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PDB: 60 件

7KPL
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Crystal structure of hEphB1 in apo form
分子名称: Ephrin type-B receptor 1
著者Ahmed, M, Wang, P, Sadek, H.
登録日2020-11-11
公開日2021-03-10
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.705 Å)
主引用文献Identification of tetracycline combinations as EphB1 tyrosine kinase inhibitors for treatment of neuropathic pain.
Proc.Natl.Acad.Sci.USA, 118, 2021
7KPM
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Crystal structure of hEphB1 bound with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Ephrin type-B receptor 1
著者Ahmed, M, Wang, P, Sadek, H.
登録日2020-11-11
公開日2021-03-10
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.608 Å)
主引用文献Identification of tetracycline combinations as EphB1 tyrosine kinase inhibitors for treatment of neuropathic pain.
Proc.Natl.Acad.Sci.USA, 118, 2021
6UMW
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BU of 6umw by Molmil
Crystal structure of hEphB1 bound with chlortetracycline
分子名称: 7-CHLOROTETRACYCLINE, Ephrin type-B receptor 1
著者Ahmed, M, Wang, P, Sadek, H.
登録日2019-10-10
公開日2020-10-14
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.982 Å)
主引用文献Identification of tetracycline combinations as EphB1 tyrosine kinase inhibitors for treatment of neuropathic pain.
Proc.Natl.Acad.Sci.USA, 118, 2021
3VFG
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Crystal structure of monoclonal antibody 3F8 Fab fragment that binds to GD2 ganglioside
分子名称: 3F8 Heavy Chain, 3F8 Light Chain
著者Ahmed, M, Goldgur, Y, Cheung, N.-K.
登録日2012-01-09
公開日2013-02-06
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献In silico Driven Redesign of a Clinically Relevant Antibody for the Treatment of GD2 Positive Tumors.
Plos One, 8, 2013
5CMA
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Anti-B7-H3 monoclonal antibody ch8H9 Fab fragment
分子名称: Antibody ch8H9 Fab heavy chain, Antibody ch8H9 Fab light chain
著者Ahmed, M, Goldgur, Y, Cheng, M, Cheung, N.K.
登録日2015-07-16
公開日2015-10-28
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Humanized Affinity-matured Monoclonal Antibody 8H9 Has Potent Antitumor Activity and Binds to FG Loop of Tumor Antigen B7-H3.
J.Biol.Chem., 290, 2015
4U13
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Crystal structure of putative polyketide cyclase (protein SMa1630) from Sinorhizobium meliloti at 2.3 A resolution
分子名称: putative polyketide cyclase SMa1630
著者Shabalin, I.G, Bacal, P, Osinski, T, Cooper, D.R, Szlachta, K, Stead, M, Grabowski, M, Hammonds, J, Ahmed, M, Hillerich, B.S, Bonanno, J, Seidel, R, Almo, S.C, Minor, W, New York Structural Genomics Research Consortium (NYSGRC)
登録日2014-07-14
公開日2014-09-10
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of a putative polyketide cyclase (protein SMa1630) from Sinorhizobium meliloti at 2.3 A resolution
to be published
4UC0
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Crystal Structure Of a purine nucleoside phosphorylase (PSI-NYSGRC-029736) from Agrobacterium vitis
分子名称: HYPOXANTHINE, Purine nucleoside phosphorylase
著者Cameron, S.A, Sampathkumar, P, Ramagopal, U.A, Attonito, J, Ahmed, M, Bhosle, R, Bonanno, J, Chamala, S, Chowdhury, S, Glenn, A.S, Hammonds, J, Hillerich, B, Love, J.D, Seidel, R, Stead, M, Toro, R, Wasserman, S.R, Schramm, V.L, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC)
登録日2014-08-13
公開日2014-10-08
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure Of a purine nucleoside phosphorylase (PSI-NYSGRC-029736) from Agrobacterium vitis
To be published
7ATS
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The LIMK1 Kinase Domain Bound To LIJTF500127
分子名称: LIM domain kinase 1, N-[3-[5-(4-Chlorophenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamide
著者Mathea, S, Chatterjee, D, Preuss, F, Yamamoto, S, Tawada, M, Nomura, I, Takagi, T, Ahmed, M, Little, W, Mueller-Knapp, S, Knapp, S.
登録日2020-10-30
公開日2020-11-25
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The LIMK1 Kinase Domain Bound To LIJTF500127
To Be Published
7ATU
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The LIMK1 Kinase Domain Bound To LIJTF500025
分子名称: (S)-2-benzyl-6-(8-chloro-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-7-oxo-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-c]pyridine-3-carboxamide, LIM domain kinase 1
著者Mathea, S, Chatterjee, D, Preuss, F, Yamamoto, S, Tawada, M, Nomura, I, Takagi, T, Ahmed, M, Little, W, Mueller-Knapp, S, Knapp, S.
登録日2020-10-30
公開日2020-12-23
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The LIMK1 Kinase Domain Bound To LIJTF500025
To Be Published
4WCZ
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Crystal structure of a putative enoyl-CoA hydratase/isomerase from Novosphingobium aromaticivorans
分子名称: Enoyl-CoA hydratase/isomerase
著者Tkaczuk, K.L, Cooper, D.R, Chapman, H.C, Niedzialkowska, E, Cymborowski, M.T, Hillerich, B.S, Stead, M, Ahmed, M, Hammonds, J, Bonanno, J, Seidel, R, Almo, S.C, Minor, W, New York Structural Genomics Research Consortium (NYSGRC)
登録日2014-09-05
公開日2014-12-03
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Crystal structure of a putative enoyl-CoA hydratase/isomerase from Novosphingobium aromaticivorans
to be published
2BBR
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Crystal Structure of MC159 Reveals Molecular Mechanism of DISC Assembly and vFLIP Inhibition
分子名称: AZIDE ION, Viral CASP8 and FADD-like apoptosis regulator
著者Yang, J.K, Wang, L, Zheng, L, Wan, F, Ahmed, M, Lenardo, M.J, Wu, H.
登録日2005-10-17
公開日2006-02-14
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Crystal structure of MC159 reveals molecular mechanism of DISC assembly and FLIP inhibition.
Mol.Cell, 20, 2005
2BBZ
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Crystal Structure of MC159 Reveals Molecular Mechanism of DISC Assembly and vFLIP Inhibition
分子名称: Viral CASP8 and FADD-like apoptosis regulator
著者Yang, J.K, Wang, L, Zheng, L, Wan, F, Ahmed, M, Lenardo, M.J, Wu, H.
登録日2005-10-18
公開日2006-02-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Crystal structure of MC159 reveals molecular mechanism of DISC assembly and FLIP inhibition.
Mol.Cell, 20, 2005
5M1U
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Solution structure of CsgF in DHPC micelles
分子名称: Curli production assembly/transport component CsgF
著者Spehr, J, Schubeis, T, Ahmed, M, Ritter, C.
登録日2016-10-10
公開日2017-10-11
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structural and functional characterization of the Curli adaptor protein CsgF.
FEBS Lett., 592, 2018
8FMP
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BU of 8fmp by Molmil
Complex structure of K210 deletion Troponin complex with pamidronate
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.24 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMT
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BU of 8fmt by Molmil
Complex structure of TnnT-R205L Troponin complex
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMM
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Complex structure of wild type Troponin complex
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-23
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.112 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMQ
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BU of 8fmq by Molmil
Complex structure of K210 deletion Troponin complex with alendronate
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.248 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMN
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BU of 8fmn by Molmil
Complex structure of K210 deletion Troponin complex
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-23
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.101 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMO
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Complex structure of K210 deletion Troponin complex with risedronate
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (2.612 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMS
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BU of 8fms by Molmil
Complex structure of K210 deletion Troponin complex with neridronate
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.435 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
8FMR
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BU of 8fmr by Molmil
Complex structure of K210 deletion Troponin complex with ibandronate
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles, ...
著者Wang, P, Ahmed, M, Sadek, H.
登録日2022-12-24
公開日2024-01-31
実験手法X-RAY DIFFRACTION (3.238 Å)
主引用文献Structural and Phenotypic Correction of K210del Genetic Cardiomyopathy by an FDA Approved drug
To Be Published
2M4M
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BU of 2m4m by Molmil
Solution structure of the RRM domain of the hypothetical protein CAGL0M09691g from Candida glabrata
分子名称: hypothetical protein
著者Harris, R, Hillerich, B, Ahmed, M, Bonanno, J.B, Chamala, S, Evans, B, Lafleur, J, Hammonds, J, Washington, E, Stead, M, Love, J, Attonito, J, Patel, H, Seidel, R.D, Chook, Y.M, Rout, M.P, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC), Nucleocytoplasmic Transport: a Target for Cellular Control (NPCXstals)
登録日2013-02-07
公開日2013-02-27
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structure of the RRM domain of the hypothetical protein CAGL0M09691g from Candida glabrata
To be Published
2M72
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Solution structure of uncharacterized thioredoxin-like protein PG_2175 from Porphyromonas gingivalis
分子名称: Uncharacterized thioredoxin-like protein
著者Harris, R, Ahmed, M, Attonito, J, Bonanno, J.B, Chamala, S, Chowdhury, S, Evans, B, Fiser, A, Glenn, A.S, Hammonds, J, Hillerich, B, Khafizov, K, Lafleur, J, Love, J.D, Seidel, R.D, Stead, M, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC)
登録日2013-04-16
公開日2013-05-15
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structure of uncharacterized thioredoxin-like protein PG_2175 from Porphyromonas gingivalis
To be Published
2M71
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Solution structure of the a C-terminal domain of translation initiation factor IF-3 from Campylobacter jejuni
分子名称: Translation initiation factor IF-3
著者Harris, R, Ahmed, M, Attonito, J, Bonanno, J.B, Chamala, S, Chowdhury, S, Evans, B, Fiser, A, Glenn, A.S, Hammonds, J, Hillerich, B, Khafizov, K, Lafleur, J, Love, J.D, Seidel, R.D, Stead, M, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC)
登録日2013-04-16
公開日2013-05-15
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structure of the a C-terminal domain of translation initiation factor IF-3 from Campylobacter jejuni
To be Published
2M4N
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Solution structure of the putative Ras interaction domain of AFD-1, isoform a from Caenorhabditis elegans
分子名称: Protein AFD-1, isoform a
著者Harris, R, Hillerich, B, Ahmed, M, Bonanno, J.B, Chamala, S, Evans, B, Lafleur, J, Hammonds, J, Washington, E, Stead, M, Love, J, Attonito, J, Seidel, R.D, Liddington, R.C, Weis, W.I, Nelson, W.J, Girvin, M.E, Almo, S.C, New York Structural Genomics Research Consortium (NYSGRC), Assembly, Dynamics and Evolution of Cell-Cell and Cell-Matrix Adhesions (CELLMAT)
登録日2013-02-07
公開日2013-03-20
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Solution structure of the putative Ras interaction domain of AFD-1, isoform a from Caenorhabditis elegans
To be Published

 

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