7DVK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7dvk by Molmil](/molmil-images/mine/7dvk) | |
7DVI
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7dvi by Molmil](/molmil-images/mine/7dvi) | |
6K26
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6k26 by Molmil](/molmil-images/mine/6k26) | |
6KSG
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6ksg by Molmil](/molmil-images/mine/6ksg) | Vibrio cholerae Methionine Aminopeptidase in holo form | 分子名称: | GLYCEROL, Methionine aminopeptidase, NICKEL (II) ION, ... | 著者 | Pillalamarri, V, Addlagatta, A. | 登録日 | 2019-08-23 | 公開日 | 2020-08-26 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Methionine aminopeptidases with short sequence inserts within the catalytic domain are differentially inhibited: Structural and biochemical studies of three proteins from Vibrio spp. Eur.J.Med.Chem., 209, 2020
|
|
6LH7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6lh7 by Molmil](/molmil-images/mine/6lh7) | |
6LZB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6lzb by Molmil](/molmil-images/mine/6lzb) | crystal structure of Human Methionine aminopeptidase (HsMetAP1b) in complex with AN-P2-5H-06 | 分子名称: | 1-[(3-methoxyphenyl)methyl]-~{N}-oxidanyl-pyrrolo[2,3-b]pyridine-5-carboxamide, COBALT (II) ION, GLYCEROL, ... | 著者 | sandeep, C.B, Addlagatta, A. | 登録日 | 2020-02-18 | 公開日 | 2021-02-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Selective inhibition of Helicobacter pylori methionine aminopeptidase by azaindole hydroxamic acid derivatives: Design, synthesis, in vitro biochemical and structural studies. Bioorg.Chem., 115, 2021
|
|
6LZC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6lzc by Molmil](/molmil-images/mine/6lzc) | crystal structure of Human Methionine aminopeptidase (HsMetAP1b) in complex with KV-P2-4H-05 | 分子名称: | COBALT (II) ION, GLYCEROL, MAGNESIUM ION, ... | 著者 | Sandeep, C.B, Addlagatta, A. | 登録日 | 2020-02-18 | 公開日 | 2021-02-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Selective inhibition of Helicobacter pylori methionine aminopeptidase by azaindole hydroxamic acid derivatives: Design, synthesis, in vitro biochemical and structural studies. Bioorg.Chem., 115, 2021
|
|
4Q4I
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4q4i by Molmil](/molmil-images/mine/4q4i) | Crystal structure of E.coli aminopeptidase N in complex with amastatin | 分子名称: | Amastatin, Aminopeptidase N, GLYCEROL, ... | 著者 | Reddi, R, Ganji, R.J, Addlagatta, A. | 登録日 | 2014-04-14 | 公開日 | 2015-04-15 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Structural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: Crystal structure in complex with E. coli aminopeptidase N. Protein Sci., 24, 2015
|
|
4OOK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4ook by Molmil](/molmil-images/mine/4ook) | |
4Q4E
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4q4e by Molmil](/molmil-images/mine/4q4e) | Crystal structure of E.coli aminopeptidase N in complex with actinonin | 分子名称: | ACTINONIN, Aminopeptidase N, GLYCEROL, ... | 著者 | Reddi, R, Ganji, R.J, Addlagatta, A. | 登録日 | 2014-04-14 | 公開日 | 2015-04-15 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: Crystal structure in complex with E. coli aminopeptidase N. Protein Sci., 24, 2015
|
|
3ROR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3ror by Molmil](/molmil-images/mine/3ror) | |
6M00
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6m00 by Molmil](/molmil-images/mine/6m00) | |
4U6W
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u6w by Molmil](/molmil-images/mine/4u6w) | |
4U71
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u71 by Molmil](/molmil-images/mine/4u71) | |
4U75
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u75 by Molmil](/molmil-images/mine/4u75) | HsMetAP (F309M) in complex with Methionine | 分子名称: | COBALT (II) ION, GLYCEROL, METHIONINE, ... | 著者 | Arya, T, Addlagatta, A. | 登録日 | 2014-07-30 | 公開日 | 2015-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Identification of the Molecular Basis of Inhibitor Selectivity between the Human and Streptococcal Type I Methionine Aminopeptidases J.Med.Chem., 58, 2015
|
|
4U6E
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u6e by Molmil](/molmil-images/mine/4u6e) | HsMetAP in complex with (amino(phenyl)methyl)phosphonic acid | 分子名称: | COBALT (II) ION, Methionine aminopeptidase 1, [(R)-amino(phenyl)methyl]phosphonic acid | 著者 | Arya, T, Addlagatta, A. | 登録日 | 2014-07-28 | 公開日 | 2015-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Identification of the Molecular Basis of Inhibitor Selectivity between the Human and Streptococcal Type I Methionine Aminopeptidases J.Med.Chem., 58, 2015
|
|
4U6Z
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u6z by Molmil](/molmil-images/mine/4u6z) | |
4U1B
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u1b by Molmil](/molmil-images/mine/4u1b) | |
4U6J
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u6j by Molmil](/molmil-images/mine/4u6j) | HsMetAP in complex with methionine | 分子名称: | COBALT (II) ION, GLYCEROL, METHIONINE, ... | 著者 | Arya, T, Addlagatta, A. | 登録日 | 2014-07-29 | 公開日 | 2015-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Identification of the Molecular Basis of Inhibitor Selectivity between the Human and Streptococcal Type I Methionine Aminopeptidases J.Med.Chem., 58, 2015
|
|
4U6C
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u6c by Molmil](/molmil-images/mine/4u6c) | |
4U69
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u69 by Molmil](/molmil-images/mine/4u69) | |
4U70
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u70 by Molmil](/molmil-images/mine/4u70) | |
4U76
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u76 by Molmil](/molmil-images/mine/4u76) | HsMetAP (F309M) holo form | 分子名称: | COBALT (II) ION, GLYCEROL, Methionine aminopeptidase 1, ... | 著者 | Arya, T, Addlagatta, A. | 登録日 | 2014-07-30 | 公開日 | 2015-03-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Identification of the Molecular Basis of Inhibitor Selectivity between the Human and Streptococcal Type I Methionine Aminopeptidases J.Med.Chem., 58, 2015
|
|
4U73
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4u73 by Molmil](/molmil-images/mine/4u73) | |
5ZI7
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5zi7 by Molmil](/molmil-images/mine/5zi7) | |