7ZC8
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![BU of 7zc8 by Molmil](/molmil-images/mine/7zc8) | |
8P6K
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![BU of 8p6k by Molmil](/molmil-images/mine/8p6k) | |
8P6J
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![BU of 8p6j by Molmil](/molmil-images/mine/8p6j) | |
7Q9Q
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![BU of 7q9q by Molmil](/molmil-images/mine/7q9q) | |
7Q9U
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![BU of 7q9u by Molmil](/molmil-images/mine/7q9u) | |
7Q9S
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![BU of 7q9s by Molmil](/molmil-images/mine/7q9s) | Crystal structure of PDE6D KRas peptide complex with Compound-1 | Descriptor: | 1,2-ETHANEDIOL, 2-methyl-3-(1~{H}-pyrazol-5-yl)imidazo[1,2-a]pyridine, DIMETHYL SULFOXIDE, ... | Authors: | Yelland, T, Ismail, S. | Deposit date: | 2021-11-14 | Release date: | 2022-01-19 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
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7Q9R
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![BU of 7q9r by Molmil](/molmil-images/mine/7q9r) | Cocrystal structure of PDE6D bound to NRAS peptide | Descriptor: | 1,2-ETHANEDIOL, FARNESYL, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta, ... | Authors: | Yelland, T, Ismail, S. | Deposit date: | 2021-11-14 | Release date: | 2022-01-19 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
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7QJK
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![BU of 7qjk by Molmil](/molmil-images/mine/7qjk) | Crystal structure of PDE6D in complex with Compound-2 | Descriptor: | 1,2-ETHANEDIOL, N-(phenylmethyl)pyridin-2-amine, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta, ... | Authors: | Yelland, T, Ismail, S. | Deposit date: | 2021-12-16 | Release date: | 2022-01-26 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (3.1 Å) | Cite: | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
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7QF9
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![BU of 7qf9 by Molmil](/molmil-images/mine/7qf9) | Crystal structure of PDE6D bound to HRas peptide | Descriptor: | 1,2-ETHANEDIOL, FARNESYL, HRas peptide, ... | Authors: | Yelland, T, Ismail, I. | Deposit date: | 2021-12-05 | Release date: | 2022-02-09 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Stabilization of the RAS:PDE6D Complex Is a Novel Strategy to Inhibit RAS Signaling. J.Med.Chem., 65, 2022
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