6DH9
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5Z8U
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6DGO
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![BU of 6dgo by Molmil](/molmil-images/mine/6dgo) | Crystal Structure of Human PPARgamma Ligand Binding Domain in Complex with Troglitazone | 分子名称: | (5S)-5-[(4-{[(2R)-6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-2-yl]methoxy}phenyl)methyl]-1,3-thiazolidine-2,4-dione, Peroxisome proliferator-activated receptor gamma | 著者 | Shang, J, Kojetin, D.J. | 登録日 | 2018-05-17 | 公開日 | 2019-05-22 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Quantitative structural assessment of graded receptor agonism. Proc.Natl.Acad.Sci.USA, 116, 2019
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5T9P
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5ZY9
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![BU of 5zy9 by Molmil](/molmil-images/mine/5zy9) | Structural basis for a tRNA synthetase | 分子名称: | (1R,2R)-2-[(2S,4E,6E,8R,9S,11R,13S,15S,16S)-7-cyano-8,16-dihydroxy-9,11,13,15-tetramethyl-18-oxooxacyclooctadeca-4,6-dien-2-yl]cyclopentanecarboxylic acid, Threonyl-tRNA synthase, ZINC ION | 著者 | Zhang, J. | 登録日 | 2018-05-23 | 公開日 | 2019-06-12 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for inhibition of
translational functions on a tRNA synthetase To Be Published
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4RP9
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![BU of 4rp9 by Molmil](/molmil-images/mine/4rp9) | Bacterial vitamin C transporter UlaA/SgaT in C2 form | 分子名称: | ASCORBIC ACID, Ascorbate-specific permease IIC component UlaA, PENTAETHYLENE GLYCOL, ... | 著者 | Wang, J.W. | 登録日 | 2014-10-29 | 公開日 | 2015-03-04 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.651 Å) | 主引用文献 | Crystal structure of a phosphorylation-coupled vitamin C transporter. Nat.Struct.Mol.Biol., 22, 2015
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2KIX
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3AXD
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![BU of 3axd by Molmil](/molmil-images/mine/3axd) | The truncated Fibrobacter succinogenes 1,3-1,4-beta-D-glucanase V18Y/W203Y in apo-form | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Beta-glucanase, CALCIUM ION | 著者 | Huang, J.W, Cheng, Y.S, Ko, T.P, Lin, C.Y, Lai, H.L, Chen, C.C, Ma, Y, Huang, C.H, Zheng, Y, Liu, J.R, Guo, R.T. | 登録日 | 2011-04-03 | 公開日 | 2012-02-15 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Rational design to improve thermostability and specific activity of the truncated Fibrobacter succinogenes 1,3-1,4-beta-D-glucanase Appl.Microbiol.Biotechnol., 94, 2012
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2DLJ
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3SR9
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![BU of 3sr9 by Molmil](/molmil-images/mine/3sr9) | Crystal structure of mouse PTPsigma | 分子名称: | Receptor-type tyrosine-protein phosphatase S | 著者 | Wang, J, Hou, L, Li, J, Ding, J. | 登録日 | 2011-07-07 | 公開日 | 2012-05-30 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural insights into the homology and differences between mouse protein tyrosine phosphatase-sigma and human protein tyrosine phosphatase-sigma Acta Biochim.Biophys.Sin., 43, 2011
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2KJ1
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2KHY
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7YIC
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7CCP
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6IPP
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![BU of 6ipp by Molmil](/molmil-images/mine/6ipp) | Non-native ferritin 8-mer mutant-C90A/C102A/C130A/D144C | 分子名称: | FE (III) ION, Ferritin heavy chain | 著者 | Zang, J, Chen, H, Zhou, K, Zhao, G. | 登録日 | 2018-11-03 | 公開日 | 2019-03-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.699 Å) | 主引用文献 | Disulfide-mediated conversion of 8-mer bowl-like protein architecture into three different nanocages. Nat Commun, 10, 2019
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2KZL
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7CBZ
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![BU of 7cbz by Molmil](/molmil-images/mine/7cbz) | Crystal structure of T2R-TTL-A31 complex | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-[5-[4-[2-[4-(2-cyclopropylethanoyl)piperazin-1-yl]ethoxy]phenyl]pyridin-2-yl]-N-(phenylmethyl)ethanamide, CALCIUM ION, ... | 著者 | Yang, J.H, Yan, W. | 登録日 | 2020-06-15 | 公開日 | 2021-06-23 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Design, Synthesis, and Bioactivity Evaluation of Dual-Target Inhibitors of Tubulin and Src Kinase Guided by Crystal Structure. J.Med.Chem., 64, 2021
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5BP0
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![BU of 5bp0 by Molmil](/molmil-images/mine/5bp0) | X-ray crystal structure of Lymnaea stagnalis acetylcholine binding protein (Ls-AChBP) in complex with 5-Fluoronicotine (TI-4650) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 5-fluoronicotine, Acetylcholine-binding protein, ... | 著者 | Bobango, J, Sankaran, B, Park, J.F, Wu, J, Talley, T.T. | 登録日 | 2015-05-27 | 公開日 | 2015-06-24 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Comparisons of Binding Affinities for Neuronal Nicotinic Receptors (NNRs) and AChBPs To Be Published
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5BRX
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![BU of 5brx by Molmil](/molmil-images/mine/5brx) | X-ray crystal structure of Aplysia californica (Ac-AChBP) in complex with 2-pyridyl azatricyclo[3.3.1.13,7]decane; 2-pyridylazaadamantane; 2-Aza (TI-8480) | 分子名称: | (2R,3S,5R,7S)-2-(pyridin-3-yl)-1-azatricyclo[3.3.1.1~3,7~]decane, SULFATE ION, Soluble acetylcholine receptor, ... | 著者 | Bobango, J, Sankaran, B, Park, J.F, Wu, J, Talley, T.T. | 登録日 | 2015-06-01 | 公開日 | 2015-06-24 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Comparisons of Binding Affinities for Neuronal Nicotinic Receptors (NNRs) and AChBPs To Be Published
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6ADX
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![BU of 6adx by Molmil](/molmil-images/mine/6adx) | Crystal structure of the Zika virus NS3 helicase (ADP-Mn2+ complex, form 1) | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, Serine protease NS3 | 著者 | Fang, J, Lu, G, Gong, P. | 登録日 | 2018-08-02 | 公開日 | 2019-03-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.752 Å) | 主引用文献 | Crystallographic Snapshots of the Zika Virus NS3 Helicase Help Visualize the Reactant Water Replenishment. ACS Infect Dis, 5, 2019
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6ADY
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![BU of 6ady by Molmil](/molmil-images/mine/6ady) | Crystal structure of the Zika virus NS3 helicase (ADP-Mn2+ complex, form 2) | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MANGANESE (II) ION, Serine protease NS3 | 著者 | Fang, J, Lu, G, Gong, P. | 登録日 | 2018-08-02 | 公開日 | 2019-03-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystallographic Snapshots of the Zika Virus NS3 Helicase Help Visualize the Reactant Water Replenishment. ACS Infect Dis, 5, 2019
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7JMK
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1RE5
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![BU of 1re5 by Molmil](/molmil-images/mine/1re5) | Crystal structure of 3-carboxy-cis,cis-muconate lactonizing enzyme from Pseudomonas putida | 分子名称: | 2,3-DIHYDROXY-1,4-DITHIOBUTANE, 3-carboxy-cis,cis-muconate cycloisomerase, CITRIC ACID | 著者 | Yang, J, Wang, Y, Woolridge, E.M, Petsko, G.A, Kozarich, J.W, Ringe, D. | 登録日 | 2003-11-06 | 公開日 | 2004-06-08 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal Structure of 3-Carboxy-cis,cis-muconate Lactonizing Enzyme from Pseudomonas putida, a Fumarase Class II Type Cycloisomerase: Enzyme Evolution in Parallel Pathways. Biochemistry, 43, 2004
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5BW2
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![BU of 5bw2 by Molmil](/molmil-images/mine/5bw2) | X-ray crystal structure of Aplysia californica acetylcholine binding protein (Ac-AChBP) Y55W in complex with 2-Pyridin-3-yl-1-aza-bicyclo[2.2.2]octane; 2-(3-pyridyl)quinuclidine; 2-PQ (TI-4699) | 分子名称: | (2R)-2-(pyridin-3-yl)-1-azabicyclo[2.2.2]octane, Soluble acetylcholine receptor | 著者 | Bobango, J, Sankaran, B, Park, J.F, Wu, J, Talley, T.T. | 登録日 | 2015-06-05 | 公開日 | 2015-06-24 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Comparisons of Binding Affinities for Neuronal Nicotinic Receptors (NNRs) and AChBPs To Be Published
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4LL1
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![BU of 4ll1 by Molmil](/molmil-images/mine/4ll1) | The structure of the TRX and TXNIP complex | 分子名称: | Thioredoxin, Thioredoxin-interacting protein | 著者 | Hwang, J, Kim, M.H. | 登録日 | 2013-07-09 | 公開日 | 2014-02-05 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The structural basis for the negative regulation of thioredoxin by thioredoxin-interacting protein Nat Commun, 5, 2014
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