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5CB4

Crystal structure of T2R-TTL-Tivantinib complex

Summary for 5CB4
Entry DOI10.2210/pdb5cb4/pdb
Related5C8Y 5CA0 5CA1
DescriptorTubulin alpha, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, (3R,4R)-3-(5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl)-4-(1H-indol-3-yl)pyrrolidine-2,5-dione, ... (13 entities in total)
Functional Keywordsinhibitor, complex, tubulin, structural protein
Biological sourceRattus norvegicus (Rat)
More
Cellular locationGolgi apparatus : P63043
Total number of polymer chains6
Total formula weight264922.18
Authors
Wang, Y.,Yu, Y.,Chen, Q.,Yang, J. (deposition date: 2015-06-30, release date: 2015-11-04, Last modification date: 2024-03-20)
Primary citationWang, Y.,Zhang, H.,Gigant, B.,Yu, Y.,Wu, Y.,Chen, X.,Lai, Q.,Yang, Z.,Chen, Q.,Yang, J.
Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283:102-111, 2016
Cited by
PubMed: 26462166
DOI: 10.1111/febs.13555
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.193 Å)
Structure validation

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