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Progesterone receptor ligand binding domain in complex with the nonsteroidal agonist tanaproget
Descriptor:	5-(4,4-DIMETHYL-2-THIOXO-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-6-YL)-1-METHYL-1H-PYRROLE-2-CARBONITRILE, Progesterone receptor, SULFATE ION
Authors:	Zhang, Z, Olland, A.M, Zhu, Y, Cohen, J, Berrodin, T, Chippari, S, Appavu, C, Li, S, Wilhem, J, Chopra, R, Fensome, A, Zhang, P, Wrobel, J, Unwalla, R.J, Lyttle, C.R, Winneker, R.C.
Deposit date:	2005-05-30
Release date:	2005-07-05
Last modified:	2023-08-23
Method:	X-RAY DIFFRACTION (2 Å)
Cite:	Molecular and pharmacological properties of a potent and selective novel nonsteroidal progesterone receptor agonist tanaproget J.Biol.Chem., 280, 2005

Crystal Structure Of The Androgen Receptor Ligand Binding Domain In Complex With 5-(2-fluoro-4-hydroxyphenyl)-1-methyl-1H-pyrrole-2-carbonitrile
Descriptor:	5-(2-fluoro-4-hydroxyphenyl)-1-methyl-1H-pyrrole-2-carbonitrile, Androgen receptor
Authors:	Parris, K, Unwalla, R.
Deposit date:	2017-05-02
Release date:	2018-03-14
Last modified:	2024-03-13
Method:	X-RAY DIFFRACTION (2.35 Å)
Cite:	Structure-Based Approach To Identify 5-[4-Hydroxyphenyl]pyrrole-2-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators. J. Med. Chem., 60, 2017