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3TKG
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BU of 3tkg by Molmil
crystal structure of HIV model protease precursor/saquinavir complex
Descriptor: (2S)-N-[(2S,3R)-4-[(2S,3S,4aS,8aS)-3-(tert-butylcarbamoyl)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-hydroxy-1 -phenyl-butan-2-yl]-2-(quinolin-2-ylcarbonylamino)butanediamide, CHLORIDE ION, GLYCEROL, ...
Authors:Agniswamy, J, Sayer, J, Weber, I, Louis, J.
Deposit date:2011-08-26
Release date:2012-04-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.36 Å)
Cite:Terminal interface conformations modulate dimer stability prior to amino terminal autoprocessing of HIV-1 protease.
Biochemistry, 51, 2012
3TL9
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BU of 3tl9 by Molmil
crystal structure of HIV protease model precursor/Saquinavir complex
Descriptor: (2S)-N-[(2S,3R)-4-[(2S,3S,4aS,8aS)-3-(tert-butylcarbamoyl)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-hydroxy-1 -phenyl-butan-2-yl]-2-(quinolin-2-ylcarbonylamino)butanediamide, CHLORIDE ION, GLYCEROL, ...
Authors:Agniswamy, J, Sayer, J, Weber, I, Louis, J.
Deposit date:2011-08-29
Release date:2012-04-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.32 Å)
Cite:Terminal interface conformations modulate dimer stability prior to amino terminal autoprocessing of HIV-1 protease.
Biochemistry, 51, 2012
3TKW
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BU of 3tkw by Molmil
Crystal structure of HIV protease model precursor/Darunavir complex
Descriptor: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, CHLORIDE ION, GLYCEROL, ...
Authors:Agniswamy, J, Sayer, J, Weber, I, Louis, J.
Deposit date:2011-08-29
Release date:2012-04-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Terminal interface conformations modulate dimer stability prior to amino terminal autoprocessing of HIV-1 protease.
Biochemistry, 51, 2012

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