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4HKE
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BU of 4hke by Molmil
Crystal Structure of MoxT of Bacillus anthracis
分子名称: Addiction module toxin component PemK, SULFATE ION
著者Verma, S, Kumar, S, Gourinath, S, Bhatnagar, R.
登録日2012-10-15
公開日2013-11-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Structural basis of Bacillus anthracis MoxXT disruption and the modulation of MoxT ribonuclease activity by rationally designed peptides.
J.Biomol.Struct.Dyn., 33, 2015
7FC7
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BU of 7fc7 by Molmil
Acyl-Coenzyme A Binding Protein 96 (LMJ_17_0780) of Leishmania Major in complex with Coenzyme A
分子名称: ACB domain-containing protein, COENZYME A
著者Verma, S, Makde, R.D, Sundd, M.
登録日2021-07-14
公開日2023-01-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Acyl-Coenzyme A Binding Protein 96 (LMJ_17_0780) of Leishmania Major in complex with Coenzyme A
To be published
7WFS
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BU of 7wfs by Molmil
Acyl-Coenzyme A Binding Protein 103 (LMJF_17_0620) of Leishmania major in triclinic crystal form
分子名称: ACB domain-containing protein
著者Verma, S, Sundd, M.
登録日2021-12-27
公開日2023-02-01
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Acyl-Coenzyme A Binding Protein 103 (LMJF_17_0620) of Leishmania major in monoclinic crystal form
TO BE PUBLISHED
7DES
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BU of 7des by Molmil
Acyl-Coenzyme A Binding Protein 103 (LMJF_17_0620) of Leishmania Major
分子名称: ACB domain-containing protein, FORMIC ACID
著者Verma, S, Sundd, M, Makde, R.D.
登録日2020-11-04
公開日2022-05-04
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Acyl-Coenzyme A Binding Protein 103 (LMJF_17_0620) of Leishmania Major
To Be Published
4LOO
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BU of 4loo by Molmil
Structural basis of autoactivation of p38 alpha induced by TAB1 (Monoclinic crystal form)
分子名称: 4-(4-FLUOROPHENYL)-1-(4-PIPERIDINYL)-5-(2-AMINO-4-PYRIMIDINYL)-IMIDAZOLE, Mitogen-activated protein kinase 14, TGF-beta-activated kinase 1 and MAP3K7-binding protein 1
著者Chaikuad, A, DeNicola, G.F, Krojer, T, Allerston, C.K, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Marber, M.S, Knapp, S, Structural Genomics Consortium (SGC)
登録日2013-07-13
公開日2013-08-21
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Mechanism and consequence of the autoactivation of p38 alpha mitogen-activated protein kinase promoted by TAB1.
Nat.Struct.Mol.Biol., 20, 2013
4LOQ
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BU of 4loq by Molmil
Structural basis of autoactivation of p38 alpha induced by TAB1 (Tetragonal crystal form with bound sulphate)
分子名称: 1,2-ETHANEDIOL, 4-(4-FLUOROPHENYL)-1-(4-PIPERIDINYL)-5-(2-AMINO-4-PYRIMIDINYL)-IMIDAZOLE, Mitogen-activated protein kinase 14, ...
著者Chaikuad, A, DeNicola, G.F, Yue, W.W, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Marber, M.S, Knapp, S, Structural Genomics Consortium (SGC)
登録日2013-07-13
公開日2013-08-21
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.319 Å)
主引用文献Mechanism and consequence of the autoactivation of p38 alpha mitogen-activated protein kinase promoted by TAB1.
Nat.Struct.Mol.Biol., 20, 2013
4LOP
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BU of 4lop by Molmil
Structural basis of autoactivation of p38 alpha induced by TAB1 (Tetragonal crystal form)
分子名称: 1,2-ETHANEDIOL, 4-(4-FLUOROPHENYL)-1-(4-PIPERIDINYL)-5-(2-AMINO-4-PYRIMIDINYL)-IMIDAZOLE, L(+)-TARTARIC ACID, ...
著者Chaikuad, A, DeNicola, G.F, Krojer, T, Allerston, C.K, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Marber, M.S, Knapp, S, Structural Genomics Consortium (SGC)
登録日2013-07-13
公開日2013-08-21
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.049 Å)
主引用文献Mechanism and consequence of the autoactivation of p38 alpha mitogen-activated protein kinase promoted by TAB1.
Nat.Struct.Mol.Biol., 20, 2013
7DBS
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BU of 7dbs by Molmil
Crystal Structure Of Biotin Protein Ligase From Leishmania Major in complex with Biotin
分子名称: BIOTIN, Biotin/lipoate protein ligase-like protein
著者Rajak, M, Sundd, M.
登録日2020-10-21
公開日2021-04-14
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Leishmania major biotin protein ligase forms a unique cross-handshake dimer.
Acta Crystallogr D Struct Biol, 77, 2021
5W2P
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BU of 5w2p by Molmil
Crystal structure of Mycobacterium tuberculosis KasA in complex with 6U5
分子名称: 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, GLYCEROL, ...
著者Capodagli, G.C, Neiditch, M.B.
登録日2017-06-06
公開日2018-12-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA.
MBio, 9, 2018
5W2Q
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BU of 5w2q by Molmil
Crystal structure of Mycobacterium tuberculosis KasA in complex with 6U5
分子名称: 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, GLYCEROL, ...
著者Capodagli, G.C, Neiditch, M.B.
登録日2017-06-06
公開日2018-12-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA.
MBio, 9, 2018
5W2O
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BU of 5w2o by Molmil
Crystal structure of Mycobacterium tuberculosis KasA
分子名称: 3,3',3''-phosphanetriyltripropanoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 1, CHLORIDE ION, ...
著者Capodagli, G.C, Neiditch, M.B.
登録日2017-06-06
公開日2018-12-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA.
MBio, 9, 2018
5W2S
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BU of 5w2s by Molmil
Crystal Structure of Mycobacterium Tuberculosis KasA in complex with KMG
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 1, GLYCEROL, ISOPROPYL ALCOHOL, ...
著者Capodagli, G.C, Neiditch, M.B.
登録日2017-06-06
公開日2018-12-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.399 Å)
主引用文献Synergistic Lethality of a Binary Inhibitor of Mycobacterium tuberculosis KasA.
MBio, 9, 2018
6JHU
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BU of 6jhu by Molmil
Crystal Structure Of Biotin Protein Ligase From Leishmania Major in complex with Biotinyl-5-AMP
分子名称: BIOTINYL-5-AMP, Biotin/lipoate protein ligase-like protein, SULFATE ION
著者Rajak, M, Patel, A, Sundd, M.
登録日2019-02-19
公開日2020-04-08
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Leishmania major biotin protein ligase forms a unique cross-handshake dimer
Acta Crystallogr.,Sect.D, 77, 2021
5NZZ
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BU of 5nzz by Molmil
Crystal structure of phosphorylated p38aMAPK in complex with TAB1
分子名称: MAGNESIUM ION, Mitogen-activated protein kinase 14, NICKEL (II) ION, ...
著者Nichols, C.E, De Nicola, G.F.
登録日2017-05-15
公開日2018-05-30
最終更新日2018-09-19
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The TAB1-p38 alpha complex aggravates myocardial injury and can be targeted by small molecules.
JCI Insight, 3, 2018
5O90
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BU of 5o90 by Molmil
Crystal structure of a P38alpha T185G mutant in complex with TAB1 peptide.
分子名称: 4-(4-FLUOROPHENYL)-1-(4-PIPERIDINYL)-5-(2-AMINO-4-PYRIMIDINYL)-IMIDAZOLE, Mitogen-activated protein kinase 14, TGF-beta-activated kinase 1 and MAP3K7-binding protein 1
著者Nichols, C.E, De Nicola, G.F, Thapa, D.
登録日2017-06-15
公開日2018-01-31
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献TAB1-Induced Autoactivation of p38 alpha Mitogen-Activated Protein Kinase Is Crucially Dependent on Threonine 185.
Mol. Cell. Biol., 38, 2018

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件を2024-04-24に公開中

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