K.M, Starbird, C.A, Chen, Q, Perry, N.A, Berndt, S, Yamakawa, I, Loukachevitch, L.V, Iverson, T.M.
登録日2016-08-25
公開日2017-09-06
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.1004 Å)
主引用文献The Structure of the Bifunctional Everninomicin Biosynthetic Enzyme EvdMO1 Suggests Independent Activity of the Fused Methyltransferase-Oxidase Domains.
Biochemistry, 57, 2018

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