7ATS
The LIMK1 Kinase Domain Bound To LIJTF500127
Summary for 7ATS
Entry DOI | 10.2210/pdb7ats/pdb |
Descriptor | LIM domain kinase 1, N-[3-[5-(4-Chlorophenyl)-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamide (2 entities in total) |
Functional Keywords | kinase inhibitor active site cfl1 actin cytoskeleton, signaling protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 36518.71 |
Authors | Mathea, S.,Chatterjee, D.,Preuss, F.,Yamamoto, S.,Tawada, M.,Nomura, I.,Takagi, T.,Ahmed, M.,Little, W.,Mueller-Knapp, S.,Knapp, S. (deposition date: 2020-10-30, release date: 2020-11-25, Last modification date: 2024-01-31) |
Primary citation | Mathea, S.,Chatterjee, D.,Preuss, F.,Yamamoto, S.,Tawada, M.,Nomura, I.,Takagi, T.,Ahmed, M.,Little, W.,Mueller-Knapp, S.,Knapp, S. The LIMK1 Kinase Domain Bound To LIJTF500127 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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